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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T0802 | Procaine hydrochloride | Novocaine HCl,Procaine HCl | Histone Demethylase , 5-HT Receptor , DNA/RNA Synthesis , Sodium Channel , NMDAR , AChR |
Procaine hydrochloride (Novocaine HCl) is the hydrochloride salt form of procaine, a benzoic acid derivative with local anesthetic and antiarrhythmic properties. Procaine binds to and inhibits voltage-gated sodiumchannel... | |||
T0029 | Procaine | Duracaine,Spinocaine,Novocaine,Vitamin H3 | Histone Demethylase , DNA/RNA Synthesis , Sodium Channel |
Procaine (Vitamin H3) is a local anesthetic of the ester type that has a slow onset and a short duration of action. It is mainly used for infiltration anesthesia, peripheral nerve block, and spinal block. | |||
T8598 | CHEMBL241987 | 2-PHENYL-2,5-DIHYDRO-4H-PYRAZOLO[3,4-C]QUINOLIN-4-ONE | Adenosine Receptor |
CHEMBL241987 targets the Adenosine receptor A3 (human) | |||
T19241 | Cloquintocet-mexyl | Others | |
Cloquintocet-mexyl, a herbicide, targets and controls coarse annual grasses within the Poaceae family. | |||
T8635 | CI 75300 | P2X Receptor | |
CI 75300 targets the P2X purinoceptor 7 (human). | |||
T19849L | 2-PADQZ hydrochloride | 2-PADQZ hydrochloride (60547-97-9 Free base) | Antiviral , Influenza Virus |
2-PADQZ hydrochloride shows antiviral activity and targets influenza A virus RNA promoter. | |||
T8912 | 5-ETHYL-4,5,6,7-TETRAHYDRO-THIAZOLO[5,4-C]PYRIDIN-2-YLAMINE | PLK | |
5-ETHYL-4,5,6,7-TETRAHYDRO-THIAZOLO[5,4-C]PYRIDIN-2-YLAMINE targets PLK1. | |||
T9061 | EN4 | EN4 MYC inhibitor | c-Myc |
EN4 (EN4 MYC inhibitor) MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC. It is selective for c-MYC over N-MYC and L-MYC, and inhibits MYC transcriptional activity, downregulates MYC targets, an... | |||
T8913 | 1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID | GRK | |
1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2. | |||
T9827 | Carfenazine | Dopamine Receptor | |
carfenazine targets the Dopamine receptor and is used for schizophrenia research. | |||
T8672 | 2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE | BisOPP-A | Thyroid hormone receptor(THR) |
2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE is targets the thyroid stimulating hormone receptor (human) | |||
TNU0436 | 2-Thiocytidine | Apoptosis , Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis | |
2-Thiocytidine is a purine nucleoside analog that targets malignant tumors of the inert lymphatic system and has a broad spectrum of antitumor activity.2-Thiocytidine induces apoptosis by inhibiting DNA synthesis.2-Thioc... | |||
T8584 | 6-Phenyldihydropyrimidine-2,4(1h,3h)-dione | 2,4(1H,3H)-Pyrimidinedione,dihydro-6-phenyl- | Others |
6-Phenyldihydropyrimidine-2,4(1h,3h)-dione targets the polypyrimidine tract-binding protein 1 isoform a (human) | |||
T10232 | Acetophenazine dimaleate | Dopamine Receptor | |
Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor. | |||
T6094 | MK-2461 | MK2461 | c-Met/HGFR |
MK-2461 is a novel inhibitor that targets multiple proteins and competitively binds to ATP sites, specifically inhibiting the activated c-Met protein with an average inhibitory concentration (IC50) of 2.5 nM. | |||
T0998 | Diazinon | Dimpylate | AChE , Parasite |
Diazinon (Dimpylate) is a thiophosphoric acid ester, functioning as a nonsystemic organophosphate insecticide that effectively targets and controls a variety of pests including cockroaches, silverfish, ants, and fleas. | |||
T62620 | ZY-444 | ||
ZY-444 is a small molecule that inhibits the progression of breast cancer and targets pyruvate carboxylase. | |||
T5173 | SBI-0640756 | SBI 0640756,SBI-756 | PERK , Autophagy |
SBI-0640756 (SBI-756) (SBI-756) is a first-in-class inhibitor that targets eIF4G1 and disrupts the eIF4F complex. | |||
T9884 | EN523 | Others | |
EN523 targets non-catalytic allosteric cysteine C23 in K48 ubiquitin-specific deuquitinase OTUB1. | |||
T16925 | SQ109 | NSC 722041 | Others , Parasite |
SQ109 (NSC-722041) is an effective inhibitor of the trypomastigote form of the parasite (IC50 = 50 nM). SQ109 is an antitubercular agent and targets MmpL3. |