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20

Compounds

Cat No. Product Name Synonyms Targets
T5722 Nevadensin Pedunculin Anti-infection , Antibacterial
Nevadensin is an important herb-based constituent inhibiting estragole bioactivation. Nevadensin protects against a methyleugenol-induced marker of hepatocarcinogenicity in male F344 rat. It also exhibits inhibition acti...
T4316 ML365 Potassium Channel
ML365 is a novel selective small molecule inhibitor of TASK1(KCNK3).
T0280 Spiperone Spiroperidol,Spiropitan Dopamine Receptor
Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds. It has been recommended in the treatment of SCHIZOPHRENIA.
TP1088 N-Acetylcarnosine N-Acetyl-L-carnosine Others
N-Acetylcarnosine (N-Acetyl-L-carnosine) is thought to be able to combat some of the effects of oxidative stress as it has anti-oxidant properties.
T12146 N-Desmethyl-Apalutamide N-Desmethyl Apalutamide P450 , Androgen Receptor
N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
T4104 Ophiopojaponin C Ophiopogonin C Others
Ophiopogonin C' pharmacological activities may be related to the substances in nucleus mainly.
T3O2709 Bronze Red Scarlet 808 Others
Bronze Red, an amide class organic compound, is utilized for content determination, identification, and pharmacological experiments.
TQ0264 Nigakinone Others
Nigakinone, isolated from Kumu, is an alkaloid with the pharmacological activity.
T7324 Chelidonine hydrochloride Others
Chelidonine hydrochloride is one of the alkaloids of Chelidonium majus, which has broad pharmacological activities
T2837 Chrysin 5, 7-Dihydroxyflavone,NSC 407436,5,7-Dihydroxyflavone Estrogen Receptor/ERR , Antioxidant
Chrysin (5,7-Dihydroxyflavone) exhibits many biological activities and pharmacological effects, including antioxidant, anti-inflammatory, anticancer, and antiviral activities.
T3S1251 Neoruscogenin ROR
1. Neoruscogenin represents a universal pharmacological tool for RORα research due to its specific selectivity profile versus other nuclear receptors.
T3362 Eupatilin NSC 122413 PPAR , Autophagy
Eupatilin (NSC-122413), a flavone derived from Artemisia princepsPampanini, is a PPARα agonist, with pharmacological activity.
T4878 Hecogenin Hocogenin Others , Antifungal
Hecogenin (Hocogenin), a steroid saponin derived from Agave sisalana, serves as a specific inhibitor for human UDP-glucuronosyltransferases. Notably, it exhibits a broad range of pharmacological activities, such as anti-...
T2891 Ammonium glycyrrhizinate Glycamil,Monoammonium glycyrrhizinate,Ammonium Glycyrrhizate,Monoammonium glycyrrhizinate hydrate,Glycyrram Others
Ammonium glycyrrhizinate (Glycyrram) has various pharmacological actions such as anti-inflammatory, antiallergic, antigastriculcer, and antihepatitis activities.
T22416 RO495 CS-2667 Tyrosine Kinases , JAK
RO495 (CS-2667), a potent inhibitor of TYK2, inhibits TYK2 with IC50 of 1.5nM as tested in cell-based pharmacological assays
T4S1659 Xanthotoxol 8-Hydroxypsoralen,8-Hydroxyfuranocoumarin,Psoralen,8-Hydroxypsoralene Reactive Oxygen Species , 5-HT Receptor , Endogenous Metabolite
Xanthotoxol (Psoralen) is a biologically active linear furocoumarin, shows strong pharmacological activities as anti-inflammatory, antioxidant, 5-HT antagonistic, and neuroprotective effects.
T7443 4'-Methoxychalcone PARP , PPAR
4'-Methoxychalcone with a variety of pharmacological activities, such as anti-tumor and anti-inflammatory activities.
TN1714 Grosvenorine Grosvenorin Antibacterial
Grosvenorine (Grosvenorin) exhibits good antibacterial and antioxidant activities, with its metabolites possessing more potent activities, intestinal bacteria play an important role in the gastrointestinal metabolism of ...
T15233 Endovion NS3728 Chloride channel
Endovion (NS3728) is a pharmacological anion channel and an Anoctamin-1 (ANO 1) channel inhibitor. Endovion is also the specific VRAC/VSOAC blocker.
T2817 Picroside II Vanilloyl catalpol,6-Vanilloylcatalpol Apoptosis , Others , Influenza Virus , NF-κB , Reactive Oxygen Species
Picroside II (Vanilloyl catalpol) is the main active ingredient in iridoid glycosides. It has antioxidant, anti-inflammatory, immune regulatory, anti-virus and other pharmacological activities.

Compounds

Nevadensin
T5722
Synonym: Pedunculin
Target: Anti-infection, Antibacterial
ML365
T4316
Synonym:
Target: Potassium Channel
Spiperone
T0280
Synonym: Spiroperidol,Spiropitan
Target: Dopamine Receptor
N-Acetylcarnosine
TP1088
Synonym: N-Acetyl-L-carnosine
Target: Others
N-Desmethyl-Apalutamide
T12146
Synonym: N-Desmethyl Apalutamide
Target: P450, Androgen Receptor
Ophiopojaponin C
T4104
Synonym: Ophiopogonin C
Target: Others
Bronze Red
T3O2709
Synonym: Scarlet 808
Target: Others
Nigakinone
TQ0264
Synonym:
Target: Others
Chelidonine hydrochloride
T7324
Synonym:
Target: Others
Chrysin
T2837
Synonym: 5, 7-Dihydroxyflavone,NSC 407436,5,7-Dihydroxyflavone
Target: Estrogen Receptor/ERR, Antioxidant
Neoruscogenin
T3S1251
Synonym:
Target: ROR
Eupatilin
T3362
Synonym: NSC 122413
Target: PPAR, Autophagy
Hecogenin
T4878
Synonym: Hocogenin
Target: Others, Antifungal
Ammonium glycyrrhizinate
T2891
Synonym: Glycamil,Monoammonium glycyrrhizinate,Ammonium Glycyrrhizate,Monoammonium glycyrrhizinate hydrate,Glycyrram
Target: Others
RO495
T22416
Synonym: CS-2667
Target: Tyrosine Kinases, JAK
Xanthotoxol
T4S1659
Synonym: 8-Hydroxypsoralen,8-Hydroxyfuranocoumarin,Psoralen,8-Hydroxypsoralene
Target: Reactive Oxygen Species, 5-HT Receptor, Endogenous Metabolite
4'-Methoxychalcone
T7443
Synonym:
Target: PARP, PPAR
Grosvenorine
TN1714
Synonym: Grosvenorin
Target: Antibacterial
Endovion
T15233
Synonym: NS3728
Target: Chloride channel
Picroside II
T2817
Synonym: Vanilloyl catalpol,6-Vanilloylcatalpol
Target: Apoptosis, Others, Influenza Virus, NF-κB, Reactive Oxygen Species
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TargetMol