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20

Compounds

Cat No. Product Name Synonyms Targets
T1154 Rifaximin DNA/RNA Synthesis , Antibacterial , Antibiotic
Rifaximin is an orally administered, semi-synthetic, nonsystemic antibiotic derived from rifamycin SV with antibacterial activity. Rifaximin binds to the beta-subunit of bacterial DNA-dependent RNA polymerase, inhibiting...
T22671 CJ 033466 5-HT Receptor
CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.
T5051 Isopropamide Iodide AChR
Isopropamide iodide is a long-acting anticholinergic drug. It is used in the treatment of peptic ulcers and other gastrointestinal disorders. It also acts as a muscarinic receptor antagonist which can be applied to the t...
T38612 Linaprazan glurate Others
Linaprazan glurate inhibits exogenously or endogenously stimulated gastric acid secretion. Linaprazan glurate can be used in studies about gastrointestinal inflammatory diseases and peptic ulcer diseases.
T5S1172 Tiliroside Tribuloside Antioxidant
1. Tiliroside (Tribuloside) shows anticarcinogenic activity. 2. Tiliroside shows hepatoprotective activity. 3. Tiliroside shows antioxidant and anti-inflammatory activity, can inhibit neuroinflammation in neurodegenerati...
TN1008 Psoralenoside CaMK , Calcium Channel , Histamine Receptor
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activity, antitumor effects and antibacterial activity.
T21422 Methylnaltrexone bromide Relistor,MOA-728,MOA 728,Methylnaltrexone,MOA728 Opioid Receptor
Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists. Methylnaltrexone bromide acts to reverse some of the side effects of opioid drugs such as constipation without af...
T7022 PEG300 Polyethylene glycol 300 Others
PEG300 (Polyethylene glycol 300) is a polymer formed from repeating units of ethylene glycol that is water soluble, low immunogenicity, and biocompatible. PEG300 is a neutral polymer with a molecular weight of 300.
T6935 Nirogacestat PF-03084014,PF-3084014,PF03084014,PF 03084014 Apoptosis , Gamma-secretase
Nirogacestat (PF 03084014) is a specific γ-secretase inhibitor (IC50: 6.2 nM, in a cell-free assay).
T0794 Mepenzolate Bromide Colibantil,Cantil,Cantilaque AChR
Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.
T0199 Cephradine Anspor,Cephradin,Velosef,SQ-11436,Sefril TOPK , Antibacterial , Antibiotic
Cephradine (Anspor) is a beta-lactam, first-generation cephalosporin antibiotic with bactericidal activity.
T0700 Ursodeoxycholic acid UDCA,Ursodiol Potassium Channel , Endogenous Metabolite
Ursodeoxycholic acid (UDCA) can be used to dissolve gallstones and reduce cholesterol absorption.
T1551 Tegaserod maleate HTF-919,SDZ-HTF-919 5-HT Receptor
Tegaserod maleate (SDZ-HTF-919) is a 5-HT4 agonist manufactured by Novartis and used for the management of irritable bowel syndrome and constipation. Its use was the only drug approved by the United States Food and Drug ...
T24047 Etilevodopa hydrochloride Levodopa ethyl ester,Etilevodopa HCl, L-DOPA ethyl ester Others , Dopamine Receptor , Drug Metabolite
Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.
T1291 Cisapride Prepulsid,R 51619,Pridesia,Kaudalit,(±)-Cisaprid,Kinestase Potassium Channel , 5-HT Receptor , HER
Cisapride (R 51619) is a serotonin type 4 (5-HT4) receptor agonists are potent prokinetic agents that act on serotonin receptors in the intestine and promote intestinal peristalsis, increase gastric emptying and decrease...
TP1793 Nociceptin (1-13), amide Opioid Receptor
Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain membranes.
T16083 Mizagliflozin GSK-1614235 free base,KGA-3235 free base,DSP-3235 free base SGLT
Mizagliflozin (GSK-1614235 free base) is a sodium-glucose transporter inhibitor( Ki of 27 nM for human SGLT1). Mizagliflozin displays 303-fold selectivity over SGLT2. Mizagliflozin is used as an antidiabetic drug that ca...
T29078 Ursodeoxycholic acid sodium UDCA Na,UDCA sodium,Sodium Ursodeoxycholate,Ursodiol sodium,Ursodeoxycholic Acid (sodium salt),Ursodeoxycholate sodium FXR , Endogenous Metabolite , GPCR19
Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities. Ursodeoxycholic acid sodium acts as signaling molecule, exerting it...
T13570 Benzamide Derivative 1 Others
Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.
T13997 AU-224 Others
AU-224 is an orally available benzamide derivative that is a potent gastrointestinal prokinetic.

Compounds

Rifaximin
T1154
Synonym:
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
CJ 033466
T22671
Synonym:
Target: 5-HT Receptor
Isopropamide Iodide
T5051
Synonym:
Target: AChR
Linaprazan glurate
T38612
Synonym:
Target: Others
Tiliroside
T5S1172
Synonym: Tribuloside
Target: Antioxidant
Psoralenoside
TN1008
Synonym:
Target: CaMK, Calcium Channel, Histamine Receptor
Methylnaltrexone bromide
T21422
Synonym: Relistor,MOA-728,MOA 728,Methylnaltrexone,MOA728
Target: Opioid Receptor
PEG300
T7022
Synonym: Polyethylene glycol 300
Target: Others
Nirogacestat
T6935
Synonym: PF-03084014,PF-3084014,PF03084014,PF 03084014
Target: Apoptosis, Gamma-secretase
Mepenzolate Bromide
T0794
Synonym: Colibantil,Cantil,Cantilaque
Target: AChR
Cephradine
T0199
Synonym: Anspor,Cephradin,Velosef,SQ-11436,Sefril
Target: TOPK, Antibacterial, Antibiotic
Ursodeoxycholic acid
T0700
Synonym: UDCA,Ursodiol
Target: Potassium Channel, Endogenous Metabolite
Tegaserod maleate
T1551
Synonym: HTF-919,SDZ-HTF-919
Target: 5-HT Receptor
Etilevodopa hydrochloride
T24047
Synonym: Levodopa ethyl ester,Etilevodopa HCl, L-DOPA ethyl ester
Target: Others, Dopamine Receptor, Drug Metabolite
Cisapride
T1291
Synonym: Prepulsid,R 51619,Pridesia,Kaudalit,(±)-Cisaprid,Kinestase
Target: Potassium Channel, 5-HT Receptor, HER
Nociceptin (1-13), amide
TP1793
Synonym:
Target: Opioid Receptor
Mizagliflozin
T16083
Synonym: GSK-1614235 free base,KGA-3235 free base,DSP-3235 free base
Target: SGLT
Ursodeoxycholic acid sodium
T29078
Synonym: UDCA Na,UDCA sodium,Sodium Ursodeoxycholate,Ursodiol sodium,Ursodeoxycholic Acid (sodium salt),Ursodeoxycholate sodium
Target: FXR, Endogenous Metabolite, GPCR19
Benzamide Derivative 1
T13570
Synonym:
Target: Others
AU-224
T13997
Synonym:
Target: Others
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TargetMol