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Compounds

Natural Products

Recombinant Proteins

Cat No.	Product Name	Synonyms	Targets
T34905	Totrombopag	SB559448,SB 559448,SB-559448,LGD-4665,Synonym 2,LGD 4665,LGD4665
	Totrombopag (SB559448) is a candidate compound for action on RSV polymerase.
TQ0223	Lusutrombopag	S-888711,Mulpleta	Thrombin , Thrombopoietin Receptor
	Lusutrombopag (Mulpleta) is an orally bioavailable, small molecule thrombopoietin (TPO) receptor agonist for chronic liver disease (CLD) patients with thrombocytopenia prior to elective invasive surgery.		Thrombin , Thrombopoietin Receptor
T20641	Propagermanium	Dipropanoic acid germanium sequioxide,SK-818,Ge 132,Ge132,SK 818,Ge-132	Others
	Propagermanium (Ge132), an organometallic compound of germanium, has been used as a therapeutic agent against chronic hepatitis B in Japan.		Others
T1088	Repaglinide	AG-EE 388 ZW,AG-EE 623ZW	Potassium Channel , PPAR
	Repaglinide (AG-EE 623ZW) is a benzoic acid derivative that stimulates insulin secretion from the pancreas and is used in the therapy of type 2 diabetes. Repaglinide has been linked to rare instances of clinically appare...		Potassium Channel , PPAR
T1766	Empagliflozin	BI 10773	SGLT
	Empagliflozin (BI 10773) is an SGLT-2 inhibitor (IC50=3.1 nM) that is potent and selective, with more than 300-fold selectivity for SGLT-1/4/5/6. Empagliflozin is used for the treatment of type 2 diabetes.		SGLT
T15259	Evatanepag	CP-533536 free acid	Prostaglandin Receptor
	Evatanepag (CP-533536 free acid) is an EP2 receptor selective prostaglandin E2 (PGE2) agonist that induces local bone formation with EC50 of 0.3 nM.CP-533536 demonstrated the ability to heal fractures when administered l...		Prostaglandin Receptor
T3174	Taprenepag	CP-544326	Prostaglandin Receptor
	Taprenepag (CP-544326) (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (EC50 = 2.8 nM). Taprenepag has been used in trials studying the treatment of Ocular Hypertension and Glaucoma, Open-Angle.		Prostaglandin Receptor
T67849	O-Desethyl Dapagliflozin	Empagliflozin-4	SGLT
	O-Desethyl Dapagliflozin (Empagliflozin-4) is a SGLT2 inhibitor, IC50=33nM.		SGLT
T15273	Fedovapagon	VA483,A106483	Vasopressin Receptor
	Fedovapagon (VA106483) is a selective and potent agonist of the vasopressin V2 receptor (V2R) that inhibits the growth of intersegmental vessels in zebrafish. Fedovapagon can be used to study overactive bladder, nocturia...		Vasopressin Receptor
T4460	Dapagliflozin ((2S)-1,2-propanediol, hydrate)	BMS-512148 (2S)-1,2-propanediol, hydrate,Dapagliflozin propanediol monohydrate	SGLT
	Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) is a selective, orally active inhibitor of the renal sodium-glucose co-transporter type 2 (SGLT2). It is in development for the tre...		SGLT
T2389	Dapagliflozin	BMS-512148	SGLT , HIF
	Dapagliflozin (BMS-512148) is a selective sodium-glucose co-transporter subtype 2 (SGLT2) inhibitor with antihyperglycemic activity.		SGLT , HIF
T6750	Opaganib	ABC294640	S1P Receptor
	Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).		S1P Receptor
T3216	Selexipag	NS-304,ACT-293987,Uptravi	Others , Prostaglandin Receptor
	Selexipag (ACT-293987)(NS-304) is prostacyclin receptor agonist that causes vasodilation in pulmonary vasculature and is used in the therapy of pulmonary arterial hypertension (PAH).		Others , Prostaglandin Receptor
T22870	IPAG		Opioid Receptor
	IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.		Opioid Receptor
T2562	Eltrombopag	SB-497115,SB-497115-GR	Thrombin
	Eltrombopag (SB-497115-GR), an orally active thrombopoietin receptor agonist with megakaryopoiesis stimulating activity, binds to and stimulates the platelet thrombopoietin receptor (TPO-R or CD110).		Thrombin
T7417	Avatrombopag	YM477,AKR-501,E5501	Thrombin , Thrombopoietin Receptor
	Avatrombopag (YM477) is a new oral thrombopoietin (TPO) receptor agonist, activating TPO receptor and increasing megakaryocytic proliferation/differentiation and platelet production.		Thrombin , Thrombopoietin Receptor
T4635	Ralinepag	APD811	Others , Prostaglandin Receptor
	Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human and rat IP receptor and human DP1 receptor, respectively.		Others , Prostaglandin Receptor
T6825	Eltrombopag Olamine	Promacta Olamine,Revolade,Eltrombopag diethanolamine salt,SB497115,SB-497115GR	Thrombin
	Eltrombopag Olamine (Eltrombopag diethanolamine salt) is the orally active ethanolamine salt of eltrombopag, a small-molecule, nonpeptide thrombopoietin receptor agonist with megakaryopoiesis-stimulating activity. Eltrom...		Thrombin
T34644	Simenepag isopropyl	AGN210669,AGN-210669,AGN 210669
	Simenepag isopropyl can be used for the treatment of Glaucoma, Ocular Hypertension.
T13497	3'-Hydroxy Repaglinide		Others
	3'-Hydroxy Repaglinide is a main CYP2C8 metabolite of Repaglinide. Repaglinide is a carbamoylmethyl benzoic acid derivative and used as the treatment of type II diabetes.		Others
T61876	Sipagladenant
	Sipagladenant (Compound I) is an orally active inverse agonist targeting the adenosine receptor A2A [1]. It possesses potential for utilization in research pertaining to frontal lobe dysfunction [2].
T64667	10× SDS-PAGE SDS Running Buffer		Others
	10× SDS-PAGE SDS Running Buffer is a 10-fold concentrated buffer for SDS-PAGE (SDS-denaturing polyacrylamide gel electrophoresis), with the main components of trimethylolaminomethane (Tris), glycine (Glycine) and sodium ...		Others
T25547	Isospaglumate sodium	Isospaglumate trisodium,Sodium isospaglumate
	Isospaglumate sodium is the sodium salt of isospaglumate which is an antiallergic agent.
T40654	Avatrombopag hydrochloride	AKR-501 hydrochloride,YM477hydrochloride,E5501hydrochloride
	Avatrombopag hydrochloride (AKR-501) is an orally active, nonpeptide agonist of the thrombopoietin (TPO) receptor with an EC 50 of 3.3 nM. It effectively mimics the biological activities of TPO, stimulating platelet prod...
T16988	Taprenepag isopropyl	PF-04217329	Prostaglandin Receptor
	Taprenepag isopropyl is a highly selective agonist of the EP2 receptor.		Prostaglandin Receptor
T76822	Pagibaximab
	Pagibaximab, a chimeric IgG1 antibody, targets the lipoteichoic acid on the surfaces of S. aureus and S. epidermidis, and is utilized for the prevention of staphylococcal sepsis [1].
T76057	Glepaglutide acetate
	Glepaglutide (ZP1848) acetate is a long-acting glucagon-like peptide-2 (GLP-2) analogue and a potent GLP-2 receptor (GLP-2R) agonist. It significantly reduces fecal output and enhances intestinal absorption while also mi...
T16388	Omidenepag isopropyl		Prostaglandin Receptor
	Omidenepag isopropyl is converted to the active product Omidenepag during corneal penetration. Omidenepag isopropyl is a selective EP2 receptor agonist. Omidenepag isopropyl displays only a weak affinity for EP1, EP2, an...		Prostaglandin Receptor
T69755	Evatanepag sodium
	Evatanepag, also known as CP-533536, is an EP2 receptor selective prostaglandin E2 (PGE2) agonist that induces local bone formation. CP-533536 demonstrated the ability to heal fractures when administered locally as a sin...
T126029	8-cis-Cinnamoylharpagide
	8-cis-Cinnamoylharpagide is a useful organic compound for research related to life sciences. The catalog number is T126029 and the CAS number is 133645-36-0.
T29708	Aganepag isopropyl	AGN-210961,AGN 210961,AGN210961
	Aganepag isopropyl can be used to treat Glaucoma.
T68560	Totrombopag choline
	Totrombopag, also known LGD-4665, GSK2285921 and SB559448, is an oral thromobopoietin receptor agonist, is being developed as a new generation small molecule thrombopoietin (TPO) mimetic. It is a highly selective and po...
T64615	EMpagliflozin iMpurity 5
	(2S,3R,4R,5S,6R)-2-(4-Chloro-3-(4-hydroxybenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol is a useful organic compound for research related to life sciences and the catalog number is T64615.
T76056	Glepaglutide
	Glepaglutide (ZP1848), a long-acting glucagon-like peptide-2 (GLP-2) analogue, functions as a potent agonist of the GLP-2 receptor (GLP-2R), effectively reducing fecal output and enhancing intestinal absorption, while al...
T79850	Irpagratinib	ABSK011	FGFR
	Irpagratinib (ABSK011) is an orally active fibroblast growth factor receptor (FGFR) tyrosine kinase inhibitor with specificity for FGFR4, exhibiting an IC50 of less than 10 nM. It effectively inhibits FGFR4 auto-phosphor...		FGFR
T35619	Dapagliflozin-3-O-β-D-Glucuronide
	Dapagliflozin-3-O-β-D-glucuronide is a metabolite of dapagliflozin . Dapagliflozin is a first generation selective sodium glucose cotransporter (SGLT) 2 inhibitor that blocks glucose transport.[1] Dapagliflozin is metab...
T124813	N-Methylsarpagine methosalt
	N-Methylsarpagine methosalt is a useful organic compound for research related to life sciences and the catalog number is T124813.
T62906	Lazuvapagon
	Lazuvapagon is a vasopressin V2 receptor agonist that can be used to study enuresis.
T27536	Hetrombopag olamine
	Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity.
T38602	(E/Z)-Eltrombopag 13C4	(E/Z)-Eltrombopag 13C4,(E/Z)-SB-497115 13C4
	(E/Z)-Eltrombopag 13C4 ((E/Z)-SB-497115 13C4) is a mixture complex of E-Eltrombopag and Z-Eltrombopag, with 13C labeled. Z-Eltrombopag is a thrombopoietin (TPO) receptor agonist developed for certain conditions that lead...
T29707	Aganepag ethanediol	AGN-212409,AGN212409
	Aganepag ethanediol, an IOP-lowering agent, is an antiglaucoma agent. Aganepag ethanediol is a selective EP2 receptor agonist.
T14139	Aganepag	AGN 210937	Prostaglandin Receptor
	Aganepag, a potent Prostanoid EP2 receptor agonist, exhibits remarkable selectivity with an EC50 of 0.19 nM, demonstrating no activity at the EP4 receptor. Its applications are primarily in the fields of wound healing, s...		Prostaglandin Receptor
T126028	8-O-4-Hydroxycinnamoylharpagide
	8-O-4-Hydroxycinnamoylharpagide is a useful organic compound for research related to life sciences. The catalog number is T126028 and the CAS number is 133645-37-1.
T124431	Pagoside

T68888	Avatrombopag maleate
	Avatrombopag, also known as AKR-501, YM477, AS 1670542 or E5501, is a novel orally-active thrombopoietin (TPO) receptor agonist. AKR-501 specifically targeted the TPO receptor and stimulated megakaryocytopoiesis througho...
T16389	Omidenepag		Prostaglandin Receptor
	Omidenepag is a pharmacologically active form of Omidenepag Isopropyl and is a selective, non-prostanoid EP2 receptor agonist (EC50: 1.1 nM). Omidenepag displays binding affinities (IC50: 10 nM for h-EP2).		Prostaglandin Receptor
T71301	Opaganib HCl
	ABC294640, also known as Opaganib, is an orally available, aryladamantane compound and selective inhibitor of sphingosine kinase-2 (SK2) with potential antineoplastic activity. Upon administration, ABC294640 competitivel...
TQ0285L	Spaglumic acid acetate	Isospaglumic acid acetate,Spaglumic acid acetate（3106-85-2 Free base）	Endogenous Metabolite
	Spaglumic acid acetate (Isospaglumic acid acetate) is a neuropeptide found in millimolar concentrations in brain.		Endogenous Metabolite
T72265	Eltrombopag methyl ester
	Eltrombopag Methyl Ester, a derivative of Eltrombopag, functions as a thrombopoietin (Tpo) receptor agonist to enhance platelet production and is employed in the study of certain thrombocytopenia variants.
T124022	8-p-Coumaroylharpagide

Compounds

Totrombopag

T34905

Synonym: SB559448,SB 559448,SB-559448,LGD-4665,Synonym 2,LGD 4665,LGD4665

Target:

Lusutrombopag

TQ0223

Synonym: S-888711,Mulpleta

Target: Thrombin, Thrombopoietin Receptor

Propagermanium

T20641

Synonym: Dipropanoic acid germanium sequioxide,SK-818,Ge 132,Ge132,SK 818,Ge-132

Target: Others

Repaglinide

T1088

Synonym: AG-EE 388 ZW,AG-EE 623ZW

Target: Potassium Channel, PPAR

Synonym: CP-533536 free acid

Target: Prostaglandin Receptor

Taprenepag

T3174

Synonym: CP-544326

Target: Prostaglandin Receptor

O-Desethyl Dapagliflozin

T67849

Synonym: Empagliflozin-4

Target: SGLT

Fedovapagon

T15273

Synonym: VA483,A106483

Target: Vasopressin Receptor

Dapagliflozin ((2S)-1,2-propanediol, hydrate)

T4460

Synonym: BMS-512148 (2S)-1,2-propanediol, hydrate,Dapagliflozin propanediol monohydrate

Cat No.	Product Name	Synonyms	Targets
TQ0285	Spaglumic acid	N-Acetylaspartylglutamic acid,NAAG	Endogenous Metabolite
	Spaglumic acid (N-Acetylaspartylglutamic acid) is a neuropeptide found in millimolar concentrations in the brain.		Endogenous Metabolite
T6S2023	Harpagoside		Others , COX , NO Synthase
	1. Harpagoside has anti-inflammatory activity. 2. Harpagoside at 3 mM concentration, shows moderate inhibition of seed germination. 3. Harpagoside can inhibit lipopolysaccharide-induced mRNA levels and protein expression...		Others , COX , NO Synthase
T6S2024	Harpagide		Antibacterial , Parasite
	1. Harpagide has antibacterial activity. 2. Harpagide has antiviral activity. 3. Harpagide has anti-inflammatory activity.		Antibacterial , Parasite
T6S2025	8-O-Acetylharpagide	8-Acetylharpagide,3-Acetylharpagide,Acetylharpagide,8-O-Acetylharpagide	Antibacterial
	1. 8-O-Acetylharpagide has anti-inflammatory activity. 2. 8-O-Acetylharpagide has antibacteria and antiviral activities. 3. 8-O-Acetylharpagide has a biological activity on isolated smooth muscle preparations from guinea...		Antibacterial
T20617	Sarpagine	Raupin
	Sarpagine is an alkaloid with the antihypertonic effect.
TN1321	6'-O-Cinnamoyl harpagide	6'-O-Cinnamoylharpagide	Others
	6'-O-Cinnamoylharpagide has anti-inflammatory activity.		Others
TN3167	6-Epiharpagoside		Others
	6-Epiharpagoside is a natural product for research related to life sciences. The catalog number is TN3167 and the CAS number is 1151862-67-7.		Others
T74202	Hispaglabridin A
	Hispaglabridin A, an effective antioxidant, inhibits lipid peroxidation [1].
TN2953	3-Hydroxysarpagine		Topoisomerase
	3-Hydroxysarpagine is a natural product of Rauvolfia, Apocynaceae. The catalog number is TN2953 and the CAS number is 857297-90-6. 3-Hydroxysarpagine can be used as a reference standard.		Topoisomerase
TN4034	Eupaglehnin C		Others
	Eupaglehnin C shows cytotoxic (2.19 mg/ml) against HeLa-S3.		Others
TN3166	6-Epiharpagide		Others
	6-Epiharpagide is a natural product from Scrophularia ningpoensis Hemsl.		Others
TN3162	6-Epi-8-O-acetylharpagide		Others
	6-Epi-8-O-acetylharpagide is a natural product of Scrophularia, Scrophulariaceae. The catalog number is TN3162 and the CAS number is 97169-44-3. 6-Epi-8-O-acetylharpagide can be used as a reference standard.		Others
T2S1749	Protogracillin		Others
	Protogracillin may have inhibitions on platelet aggregation (PAG) and thrombosis.		Others

Cat No.	Product Name	Species	Expression System
TMPH-00294	PAG-1 Protein, Bovine, Recombinant (His & SUMOstar)	Bovine	P. pastoris (Yeast)
	Appears to be proteolytically inactive. PAG-1 Protein, Bovine, Recombinant (His & SUMOstar) is expressed in yeast with N-6xHis-sumostar tag. The predicted molecular weight is 49.8 kDa and the accession number is Q29432.
TMPH-00293	PAG-1 Protein, Bovine, Recombinant (His)	Bovine	E. coli
	Appears to be proteolytically inactive. PAG-1 Protein, Bovine, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 40.7 kDa and the accession number is Q29432.
TMPH-00295	PAG-2 Protein, Bovine, Recombinant (His)	Bovine	E. coli
	PAG2 or a processed derivative of this molecule might represent a factor that binds the LH receptor. PAG-2 Protein, Bovine, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted mole...
TMPY-01276	Peroxiredoxin 1 Protein, Human, Recombinant (His)	Human	E. coli
	Peroxiredoxin 1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 22.9 kDa and the accession number is A0A384NPQ2.
TMPY-02372	Peroxiredoxin 1 Protein, Mouse, Recombinant (His)	Mouse	E. coli
	Peroxiredoxin 1 Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 23.5 kDa and the accession number is P35700.
TMPH-03081	ACE2 Protein, Paguma larvata, Recombinant (hFc)	Paguma larvata	HEK293 Cells
	ACE2 Protein, Paguma larvata, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The predicted molecular weight is 112.7 kDa and the accession number is Q56NL1.
TMPH-00743	PhoP Protein, E. coli, Recombinant (HEK293, His & Myc)	E. coli	HEK293 Cells
	Member of the two-component regulatory system PhoP/PhoQ involved in adaptation to low Mg(2+) environments and the control of acid resistance genes. In low periplasmic Mg(2+), PhoQ phosphorylates PhoP, resulting in the ex...
TMPK-00556	BTN3A1 Protein, Cynomolgus, Recombinant (His & Avi)	Cynomolgus	HEK293 Cells
	The three butyrophilin BTN3A molecules, BTN3A1, BTN3A2, and BTN3A3, are members of the B7/butyrophilin-like group of Ig superfamily receptors, which modulate the function of T cells. BTN3A1 controls activation of human V...
TMPK-00310	BTN3A1 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	The three butyrophilin BTN3A molecules, BTN3A1, BTN3A2, and BTN3A3, are members of the B7/butyrophilin-like group of Ig superfamily receptors, which modulate the function of T cells. BTN3A1 controls activation of human V...
TMPK-00557	BTN3A1 Protein, Cynomolgus, Recombinant (His & Avi), Biotinylated	Cynomolgus	HEK293 Cells
	The three butyrophilin BTN3A molecules, BTN3A1, BTN3A2, and BTN3A3, are members of the B7/butyrophilin-like group of Ig superfamily receptors, which modulate the function of T cells. BTN3A1 controls activation of human V...