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Aganepag

Catalog No. T14139 CAS 910562-18-4

Synonyms: AGN 210937

Aganepag, a potent Prostanoid EP2 receptor agonist, exhibits remarkable selectivity with an EC50 of 0.19 nM, demonstrating no activity at the EP4 receptor. Its applications are primarily in the fields of wound healing, scar reduction, scar prevention, and the treatment and prevention of wrinkles.

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Aganepag, CAS 910562-18-4

Pack Size	Availability	Price/USD
25 mg	6-8 weeks	$ 2,270.00
50 mg	6-8 weeks	$ 2,980.00
100 mg	6-8 weeks	$ 4,000.00

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This compound is a customized synthesis product. We have a strong synthesis team with excellent synthesis technology and capabilities. However, due to various objective factors, there is a low probability that the synthesis will not be successful. If you need to learn more, please feel free to consult us, we will serve you wholeheartedly.

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Aganepag, a potent Prostanoid EP2 receptor agonist, exhibits remarkable selectivity with an EC50 of 0.19 nM, demonstrating no activity at the EP4 receptor. Its applications are primarily in the fields of wound healing, scar reduction, scar prevention, and the treatment and prevention of wrinkles.
Targets&IC50	EP2:0.19 nM （EC50）
In vitro	Aganepag (Compound 3), a powerful Prostanoid EP2 receptor agonist, exhibits an EC50 of 0.19 nM and lacks activity at the EP4 receptor. This compound is applicable in studies focused on wound healing, scar reduction and prevention, as well as the treatment and prevention of wrinkles[1].

Synonyms	AGN 210937
Molecular Weight	429.57
Formula	C24H31NO4S
CAS No.	910562-18-4

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Robert M. Burk, et al. Compounds and methods for skin repair. WO2014078434A1

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Aganepag 910562-18-4 GPCR/G Protein Immunology/Inflammation Prostaglandin Receptor AGN-210937 AGN 210937 AGN210937 inhibitor inhibit

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