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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T21967 | MEG hemisulfate | Mercaptoethylguanidine hemisulfate | NOS |
MEG hemisulfate (Mercaptoethylguanidine hemisulfate) acts as a highly potent and selective suppressor of inducible NO synthase (iNOS), demonstrating EC50 values of 11.5 μM for iNOS, 110 μM for ecNOS, and 60 μM for bNOS i... | |||
T60530 | Mercaptoethylguanidine (MEG) (dihydrobromide) | ||
Mercaptoethylguanidine (MEG) dihydrobromide is a selective inducible nitric oxide synthase inhibitor and peroxynitrite scavenger with potential for inflammatory bowel diseases research. | |||
T20992 | MEGA-9 | Nonanoyl-N-Methylglucamide | Serine Protease |
MEGA-9 (Nonanoyl-N-Methylglucamide) solubilizes membrane protein and can be used as a nonionic detergent. | |||
T31213 | Dazmegrel | UK-38,485,UK 38485,UK 38,485,UK38,485,UK-38485 | PPAR |
Dazmegrel (UK 38,485) is a potent and specific thromboxane A2 (TXA2) synthase inhibitor for the prevention of increased whole platelet aggregation in normal pregnancy. | |||
T2495 | Lomeguatrib | PaTrin-2 | DNA Methyltransferase , DNA Alkylation |
Lomeguatrib (PaTrin-2), a modified guanine base, inhibits the activity of DNA repair protein O(6)-alkylguanine-DNA alkyltransferase (MGMT) . | |||
T1396 | Bemegride | Bemegrid,3-Ethyl-3-methylglutarimide,Agipnon | GABA Receptor |
Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning. | |||
T14130 | Adomeglivant | LY2409021 | Glucagon Receptor |
Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus. | |||
T1209 | Flunixin meglumine | Banamine,Finadyne,Flunixin meglumin | COX |
Flunixin meglumine (Banamine) is an effective inhibitor of the enzyme cyclooxygenase with anti-inflammatory and antipyretic activity. | |||
T4610 | Rimegepant | BMS 927711,BMS-927711,BMS927711,BHV-3000 | CGRP Receptor |
Rimegepant (BMS 927711) is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM. | |||
T0503 | Meglumine | Meglumin,Methylglucamin,Methylglucamine | Others |
Meglumine (Meglumin), a derivative of sorbitol, is used in conjunction with iodinated organic compounds as contrast medium. | |||
T8395 | Nomegestrol acetate | Others , Progesterone Receptor | |
Nomegestrol acetate is a widely used progestin-like drug,which is characterized as a full agonist at the progesterone receptor | |||
T1284 | Megestrol acetate | SC10363,BDH1298 | Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , HIV Protease , Autophagy |
Megestrol acetate (BDH1298) is a progestogen with actions and uses similar to those of the progestogens in general. Megestrol acetate also has anti-androgenic properties. It is given by mouth in the palliative treatment ... | |||
T8173 | Delafloxacin meglumine | ABT492 meglumine,WQ-3034 meglumine,RX-3341 meglumine | Antibacterial , Antibiotic |
Delafloxacin meglumine (RX-3341 meglumine) is a broad-spectrum fluoroquinolone antibiotic. | |||
T4506 | Gadopentetate dimeglumine | Meglumine gadopentetate,SH-L-451A,Gd-DTPA,Gadopentetic acid dimeglumine,Gadopentetic acid dimeglumine salt | Others |
Gadopentetate dimeglumine (Gd-DTPA), an extracellular intravenous contrast agent, is used in combination with magnetic resonance imaging (MRI) to allow blood vessels, organs, and other non-bony tissues to be seen more cl... | |||
T20637 | Diatrizoate meglumine | Reno,Renografin,Renovist,Hypaque,Renocal,Sinografin | Others |
Diatrizoate meglumine (Renocal) is the meglumine salt of diatrizoate, it is an organic, iodinated, radiopaque X-ray contrast medium used in diagnostic radiography. | |||
T7582 | Tafamidis meglumine | Fx-1006A | Others |
Tafamidis meglumine (Fx-1006A) is a Potent and Selective Transthyretin Kinetic Stabilizer That Inhibits the Amyloid Cascade | |||
T7486 | Imeglimin hydrochloride | EMD 387008 hydrochloride | Reactive Oxygen Species , Mitochondrial Metabolism |
Imeglimin hydrochloride (EMD 387008 hydrochloride) prevents human endothelial cell death by inhibiting mitochondrial permeability transition without inhibiting mitochondrial respiration. | |||
T1790 | Fosaprepitant dimeglumine | L785298,MK-0517,Fosaprepitant dimeglumine salt | Neurokinin receptor |
Fosaprepitant dimeglumine (MK-0517) is the dimeglumine salt form of fosaprepitant, the water-soluble, N-phosphorylated prodrug of aprepitant, with antiemetic activity. Upon intravenous administration and rapid conversion... | |||
T1664 | Meglutol | Dicrotalic acid,3-Hydroxy-3-methylglutaric acid | Endogenous Metabolite , HMG-CoA Reductase , Autophagy |
Meglutol (3-Hydroxy-3-methylglutaric acid) is an antilipemic agent which lowers cholesterol, triglycerides, serum beta-lipoproteins and phospholipids. It acts by interfering with the enzymatic steps involved in the conve... | |||
T19811 | Nomegestrol | ||
Nomegestrol is a progestin. It is used in the treatment of gynecological disorders, in menopausal hormone therapy for the treatment of menopausal symptoms, and in hormonal contraceptives. |