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Search Results for " cem "

20

Compounds

Cat No. Product Name Synonyms Targets
T2331 Solithromycin OP-1068,CEM-101 Antibacterial , Antibiotic
Solithromycin (OP-1068) is an orally bioavailable antimicrobial agent that inhibits cell viability, protein synthesis, and growth rate of Streptococcus pneumoniae, Staphylococcus aureus, Staphylococcus aureus, and Haemop...
T39810 CEM114
CEM114 is a potent chemical compound known as a chemical epigenetic modifier (CEM). It functions by employing CRISPR-Cas9 systems to harness endogenous chromatin machinery, thereby exerting its epigenetic modifying effec...
T9104 TJ191 Apoptosis
TJ191 is a selective anti-cancer agent, targeting low TβRIII-expressing malignant T-cell leukemia/lymphoma cells.
T20038 2-Fluoroadenine NSC-27364,NSC 27364,NSC27364 DNA/RNA Synthesis
2-Fluoroadenine (NSC-27364) has toxicity in nonproliferating and proliferating tumor cells. 2-Fluoroadenine can be used for anticancer studies.
T6018 Zosuquidar trihydrochloride Zosuquidar (LY335979) 3HCl,RS 33295-198 trihydrochloride,RS 33295-198 (D06387) 3HCl,Zosuquidar 3HCl,LY-335979 trihydrochloride P-gp
Zosuquidar trihydrochloride (LY-335979 trihydrochloride) is a potent modulator of P-glycoprotein-mediated multi-drug resistance with Ki of 60 nM. Phase 3.
T0370 Pheniramine maleate Daneral,Inhiston,Trimetose 5-HT Receptor , Histamine Receptor
Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors, thereby inhibiting phospholipase A2 and production of the endothelium-derived re...
T5858 Sertindole Lu 23-174 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Autophagy
Sertindole (Lu 23-174) is an atypical antipsychotic that binds to dopamine D2 receptors and the serotonin (5-HT) receptor subtypes 5-HT1D, 5-HT2A, and 5-HT2C (Kds = 2.7, 20, 0.14, and 6 nM, respectively)
T16731 Rentiapril racemate (Rac)-SA-446,SA-446 racemate,(Rac)-Rentiapril Angiotensin-converting Enzyme (ACE)
Rentiapril racemate (SA-446 racemate) is the racemate of Rentiapril.Rentiapril racemate has anti-inflammatory activity and may be used in glaucoma research.
T13514 5-MethoxyPinocembroside Others
5-MethoxyPinocembroside is a flavonoid isolated from leaves of Moringa oleifera.
T4345 CeMMEC1 CeMMEC1 HCl Epigenetic Reader Domain , Carboxypeptidase , DNA/RNA Synthesis
CeMMEC1 is an inhibitor of BRD4, and also has a great affinity for TAF1(IC50=0.9 μM).
T7220 Prohydrojasmon racemate Propyl dihydrojasmonate,Prohydrojasmon Others
Prohydrojasmon racemate (Propyl dihydrojasmonate) is a synthesized plant gowth regulator, which has jasmonic acid activity.
T50055 Milacemide MAO
Milacemide is a glycine prodrug and MAO-B inhibitor. Milacemide has been studied for its effects on human memory and as a potential treatment for the symptoms of Alzheimer's disease.
T20700 Racemetirosine Others
Racemetirosine is an inhibitor of Tyrosine 3-monooxygenase, and consequently it inhibits the synthesis of catecholamines.
T13331 WAY127093B racemate PDE
WAY127093B racemate is the racemate of WAY127093B. WAY127093B is a phosphodiesterase IV inhibitor with oral activity in rats and guinea pigs.
T22253 AG-120 (racemic) Dehydrogenase
AG-120 (racemic), the racemic mixture of AG-120, is an orally available isocitrate dehydrogenase type 1 (IDH1) inhibitor, and shows potential antineoplastic activity.
T9005 VPC-80051 racemate Others
VPC-80051 is the first small molecule inhibitor of hnRNP A1 splicing activity by using a computer-aided drug discovery approach.
T22988 MK-4827 Racemate Niraparib Racemate,2-(4-piperidin-3-ylphenyl)indazole-7-carboxamide PARP
MK-4827 Racemate (Niraparib Racemate) is a selective PARP1 and PARP2 inhibitor with IC50s of 3.8 nM and 2.1 nM, respectively, over 330-fold selectivity for PARP3, V-PARP and Tank1.
TN1499 Cimiracemoside C Cimicifugoside M AMPK
Cimiracemoside C (Cimicifugoside M) is an active component of Cimicifuga racemosa. It activates AMPK and has the potential activity against diabetes.
T11178L ELN318463 racemate ELN318463 (racemate),ELN 318463 racemate Gamma-secretase
ELN318463 racemate (ELN 318463 racemate) is the racemate of ELN318463 which is an amyloid precursor protein (APP) selective γ-secretase inhibitor.
T6809 CPI-169 racemate CPI 169,CPI-169,CPI169 Epigenetic Reader Domain , Histone Methyltransferase
CPI-169 racemate (CPI 169) is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.

Compounds

Solithromycin
T2331
Synonym: OP-1068,CEM-101
Target: Antibacterial, Antibiotic
CEM114
T39810
Synonym:
Target:
TJ191
T9104
Synonym:
Target: Apoptosis
2-Fluoroadenine
T20038
Synonym: NSC-27364,NSC 27364,NSC27364
Target: DNA/RNA Synthesis
Zosuquidar trihydrochloride
T6018
Synonym: Zosuquidar (LY335979) 3HCl,RS 33295-198 trihydrochloride,RS 33295-198 (D06387) 3HCl,Zosuquidar 3HCl,LY-335979 trihydrochloride
Target: P-gp
Pheniramine maleate
T0370
Synonym: Daneral,Inhiston,Trimetose
Target: 5-HT Receptor, Histamine Receptor
Sertindole
T5858
Synonym: Lu 23-174
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Autophagy
Rentiapril racemate
T16731
Synonym: (Rac)-SA-446,SA-446 racemate,(Rac)-Rentiapril
Target: Angiotensin-converting Enzyme (ACE)
5-MethoxyPinocembroside
T13514
Synonym:
Target: Others
CeMMEC1
T4345
Synonym: CeMMEC1 HCl
Target: Epigenetic Reader Domain, Carboxypeptidase, DNA/RNA Synthesis
Prohydrojasmon racemate
T7220
Synonym: Propyl dihydrojasmonate,Prohydrojasmon
Target: Others
Milacemide
T50055
Synonym:
Target: MAO
Racemetirosine
T20700
Synonym:
Target: Others
WAY127093B racemate
T13331
Synonym:
Target: PDE
AG-120 (racemic)
T22253
Synonym:
Target: Dehydrogenase
VPC-80051 racemate
T9005
Synonym:
Target: Others
MK-4827 Racemate
T22988
Synonym: Niraparib Racemate,2-(4-piperidin-3-ylphenyl)indazole-7-carboxamide
Target: PARP
Cimiracemoside C
TN1499
Synonym: Cimicifugoside M
Target: AMPK
ELN318463 racemate
T11178L
Synonym: ELN318463 (racemate),ELN 318463 racemate
Target: Gamma-secretase
CPI-169 racemate
T6809
Synonym: CPI 169,CPI-169,CPI169
Target: Epigenetic Reader Domain, Histone Methyltransferase
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TargetMol