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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T4093 | Fabomotizole hydrochloride | Afobazole hydrochloride,CM346 hydrochloride | MAO |
Fabomotizole hydrochloride (CM346 hydrochloride), an anxiolytic drug, produces anxiolytic and neuroprotective effects. The mechanism of Afobazole remains poorly defined, however, with GABAergic, NGF, and BDNF release pro... | |||
T4370 | Resminostat hydrochloride | 4SC-201 hydrochloride,RAS2410 hydrochloride | HDAC |
Resminostat hydrochloride (RAS2410 hydrochloride) is an effective inhibitor of HDAC1/HDAC3/HDAC6 (IC50: 42.5/50.1/71.8 nM), respectively, and shows less potent activities against HDAC8 (IC50: 877 nM). | |||
T11872L | LMP744 hydrochloride | NSC706744 hydrochloride,MJ-III65 hydrochloride | Topoisomerase |
LMP744 hydrochloride (NSC-706744 hydrochloride) is a DNA intercalator and Topoisomerase I (Top1) inhibitor with antitumor activity. | |||
T62385 | Befiradol hydrochloride | NLX-112 hydrochloride,F 13640 hydrochloride | 5-HT Receptor |
Befiradol hydrochloride (NLX-112 hydrochloride) is a selective 5-hydroxytryptamine 1A (5-HT)1A receptor agonist with anxiolytic activity.Befiradol hydrochloride inhibits mutant ATXN3 aggregation. | |||
T8769 | Harmaline hydrochloride | Harmidine hydrochloride | Others |
Harmaline hydrochloride (Harmidine hydrochloride) is a fluorescent indole alkaloid from the group of harmala alkaloids and beta-carbolines. It is the partially hydrogenated form of harmine.Harmaline produces a generalize... | |||
T10898 | Samuraciclib hydrochloride | ICEC0942 hydrochloride,CT7001 hydrochloride | Apoptosis , CDK |
Samuraciclib hydrochloride (ICEC0942 hydrochloride) is a potent, selective, ATP competitive and oral active CDK7 inhibitor with IC50 of 41 nM. The selectivity of Samuraciclib hydrochloride is 45-, 15-, 230- and 30-fold h... | |||
T11004 | Desformylflustrabromine hydrochloride | dFBr hydrochloride,Deformylflustrabromine hydrochloride | AChR |
Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.48. | |||
T39740 | Acoramidis hydrochloride | AG10 hydrochloride,Alxn2060 hydrochloride | Others |
Acoramidis hydrochloride (Alxn2060 hydrochloride) is an orally active and selective kinetic stabilizer of WT and V122I- TTR (transthyretin) . Acoramidis hydrochloride is used in the study for transthyretin amyloidosis. | |||
T10221 | Abeprazan hydrochloride | DWP14012 hydrochloride,Fexuprazan hydrochloride | Proton pump |
Abeprazan hydrochloride (Fexuprazan hydrochloride) is an effective reversible potassium-competitive acid blocker with oral activity, inhibiting H+, K+ -atPase by competitive binding to potassium ions without acid activat... | |||
T1053 | Mebeverine hydrochloride | Colofac Hydrochloride,Duspatalin Hydrochloride,Duspatal Hydrochloride | Others , Sodium Channel |
Mebeverine hydrochloride (Colofac Hydrochloride), a β-phenylethylamine derivative, is a potent α1 repector inhibitor, relaxing the muscles in and around the gut. | |||
T4045 | Epetraborole hydrochloride | GSK2251052 hydrochloride | Antibacterial |
Epetraborole hydrochloride (GSK2251052 hydrochloride) is a potent and selective leucyl-tRNA synthetase inhibitor. | |||
T11508L | Camicinal hydrochloride | GSK962040 hydrochloride | Others , Motilin Receptor |
Camicinal hydrochloride (GSK962040 hydrochloride) is a selective agonist of motilin receptor (pEC50 = 7.9). | |||
T13202 | Trilaciclib hydrochloride | G1T28 hydrochloride | CDK |
Trilaciclib hydrochloride (G1T28 hydrochloride) is an inhibitor of CDK4/6 (IC50s: 1 nM and 4 nM for CDK4 and CDK6). | |||
T13302 | Viquidil hydrochloride | Quinotoxine hydrochloride | Others |
Viquidil hydrochloride (Quinotoxine hydrochloride) is an isomer of Quinidine. Viquidil hydrochloride is an agent of cerebral vasodilator with antithrombotic activity. | |||
T12225L | Nevanimibe hydrochloride | PD-132301 hydrochloride,ATR101 hydrochloride | Apoptosis , Acyltransferase |
Nevanimibe hydrochloride (PD-132301 hydrochloride) is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50 of 9 nM). | |||
T2092 | Amitifadine hydrochloride | DOV-21947 hydrochloride,EB-1010 hydrochloride | Dopamine Receptor , 5-HT Receptor , Serotonin Transporter , Norepinephrine |
Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI). | |||
T8617 | GMQ hydrochloride | NSC 403387 hydrochloride | Others |
GMQ hydrochloride (NSC-403387 hydrochloride) is a potent and selective acid-sensing ion channel (ASIC) modulator. It activates ASIC3 channels under neutral pH and blocks acid-induced maximal peak current. | |||
T7000 | Tiagabine hydrochloride | NO328 hydrochloride,NO050328 hydrochloride,TGB hydrochloride,Gabitril,Gabitril hydrochloride | GABA Receptor |
Tiagabine hydrochloride (NO050328 hydrochloride) is the hydrochloride salt form of tiagabine, a nipecotic acid derivative with anticonvulsant property. A selective gamma-aminobutyric acid (GABA) reuptake inhibitor. | |||
T2774 | Lycorine hydrochloride | Licorine hydrochloride,Galanthidine hydrochloride,Narcissine hydrochloride,Lycorine chloride,Amarylline hydrochloride | Virus Protease , HCV Protease , Antibacterial , Autophagy |
Lycorine hydrochloride (Narcissine hydrochloride) is VE-cadherin inhibitor,and has IC50 of 1.2μM in Hey1B cell.It is an HCV inhibitor with strong activity. | |||
T12565 | PRX933 hydrochloride | BVT-933 hydrochloride,GW876167 hydrochloride | 5-HT Receptor |
PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment. |