Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | In stock | $ 839.00 | |
50 mg | 6-8 weeks | $ 1,090.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 318.00 |
Description | Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI). |
Targets&IC50 | serotonin(in HEK 293 cells):12 nM, dopamine(in HEK 293 cells):96 nM, norepinephrine(in HEK 293 cells):23 nM |
Synonyms | DOV-21947 hydrochloride, EB-1010 hydrochloride |
Molecular Weight | 264.58 |
Formula | C11H12Cl3N |
CAS No. | 410074-74-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 10 mM
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Amitifadine hydrochloride 410074-74-7 GPCR/G Protein Neuroscience Norepinephrine Dopamine Receptor 5-HT Receptor Serotonin Transporter inhibit Inhibitor SERT Amitifadine EB1010 Hydrochloride Amitifadine Hydrochloride DOV-21947 hydrochloride EB 1010 DOV 21947 Hydrochloride EB-1010 Hydrochloride DOV21947 DOV 21947 DOV-21947 EB 1010 Hydrochloride SLC6A3 5-HTT EB-1010 hydrochloride EB-1010 DOV-21947 Hydrochloride EB1010 DAT SLC6A4 DOV21947 Hydrochloride Dopamine Transporter inhibitor