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20

Compounds

Cat No. Product Name Synonyms Targets
T8899 Metipranolol Adrenergic Receptor
Metipranolol (Betamann) is a type of β- Adrenergic receptors( β- A potent antagonist of adrenergic receptor on guinea pig atria β 1- Adrenergic receptors and rat uterus β The 2-adrenergic receptor exhibited the beta bloc...
T14960 Chroman 1 ROCK
Chroman 1 is an inhibitor of ROCK2 (IC50: 1 nM).
T6781 Benzenesulfonamide Benzenesulphonamide,Phenyl sulfonamide,Benzosulfonamide Carbonic Anhydrase
Benzenesulfonamide (Benzosulfonamide) ia an inhibitor of carbonic anhydrases.
T6469 Dichlorphenamide Diclofenamide,Daranide,Antidrasi Carbonic Anhydrase
Dichlorphenamide (Diclofenamide) is a carbonic anhydrase inhibitor that is used in the treatment of glaucoma.
T0142 Brinzolamide AL-4862 Carbonic Anhydrase
Brinzolamide (AL-4862) is a Carbonic Anhydrase Inhibitor. The mechanism of action of brinzolamide is as a Carbonic Anhydrase Inhibitor.
T0106 Methazolamide L584601,CL 8490 Carbonic Anhydrase
Methazolamide (CL 8490) is a carbonic anhydrase inhibitor that is used as a diuretic and in the treatment of glaucoma.
T23782 Benzolamide CL-11366,W 1803,CL 11366,CL11366,W-1803 Carbonic Anhydrase
Benzolamide (CL 11366) inhibits carbonic anhydrase effectively and low-threshold calcium currents in hippocampal pyramidal neurons.
TN1540 Cyanidin-3,5-O-diglucoside chloride Others
Cyanidin-3,5-O-diglucoside chloride has antioxidant activity. Cyanidin-3,5-O-diglucoside inhibits hyperbaric pressure-induced GLAST decrease and can be used in glaucoma studies. Cyanidin-3,5-O-diglucoside chloride is eas...
T0445 Promethazine Proazamine,Diphergan CaMK , Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , AChR , Histamine Receptor
Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
T7213 Demecarium bromide BC-48 AChE
Demecarium bromide (BC-48) is a potent cholinesterase inhibitor,and is treatment glaucoma agent.
T6408 Betaxolol Kerlone,SL 75212,Betoptic Adrenergic Receptor
Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
T20743 TG-46 TG46,TG 46 FLT , JAK
TG-46 (TG46) inhibits JAK2, FLT3, RET, JAK3 and can be used to study glaucoma.
T16731 Rentiapril racemate (Rac)-SA-446,SA-446 racemate,(Rac)-Rentiapril Angiotensin-converting Enzyme (ACE)
Rentiapril racemate (SA-446 racemate) is the racemate of Rentiapril.Rentiapril racemate has anti-inflammatory activity and may be used in glaucoma research.
T0103 Dipivefrin hydrochloride Dipivefrin HCL Adrenergic Receptor , AChR
Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
T8580 Bupranolol Adrenergic Receptor
Bupranolol is an antagonist of β2-adrenergic receptor and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.
T1287 Synephrine Oxedrine Endogenous Metabolite , Adrenergic Receptor
Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
T1231 Pilocarpine nitrate Pilagan,Pilofrin AChR
Pilocarpine nitrate (Pilagan) is a slowly hydrolyzed muscarinic agonist with no nicotinic effects. Pilocarpine is used as a miotic and in the treatment of glaucoma.
T16132 MRE3008F20 cAMP , Adenosine Receptor
MRE3008F20 is a species-selective and potent adenosine A3 receptor (AA3R) antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used in glaucoma and asthma studies.CAS 번호13483-88-88-9
T6422 Brimonidine Tartrate AGN190342 tartrate,304 tartrate,AGN190342 (tartrate),UK 14304 (tartrate),UK14304 tartrate Adrenergic Receptor
Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pressure associated with open-angle glaucoma or ocular hyperten...
T2538 Bimatoprost AGN 192024 Prostaglandin Receptor
Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular hypertension.

Compounds

Metipranolol
T8899
Synonym:
Target: Adrenergic Receptor
Chroman 1
T14960
Synonym:
Target: ROCK
Benzenesulfonamide
T6781
Synonym: Benzenesulphonamide,Phenyl sulfonamide,Benzosulfonamide
Target: Carbonic Anhydrase
Dichlorphenamide
T6469
Synonym: Diclofenamide,Daranide,Antidrasi
Target: Carbonic Anhydrase
Brinzolamide
T0142
Synonym: AL-4862
Target: Carbonic Anhydrase
Methazolamide
T0106
Synonym: L584601,CL 8490
Target: Carbonic Anhydrase
Benzolamide
T23782
Synonym: CL-11366,W 1803,CL 11366,CL11366,W-1803
Target: Carbonic Anhydrase
Cyanidin-3,5-O-diglucoside chloride
TN1540
Synonym:
Target: Others
Promethazine
T0445
Synonym: Proazamine,Diphergan
Target: CaMK, Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR, Histamine Receptor
Demecarium bromide
T7213
Synonym: BC-48
Target: AChE
Betaxolol
T6408
Synonym: Kerlone,SL 75212,Betoptic
Target: Adrenergic Receptor
TG-46
T20743
Synonym: TG46,TG 46
Target: FLT, JAK
Rentiapril racemate
T16731
Synonym: (Rac)-SA-446,SA-446 racemate,(Rac)-Rentiapril
Target: Angiotensin-converting Enzyme (ACE)
Dipivefrin hydrochloride
T0103
Synonym: Dipivefrin HCL
Target: Adrenergic Receptor, AChR
Bupranolol
T8580
Synonym:
Target: Adrenergic Receptor
Synephrine
T1287
Synonym: Oxedrine
Target: Endogenous Metabolite, Adrenergic Receptor
Pilocarpine nitrate
T1231
Synonym: Pilagan,Pilofrin
Target: AChR
MRE3008F20
T16132
Synonym:
Target: cAMP, Adenosine Receptor
Brimonidine Tartrate
T6422
Synonym: AGN190342 tartrate,304 tartrate,AGN190342 (tartrate),UK 14304 (tartrate),UK14304 tartrate
Target: Adrenergic Receptor
Bimatoprost
T2538
Synonym: AGN 192024
Target: Prostaglandin Receptor
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TargetMol