available — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T11339	Furegrelate sodium	U-63557A	PPAR
	Furegrelate sodium (U-63557A) is a selective thromboxane synthase inhibitor with oral activity. Furegrelate sodium(U-63557A) inhibits thromboxane A2 (TXA2) synthase in human platelet microsomes with an IC50 of 15 nM.		PPAR
T9865	Almonertinib mesylate		EGFR
	Almonertinib mesylate is an irreversible inhibitor of EGFR tyrosine kinase with high selectivity for EGFR-sensitizing and T790M resistance mutations. Almonertinib mesylate can be used in the non-small cell lung cancer st...		EGFR
TN5073	Strophanthidin	Strophanthidine	ATPase , Calcium Channel
	Strophanthidin (Strophanthidine) can induce calcium overload in vivo.		ATPase , Calcium Channel
T1457	Deferasirox	ICL 670,CGP-72670	Others , Ferroptosis , Antibacterial
	Deferasirox (CGP-72670) is an oral iron chelating agent used to treat chronic iron overload.		Others , Ferroptosis , Antibacterial
T2923	Apremilast	CC-10004	Apoptosis , TNF , PDE
	Apremilast (CC-10004) (CC-10004) is a potent and orally active PDE4 (IC50=74 nM) with anti-inflammation activities.		Apoptosis , TNF , PDE
T16841	SAR-260301		PI3K
	SAR-260301 is an orally available and selective inhibitor of PI3Kβ (IC50: 23 nM).		PI3K
T31668	Eribaxaban	PD 348292,PD0348292,PD-0348292,PD-348292,PD 0348292,PD348292	Factor Xa
	Eribaxaban (PD348292) is an orally available factor Xa inhibitor for the prevention and treatment of venous thromboembolism.		Factor Xa
T15715	LAS101057		Adenosine Receptor
	LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.		Adenosine Receptor
T5368	Eicosapentaenoic Acid		Histone Demethylase , Others , Endogenous Metabolite
	Eicosapentaenoic Acid (EPA) is a ω-3 fatty acid abundantly available in marine organisms.		Histone Demethylase , Others , Endogenous Metabolite
T15423	GSK-7975A		Calcium Channel
	GSK-7975A is a potent and orally available inhibitor of CRAC channel.		Calcium Channel
T27812	Leminoprazole		ATPase
	Leminoprazole is an orally available H+,K(+)-ATPase inhibitor that protects gastric mucosal cells from various cellular damages.		ATPase
T6585	SAR405838	MI773,MI 773,MI-77301,MI-773	Mdm2 , E1/E2/E3 Enzyme
	MI-773 (SAR405838 (MI 773)) is an orally available MDM2 antagonist with Ki of 0.88 nM. Phase 1.		Mdm2 , E1/E2/E3 Enzyme
T13111	Tegadifur	40497S,FD 1	Others
	Tegadifur (40497S) is an orally available antitumor compound with antimetabolic effects, often used with uracil and in the treatment of rectal adenocarcinoma.		Others
TQ0266	MSC2530818		CDK
	MSC2530818 is an effective, selective and orally available CDK8 inhibitor (IC50: 2.6 nM).		CDK
T71394	BMS-823778
	BMS-823778 is an orally available potent and selective inhibitor of 11-β-hydroxysteroid-dehydrogenase 1 (11βHSD-1). BMS-823778 is a potential therapeutic agent for type 2 diabetes mellitus (T2DM).
T26631L	Anidoxime HCl	USVP-E142,Anidoxime HCl( 34297-34-2 Free base)
	Anidoxime HCl (USVP-E142) is a novel orally available compound with anti-analgesic activity.
T33836L	Oxamisole TFA	Oxamisole TFA（99258-56-7 Free base)	Antiviral
	Oxamisole TFA is an orally available T-cell immune repair agent.		Antiviral
T23297	(S)-(+)-Dimethindene maleate		AChR , Histamine Receptor
	(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1, M3, and M4 receptors.		AChR , Histamine Receptor
T39707	AS-1763		BTK
	AS-1763 is an orally available and selective BTK inhibitor with an IC50 of 0.85 nM.		BTK
T15575	Indeglitazar	PPM 204	PPAR
	Indeglitazar (PPM 204) is orally available pan-agonist of PPAR (PPAR subtypes alpha (α), delta (δ), and gamma (γ)).		PPAR