store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
2 mg | In stock | $ 79.00 | |
5 mg | In stock | $ 128.00 | |
10 mg | In stock | $ 222.00 | |
25 mg | In stock | Inquiry | |
50 mg | 5 days | Inquiry | |
1 mL * 10 mM (in DMSO) | In stock | $ 143.00 |
Description | LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma. |
In vivo | At 3 mg/kg, LAS101057 is effective in preventing Acetyl-β-methylcholine-induced airway hyperresponsiveness (AHR), and at 10 mg/kg, it inhibits AHR to Acetyl-β-methylcholine to a level virtually equal to that seen with Hexadecadrol at 1 mg/kg[1]. |
Molecular Weight | 335.34 |
Formula | C18H14FN5O |
CAS No. | 925676-48-8 |
store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (298.20 mM)
H2O: < 0.1 mg/mL (insoluble)
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
LAS101057 925676-48-8 GPCR/G Protein Neuroscience Adenosine Receptor LAS 101057 LAS-101057 inhibitor inhibit