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20

Compounds

Cat No. Product Name Synonyms Targets
TN1148 Isopsoralenoside Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Antibacterial
Isopsoralenoside shows estrogen-like, osteoblastic proliferation accelerating, antitumor, and antibacterial effects.
T26308 Lipoxamycin hemisulfate Lipoxamycin, sulfate (2:1),U-26146D,U26146D,U 26146D,Lipoxamycin Antifungal
Lipoxamycin hemisulfate (Lipoxamycin) is an inhibitor of serine palmitoyltransferase (IC50 = 21 nM) with antifungal activity.
T5666 Dipotassium glycyrrhizinate Virus Protease
Dipotassium glycyrrhizinate is an anionic surfactant having anti-allergic and anti-inflammatory activities.
T11589 Hydroxycitric acid tripotassium hydrate Potassium citrate monohydrate ATP Citrate Lyase , HIF/HIF Prolyl-Hydroxylase , HIF
Hydroxycitric acid tripotassium hydrate (Potassium citrate monohydrate) effectively inhibits stones formation and also inhibits HIF, and has antioxidation, anti-inflammation, and anti-tumor effects. Hydroxycitric acid tr...
TQ0244 Calcipotriol monohydrate
Calcipotriol monohydrate is an analog of Vitamin D3 with a high affinity for the vitamin D receptor. Calcipotriol monohydrate can be used for studies about psoriasis.
T0200 α-Lipoic Acid Thioctic acid,DL-α-Lipoic acid,(±)-α-Lipoic acid Apoptosis , NF-κB , HIV Protease , Mitochondrial Metabolism , Endogenous Metabolite
α-Lipoic Acid (DL-α-Lipoic acid) an octanoic acid bridged with two sulfurs so that it is sometimes also called a pentanoic acid in some naming schemes. It is biosynthesized by cleavage of LINOLEIC ACID and is a coenzyme ...
T67957 Pipoxizine
Pipoxizine has an antagonistic effect on histamine-induced bronchoconstriction and may be used in the study of asthma disease.
T1523 Teniposide NSC 122819,VM26 Topoisomerase
Teniposide (VM26), a semisynthetic derivative of podophyllotoxin with antitumor activity, inhibits DNA synthesis by forming a complex with topoisomerase II and DNA.
T2136 Geniposidic Acid Apoptosis , Others , Endogenous Metabolite
Geniposidic acid, an iridoid glucoside, used in therapy of jaundice, inflammation and hepatic disorders.
T6948 Pluripotin SC1 ERK , Raf , S6 Kinase
Pluripotin (SC1) (SC1), which keep embryonic stem cell (ESC) self-renewal, is a dual inhibitor of extracellular signal-regulated kinase 1 (ERK1, MAPK3) and RasGAP.
T2930 α-Lipoic Acid Lipoic acid,Alphalipoic acid NF-κB , HIV Protease , Mitochondrial Metabolism , Endogenous Metabolite
α-Lipoic Acid (Alphalipoic acid) inhibits NF-κB-dependent HIV-1 LTR activation. α-Lipoic Acid induces endoplasmic reticulum (ER) stress-mediated apoptosis in hepatoma cells.α-Lipoic Acid is an antioxidant, which is an es...
T28419 Pipoxazole COR-3224,COR-32-24,COR 3224. Pipoxazole,COR3224,COR 32-24,COR32-24
Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.
T1745 Balipodect TAK063,TAK-063,TAK 063 PDE
Balipodect (TAK063) is a highly effective and selective PDE10A inhibitor (IC50: 0.30 nM); Its selectivity is >15000-fold over other PDEs.
T2089 Eniporide ATPase
Eniporide is a Na(+)/H(+) exchange inhibitor.
TN7041 (-)-Epipodophyllotoxin Apoptosis
(-)-Epipodophyllotoxin (2) is an antiproliferative agent against cancer cells with GI50s of 0.36 and 0.24 μM in HeLa cells and MCF-7 cells, respectively. (-)-Epipodophyllotoxin can inhibit mitotic spindle assembly in vit...
T77688 Dipotassium tetrachloroplatinate Potassium tetrachloroplatinate Others
Dipotassium tetrachloroplatinate (Potassium tetrachloroplatinate) exhibits antitumor activity in solid tumor lines and can be used in the treatment of oncological diseases. Dipotassium tetrachloroplatinate also acts as a...
T40646 Lipoteichoic acid Complement System
Lipoteichoic acid, a polymer of Staphylococcus aureus cell wall, activates the complement system by inducing C3 and inhibiting CD55, and reduces fat deposition via the IGF-1 pathway.
T21743L Beta-Lipotropin (1-10), porcine Acetate Beta-Lipotropin (1-10), porcine Acetate(77875-68-4 Free base) Others
Beta-Lipotropin (1-10), porcine Acetate (Beta-Lipotropin ) (beta-LPH) was found to contain within its C-terminal sequence the primary structure of these peptides.
T2238 Cariporide HOE-642 Sodium Channel
Cariporide (HOE-642) (HOE-642), an effective NHE1 inhibitor, has inhibitory effects on the degranulation of human platelets, the formation of platelet-leukocyte-aggregates, and the activation of the GPIIb/IIIa receptor (...
T22235 Lipoic acid R-(+)-Thioctic acid,(R)-(+)-1,2-Dithiolane-3-pentanoic acid,(R)-(+)-α-Lipoic acid Reactive Oxygen Species , Mitochondrial Metabolism , Endogenous Metabolite
Lipoic acid (R-(+)-Thioctic acid) is an organosulfur compound derived from octanoic acid. It is made in animals normally, and is essential for aerobic metabolism.

Compounds

Isopsoralenoside
TN1148
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Antibacterial
Lipoxamycin hemisulfate
T26308
Synonym: Lipoxamycin, sulfate (2:1),U-26146D,U26146D,U 26146D,Lipoxamycin
Target: Antifungal
Dipotassium glycyrrhizinate
T5666
Synonym:
Target: Virus Protease
Hydroxycitric acid tripotassium hydrate
T11589
Synonym: Potassium citrate monohydrate
Target: ATP Citrate Lyase, HIF/HIF Prolyl-Hydroxylase, HIF
Calcipotriol monohydrate
TQ0244
Synonym:
Target:
α-Lipoic Acid
T0200
Synonym: Thioctic acid,DL-α-Lipoic acid,(±)-α-Lipoic acid
Target: Apoptosis, NF-κB, HIV Protease, Mitochondrial Metabolism, Endogenous Metabolite
Pipoxizine
T67957
Synonym:
Target:
Teniposide
T1523
Synonym: NSC 122819,VM26
Target: Topoisomerase
Geniposidic Acid
T2136
Synonym:
Target: Apoptosis, Others, Endogenous Metabolite
Pluripotin
T6948
Synonym: SC1
Target: ERK, Raf, S6 Kinase
α-Lipoic Acid
T2930
Synonym: Lipoic acid,Alphalipoic acid
Target: NF-κB, HIV Protease, Mitochondrial Metabolism, Endogenous Metabolite
Pipoxazole
T28419
Synonym: COR-3224,COR-32-24,COR 3224. Pipoxazole,COR3224,COR 32-24,COR32-24
Target:
Balipodect
T1745
Synonym: TAK063,TAK-063,TAK 063
Target: PDE
Eniporide
T2089
Synonym:
Target: ATPase
(-)-Epipodophyllotoxin
TN7041
Synonym:
Target: Apoptosis
Dipotassium tetrachloroplatinate
T77688
Synonym: Potassium tetrachloroplatinate
Target: Others
Lipoteichoic acid
T40646
Synonym:
Target: Complement System
Beta-Lipotropin (1-10), porcine Acetate
T21743L
Synonym: Beta-Lipotropin (1-10), porcine Acetate(77875-68-4 Free base)
Target: Others
Cariporide
T2238
Synonym: HOE-642
Target: Sodium Channel
Lipoic acid
T22235
Synonym: R-(+)-Thioctic acid,(R)-(+)-1,2-Dithiolane-3-pentanoic acid,(R)-(+)-α-Lipoic acid
Target: Reactive Oxygen Species, Mitochondrial Metabolism, Endogenous Metabolite
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TargetMol