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20

Compounds

Cat No. Product Name Synonyms Targets
TN6791 Palvanil Hexadecanamide TRP/TRPV Channel
Palvanil (Hexadecanamide) is a fast desensitizing agonist of TRPV1. it may be promising agents in the therapy of IBS since it modulates intestinal motility and reduces visceral pain.
TN4417 Larixyl acetate Others
Larixyl acetate is a bioactive chemical.
T8959 OS-3-106 Dopamine Receptor
OS-3-106 is a novel arylamide phenylpiperazines, as partial agonists at the D3R in the adenylyl cyclase inhibition assay.
T5345 V-9302 Others
V-9302 (V9302) is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 (IC50: 9.6 uM).
T6759 AP-III-a4 ENOblock Glucokinase
AP-III-a4 (ENOblock) (ENOblock) is the first nonsubstrate analogue inhibitor of enolase with IC50 of 0.576 μM.
T50005 Sertaconazole Antifungal
Sertaconazole is a broad-spectrum antifungal.
T8528 AC1903 TRP/TRPV Channel
AC1903 is a specific inhibitor of TRPC5 channel, and has been shown to suppress severe proteinuria and prevent podocyte loss.
T6848 GSK1016790A GSK101 Calcium Channel , TRP/TRPV Channel
GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial cells.
T0031L2 Ziprasidone Geodon,Zeldox,CP-88059 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Norepinephrine , Histamine Receptor
Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T4478 CID 16020046 C390-0219 Cannabinoid Receptor
CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.
T3520 Setipiprant KYTH-105,ACT-129968 GPR , Prostaglandin Receptor
Setipiprant (ACT-129968) is an orally available, selective CRTH2 antagonist (IC50: 6.0 nM). CRTH2 is a G protein-coupled receptor for prostaglandin (PGD2). PGD2 is produced by the mast cells and is a key mediator in vari...
T6665 Sertaconazole nitrate FI-7045,Ginedermofix,FI7056,Ertaczo Antibiotic , Antifungal
Sertaconazole nitrate (FI-7045), a topical broad-spectrum antifungal, is developed to supply an additional agent for the treatment of superficial cutaneous and mucosal infections.
T0031 Ziprasidone hydrochloride monohydrate CP 88059 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Norepinephrine , Histamine Receptor
Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic activity.
T126184 Khekadaengoside K
Khekadaengoside K is a useful organic compound for research related to life sciences. The catalog number is T126184 and the CAS number is 122738-86-7.
T60523 Agomelatine hydrochloride S-20098 hydrochloride MT Receptor
Agomelatine hydrochloride (S-20098 hydrochloride) (S-20098 hydrochloride) is a specific MT1 and MT2 receptor agonist with Ki of 0.1 nM for CHO-hMT1, 0.06 nM for HEK-hMT1, 0.12 nM for CHO-hMT2, and 0.27 nM for HEK-hMT2, r...
T6934 Pexmetinib ARRY-614 Tie-2 , p38 MAPK , Autophagy
Pexmetinib (ARRY-614) (ARRY-614) is a potent, orally bioavailable, dual p38 MAPK/Tie-2 inhibitor with IC50 of 4 nM/18 nM in a HEK-293 cell line. Phase 1.
T37428 TRPC6-PAM-C20 TRPC6-PAM-C20,3-(6,7-Dimethoxy-3,3-dimethyl-3,4-dihydro-isoquinolin-1-yl)-chromen-2-one TRP/TRPV Channel
TRPC6-PAM-C20 is a selective TRPC6 positive allosteric modulator. TRPC6-PAM-C20 induces transient increase in intracellular Ca2+ in HEK cells expressing TRPC6 with an EC50 of 2.37 μM. TRPC6-PAM-C20 enhances OAG-induced p...
T16569 Praliciguat IW-1973 Others , Guanylate cyclase
Praliciguat (IW-1973) stimulates sGC in HEK-293 cells (EC50: 197 nM). Praliciguat is an effective and orally active soluble guanylate cyclase stimulator. It also enhances NO signaling and acts as a vasodilator.
T11076 Dooku1 Others
Dooku1 is an analog of Yoda1 and a selective antagonist of endogenous Piezo1 channels. Dooku1 inhibits Ca2+ entry induced by 2μMYoda1 with IC50 values of 1.3μM (in HEK 293 cells) and 1.5μM (in HUVEC). Dooku1 inhibits Yod...
T7302 CU-CPT9b CU-CPT-9b,TLR8-specific antagonist 1 TLR
CU-CPT9b (TLR8-specific antagonist 1) is an antagonist of toll-like receptor 8 (TLR8; Kd = 21 nM). It inhibits activation of NF- B induced by the TLR8 agonist R-848 in TLR8-overexpressing HEK-Blue cells with an IC50 valu...

Compounds

Palvanil
TN6791
Synonym: Hexadecanamide
Target: TRP/TRPV Channel
Larixyl acetate
TN4417
Synonym:
Target: Others
OS-3-106
T8959
Synonym:
Target: Dopamine Receptor
V-9302
T5345
Synonym:
Target: Others
AP-III-a4
T6759
Synonym: ENOblock
Target: Glucokinase
Sertaconazole
T50005
Synonym:
Target: Antifungal
AC1903
T8528
Synonym:
Target: TRP/TRPV Channel
GSK1016790A
T6848
Synonym: GSK101
Target: Calcium Channel, TRP/TRPV Channel
Ziprasidone
T0031L2
Synonym: Geodon,Zeldox,CP-88059
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Norepinephrine, Histamine Receptor
CID 16020046
T4478
Synonym: C390-0219
Target: Cannabinoid Receptor
Setipiprant
T3520
Synonym: KYTH-105,ACT-129968
Target: GPR, Prostaglandin Receptor
Sertaconazole nitrate
T6665
Synonym: FI-7045,Ginedermofix,FI7056,Ertaczo
Target: Antibiotic, Antifungal
Ziprasidone hydrochloride monohydrate
T0031
Synonym: CP 88059
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Norepinephrine, Histamine Receptor
Khekadaengoside K
T126184
Synonym:
Target:
Agomelatine hydrochloride
T60523
Synonym: S-20098 hydrochloride
Target: MT Receptor
Pexmetinib
T6934
Synonym: ARRY-614
Target: Tie-2, p38 MAPK, Autophagy
TRPC6-PAM-C20
T37428
Synonym: TRPC6-PAM-C20,3-(6,7-Dimethoxy-3,3-dimethyl-3,4-dihydro-isoquinolin-1-yl)-chromen-2-one
Target: TRP/TRPV Channel
Praliciguat
T16569
Synonym: IW-1973
Target: Others, Guanylate cyclase
Dooku1
T11076
Synonym:
Target: Others
CU-CPT9b
T7302
Synonym: CU-CPT-9b,TLR8-specific antagonist 1
Target: TLR
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TargetMol