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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T60218 | YAP/TAZ inhibitor-2 | YAP | |
YAP/TAZ inhibitor-2 is a potent and orally active TEAD-YAP/TAZ inhibitor with an EC 50 value of 3 nM. YAP/TAZ inhibitor-2 shows anti-proliferative and antitumor activity [1]. | |||
T69760 | TT-10 | TAZ-K | YAP |
TT-10 (TAZ-K), an activator of YES-associated protein (YAP)-transcriptional enhancer factor domain (TEAD) activity, has potential application in heart disease research, specifically for conditions characterized by loss o... | |||
T13364 | YAP/TAZ inhibitor-1 | ROCK | |
YAP/TAZ inhibitor-1 is an inhibitor of YAP/TAZ (IC50 of <0.100 μΜ in firefly luciferase assay). | |||
T9954 | K-975 | Others | |
K-975 is a highly selective, orally active TEAD inhibitor, effectively inhibiting protein-protein interactions between TEAD and YAP1/TAZ. | |||
T12632 | (R)-Mirtazapine | (R)-Org3770,(R)-6-Azamianserin | 5-HT Receptor |
(R)-Mirtazapine ((R)-Org3770) is the R(-)-enantiomer of Mirtazapine, which has anti-injury sensory properties in an animal model of acute thermal hyperalgesia. (R)-Mirtazapine is an antagonist of 5-HT3 receptors and a po... | |||
T68119 | Ontazolast | BIRM-270 | LTR |
Ontazolast is a small molecule leukotriene B4 receptor (LTB4R) antagonist for the treatment of immune system disorders and respiratory diseases.Ontazolast is a candidate compound for the treatment of asthma. | |||
T26986 | Cevoglitazar | LBM-642,LBM 642,LBM642 | PPAR |
Cevoglitazar (LBM-642) is a PPARɑ agonist and PPARγ agonist. Cevoglitazar potently reduces food intake and body weight in obese mice and cynomolgus monkeys. | |||
T27303 | Farglitazar | GI-262570,GI-2570,GW 262570X,GI 262570,GI262570 | PPAR |
Farglitazar (GI-262570) is a PPAR-γ agonist and insulin sensitizer that inhibits stellate cell activation by activating receptor γ via oxidative enzymes proliferators and is used in the study of diabetes. | |||
T7812 | Acitazanolast | MTCC,WP-871 | Others |
Acitazanolast (WP-871) is an anti-allergic drug candidate. | |||
T0201 | Meptazinol hydrochloride | Meptazinol HCl | Opioid Receptor |
Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties. | |||
T1622 | Rosiglitazone maleate | BRL 49653C,BRL 49653 | Ferroptosis , TRP/TRPV Channel , PPAR , Autophagy |
Rosiglitazone maleate (BRL 49653) is the maleate salt of rosiglitazone, an orally-active thiazolidinedione with antidiabetic properties and potential antineoplastic activity. | |||
T1070 | Cefmetazole sodium | Sodium cefmetazole | Antibacterial , Antibiotic |
Cefmetazole sodium (Sodium cefmetazole) is a semisynthetic cephamycin antibiotic with a broad spectrum of activity against both gram-positive and gram-negative microorganisms. It has a high rate of efficacy in many types... | |||
T3085 | Piperacetazine | Psymod,Piperacetazinum,Quide | Dopamine Receptor , 5-HT Receptor |
Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia. | |||
T0214L | Pioglitazone hydrochloride | U-72107E,AD 4833,U 72107A,Pioglitazone HCl | Ferroptosis , PPAR |
Pioglitazone hydrochloride (AD 4833) is the hydrochloride salt of an orally-active thiazolidinedione with antidiabetic properties and potential antineoplastic activity. | |||
T1262 | Tazobactam | Tazobactamum,Tazobactam acid,YTR-830H,CL-298741 | Antibacterial , Antibiotic |
Tazobactam (YTR-830H) is an antibacterial penicillin derivative which inhibits the action of bacterial beta-lactamases. | |||
T22437 | Tazofelone | LY-213829 | Others |
Tazofelone (LY-213829) is a NSAID used for the treatment of inflammatory bowel disease. | |||
T7877 | Thiacetazone | Diazam,Thioacetazone,Neustab,Neotibil | Others , Antibacterial , Antibiotic |
Thiacetazone (Diazam) is a thiosemicarbazone that thioacetazone treatment of pulmonary tuberculosis | |||
T0100 | Atazanavir sulfate | BMS-232632,BMS-232632 sulfate | P450 , SARS-CoV , HIV Protease , P-gp |
Atazanavir sulfate (BMS-232632 sulfate) is an azapeptide and HIV-PROTEASE INHIBITOR that is used in the treatment of HIV INFECTIONS and AIDS in combination with other ANTI-HIV AGENTS. | |||
T0334 | Rosiglitazone | BRL49653 | Ferroptosis , TRP/TRPV Channel , PPAR , Autophagy |
Rosiglitazone (BRL49653) is a PPARγ agonist, TRPC5 activator, and TRPM3 inhibitor with oral activity. Rosiglitazone is also a hypoglycemic agent and a thiazolidinedione insulin sensitizer. | |||
T8599 | Betazole dihydrochloride | Betazole hydrochloride | Histamine Receptor |
Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor. |