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Search Result

Search Results for " gx "

Targets

Sodium Channel

26

Compounds

1

Natural Products

11

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T9647 GX 201 GX-201 Sodium Channel
GX 201 is a selective NaV1.7 inhibitor, IC50 of < 3.2 nM for hNaV1.7.
T27520 GX-395 GX 395
GX-395 is a novel Nav1.7 inhibitor.
T27521 GX-936 GX 936,PF 05196233,PF05196233,GX936,PF-05196233
GX-936, a Nav1.7 inhibitor, inhibits Nav1.7 through a voltage-sensor trapping mechanism, likely by stabilizing inactivated states of the channel.
T22829 GX-674 Sodium Channel
GX-674 is a highly potent and selective voltage-gated sodium channel 1.7 (Nav1.7) antagonist with an IC50 value of 0.1 nM measured at -40 mV for the study of inflammatory and neuropathic pain.
T69915 GX-585
GX-585 is a novel potent inhibitor of NaV1.7 and highly selective against NaV1.5, having limited selectivity against NaV1.1 and NaV1.2.
T1439 Lacidipine SN-305,GX-1048,GR-43659X Apoptosis , Calcium Channel , Reactive Oxygen Species
Lacidipine (SN-305) is a lipophilic dihydropyridine calcium antagonist with an intrinsically slow onset of activity. Due to its long duration of action, lacidipine does not lead to reflex tachycardia. It displays specifi...
T80638 Glycinexylidide GX MEK
Glycinexylidide (GX), the active metabolite of the local anesthetic Lidocaine, exhibits properties significant in inhibiting sodium channels with complex voltage dependence and mitigates the proliferation and spread of g...
T69914 Variegatic acid
Variegatic acid is a natural inhibitor of β-hexosaminidase release and tumor necrosis factor (TNF)-α secretion from rat basophilic leukemia (RBL 2H3) cells, with IC50 values of 10.4 μM and 16.8 μM, respectively, also inh...
T5128 RGX-104 hydrochloride SB742881,RGX-104 HCl Liver X Receptor
RGX-104 hydrochloride (SB742881) is a liver X receptor (LXR) agonist with potential immunomodulating and antineoplastic activities. It modulates innate immunity via transcriptional activation of the ApoE gene.
T7535 RGX-202 β-GPA,3-Guanidinopropionic Acid AMPK , PPAR
RGX-202 (β-GPA) is a creatine analog that alters skeletal muscle energy expenditure. It reduces cellular ATP, creatine, and phosphocreatine levels and stimulates AMP-activated protein kinase (AMPK), activating PPARγ coac...
T2293 SGX-523 Raf , p38 MAPK , c-Met/HGFR , Bcr-Abl
SGX-523 is a selective Met inhibitor (IC50: 4 nM), no inhibitory to Abl, BRAFV599E, p38α, and c-Raf.
T7768 RGX-104 RGX-104 free Acid Liver X Receptor
RGX-104 (RGX-104 free Acid) free Acid is an agonist of potent liver-X nuclear hormone receptor (LXR)
T24873 TGX-115 TGX 115 PI3K
TGX-115 is a cell-permeable and potent inhibitor of the PI 3-K isoform p110β/p110δ (IC50 values of 0.13 μM for p110β and 0.63 μM for p110δ), an enzyme that regulates platelet adhesion and inhibits phosphoinositide (PI) 3...
T2661 TGX-221 TGX221 PI3K
TGX-221, an effective, specific, and cell membrane permeable inhibitor of the PI3K p110β catalytic subunit, is utilized for cancer treatment.
T10268 AGX51 Others
AGX51 is an antagonist of inhibitor of DNA binding (ID) proteins. AGX51 treatment lead to pan-Id degradation, cell cycle arrest, and cell death.
T1813 VGX-1027 VGX1027,VGX 1027,GIT 27 IL Receptor , TNF , Interleukin
VGX-1027 (GIT 27) is an isoxazole compound with various immunomodulatory properties.
TP1531 Guangxitoxin 1E
Guangxitoxin 1E acts as a gating modifier since it shifts the voltage-dependence of Kv2.1 K+ currents towards depolarized potentials.
T28168 NGX-267 AF-267B,AF267B,AF 267B,NGX 267
NGX-267, a muscarinic M1 agonist, is used potentially for the treatment of Xerostomia, Alzheimer's disease and cognitive.
T78352 N-acetylglucosamine-1-P uridyltransferase (AGX1) GlcNAc1pUT
N-acetylglucosamine-1-P uridyltransferase (AGX1) (GlcNAc1pUT) is a bifunctional enzyme that couples with GlcNAc-1-P and UTP to catalyze the synthesis of UDP-GlcNAc through an uridyltransfer reaction. It exhibits acetyltr...
T79034 GXF-111 Epigenetic Reader Domain
GXF-111, a proteolysis targeting chimera (PROTAC) molecule, efficiently induces the selective degradation of the BRD3 and BRD4-L proteins. It exhibits high binding affinities to both BRD3 BD1 and BRD3 BD2, with K i value...
T71581 SGX393
SGX393 is an inhibitor of the CML mutant Bcr-AblT315I, thereby preempting in vitro resistance when combined with nilotinib or dasatinib.
T24874 TGX-155 TGX 155,TGX155
TGX-155 is a selective PI3K inhibitor.
T28095 MrgX1-Activator-1
MrgX1-Activator-1 is a MrgX1 receptor activator.
T74899 GXH-II-052
GXH-II-052 is a potent bivalent inhibitor targeting the bromodomain and extraterminal domain (BET). It exhibits significant binding affinity to various BET proteins, including BRD4-1, BRD4-2, BRD4-T, BRDT-1, BRDT-2, and ...
T63578 Mrgx2 antagonist-1
Mrgx2 antagonist-1 is a potent antagonist of Mrgx2 (Mas-related Gene X2) and can be used to study Mrgx2-mediated diseases and disorders.
T38446 ROC-0929
ROC-0929 (compound 13a) is a potent and selective inhibitor of secreted phospholipases A2 (sPLA2s), effectively targeting hGX with an IC50 of 80 nM. It efficiently inhibits the phosphorylation of ERK1/2 and p-38. sPLA2s,...
Cat No. Product Name Synonyms Targets
TN5881 4′-O-Isobutyroylpeguangxienin
4′-O-Isobutyroylpeguangxienin is a natural product for research related to life sciences. The catalog number is TN5881 and the CAS number is 2188162-95-8.

Natural Products

4′-O-Isobutyroylpeguangxienin
TN5881
Synonym:
Target:

Recombinant Proteins

Species：
H10N8 (3)
Human (3)
H1N2 (2)
H5N6 (2)
H1N1 (1)
Expression System：
HEK293 Cells (6)
Baculovirus Insect Cells (4)
E. coli (1)
Tag：
C-His (4)
His (4)
N-His (1)
N-hFc (1)
Tag Free (1)
Cat No. Product Name Species Expression System
TMPY-04965 B3GALT5 Protein, Human, Recombinant (His) Human Baculovirus Insect Cells
B3GALT5 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 35.2 kDa and the accession number is Q9Y2C3.
TMPY-04071 B3GALT5 Protein, Human, Recombinant (hFc) Human HEK293 Cells
B3GALT5 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 61.3 kDa and the accession number is Q9Y2C3.
TMPY-02439 Rac2 Protein, Human, Recombinant (His) Human E. coli
Ras-related C3 botulinum toxin substrate 2 (Rac2) is a small G-protein belonging to the Ras subfamily of the GTPase family. Rac2 acts as an "on / off" switch for signal transduction cascades and motilities. When GDP is a...
TMPY-02662 Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA Protein (His) H10N8 Baculovirus Insect Cells
Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.9 kDa.
TMPY-00416 Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA0 Protein H10N8 Baculovirus Insect Cells
Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA0 Protein is expressed in Baculovirus insect cells. The predicted molecular weight is 60.6 kDa.
TMPY-05934 Influenza A H1N1 (A/swine/Guangxi/NS2176/2012) Neuraminidase/NA Protein (His) H1N1 HEK293 Cells
Influenza A H1N1 (A/swine/Guangxi/NS2176/2012) Neuraminidase/NA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50.5 kDa and the accession number is A0A075ESB5.
TMPY-04326 Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA1 Protein (His) H10N8 HEK293 Cells
Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 36.9 kDa.
TMPY-01513 Influenza A H1N2 (A/swine/Guangxi/13/2006) Hemagglutinin/HA Protein (His) H1N2 HEK293 Cells
Influenza A H1N2 (A/swine/Guangxi/13/2006) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is A5JQC7.
TMPY-04599 Influenza A H5N6 (A/duck/Jiangxi/95/2014) Hemagglutinin/HA1 Protein (His) H5N6 HEK293 Cells
Influenza A H5N6 (A/duck/Jiangxi/95/2014) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38.9 kDa.
TMPY-04901 Influenza A H5N6 (A/duck/Jiangxi/95/2014) Hemagglutinin/HA Protein (His) H5N6 Baculovirus Insect Cells
Influenza A H5N6 (A/duck/Jiangxi/95/2014) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 60.2 kDa.
TMPY-01514 Influenza A H1N2 (A/swine/Guangxi/13/2006) Hemagglutinin/HA1 Protein (His) H1N2 HEK293 Cells
Influenza A H1N2 (A/swine/Guangxi/13/2006) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession number is A5JQC7.
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