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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T3041 | ALK inhibitor 2 | FAK , ALK | |
ALK inhibitor 2 is a new-type and selective inhibitor for the ALK kinase. | |||
T10285 | ALK inhibitor 1 | FAK , IGF-1R , ALK | |
ALK inhibitor 1 is a selective ALK kinase inhibitor. | |||
T23483 | U 99194 maleate | U-99194A maleate,U-99194 maleate salt,U-99194 maleate | Dopamine Receptor |
U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice. | |||
T6486 | Enalapril Maleate | MK-421 Maleate,Renitec Maleate,Glioten Maleate,MK-421 (maleate),Vasotec Maleate | RAAS |
Enalapril Maleate (MK-421 Maleate), an angiotensin-converting enzyme (ACE) inhibitor, is utilized in the treatment of hypertension, chronic heart failure , and diabetic nephropathy. | |||
T1951 | Asenapine Maleate | Org 5222 maleate,Org 5222 | 5-HT Receptor |
Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually and used in the treatment of schizophrenia and manic or mixed episodes associated with bipolar 1 disor... | |||
T2222 | Carbinoxamine Maleate Salt | Lergefin,CarbinoxaMine Maleate | Histamine Receptor |
Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties. | |||
T22520 | 5-Carboxamidotryptamine maleate | 5-CT maleate | 5-HT Receptor |
5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects. | |||
T20911 | Dibutyl maleate | AI3-00644,Butyl maleate,DBM (VAN) | Others |
Dibutyl maleate (DBM (VAN)) is a diester of the Maleic Acid and can be used as an intermediate of the synthesis of antibacterial compounds. | |||
T4422 | Edonerpic maleate | T-817MA,T-817 maleate | Beta Amyloid |
Edonerpic maleate (T-817 maleate) is a neurotrophic agent which can inhibit amyloid-β peptides (Aβ). | |||
T67385 | Neratinib maleate | HKI-272 maleate | EGFR , HER |
Neratinib maleate (HKI-272 maleate) is an irreversible, orally active and highly selective inhibitor of HER2 and EGFR with IC50 values of 59 nM and 92 nM, respectively.Neratinib maleate has antitumor activity and can be ... | |||
T21556 | Hydroxytacrine maleate | Velnacrine maleate,HP 029 maleate | AChE |
Hydroxytacrine maleate (Velnacrine maleate) is a cholinesterase (cholinesterase) inhibitor that enhances memory in rodents and may be used in the study of Alzheimer's dementia of the Alzheimer type (SDAT). | |||
T3435 | Vicriviroc maleate | SCH-D (maleate),SCH-417690 (maleate) | HIV Protease , CCR |
Vicriviroc maleate (SCH-417690 (maleate))(Sch-417690) is a piperazine-based CCR5 receptor antagonist with activity against human immunodeficiency virus. The IC50 value is 0.91 nM in clinical development for the treatment... | |||
T17285 | Zatosetron maleate | LY 277359 maleate | 5-HT Receptor |
Zatosetron maleate(LY 277359 maleate) is a potent and selective serotonin 5HT3 receptor antagonist for the study of acute migraine. | |||
T0236 | Azatadine dimaleate | SCH10649,Azatadine Maleate | 5-HT Receptor , AChR , Histamine Receptor |
Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM). | |||
T3721 | Avitinib maleate | EGFR | |
Avitinib maleate is a pyrrolopyrimidine-based irreversible epidermal growth factor receptor (EGFR) inhibitor. | |||
T10232 | Acetophenazine dimaleate | Dopamine Receptor | |
Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor. | |||
T0368 | Cinepazide maleate | MD-67350,Vasodistal,Brendil | Calcium Channel |
Cinepazide maleate (MD-67350), a maleate salt form of cinepazide, is a vasodilator. | |||
T9306 | EST64454 Maleic acid salt | Others | |
EST64454 Maleic acid salt is the maleic acid salt form of EST64454.EST64454 is a highly soluble σ1 receptor antagonist clinical candidate for the treatment of pain. | |||
T1239 | Indacaterol maleate | QAB149 | Adrenergic Receptor |
Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist. | |||
T6914 | Oclacitinib maleate | PF-03394197 maleate,PF-03394197 | Tyrosine Kinases , JAK |
Oclacitinib maleate (PF-03394197 maleate) is a novel inhibitor of JAK family members with IC50 ranging from 10 to 99 nM and JAK1-dependent cytokines with IC50 ranging from 36 to 249 nM, which did not inhibit a panel of 3... |