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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T13884 | Shield-1 | Others | |
Shield-1 is a specific, high-affinity and cell-permeant ligand of FK506-binding protein-12 (FKBP), and reverses the instability by binding to mutated FKBP (mtFKBP), allowing conditional expression of mtFKBP-fused protein... | |||
T6054 | GSK256066 | PDE | |
GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380, 000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7.Phase 2. | |||
T26085 | Rilapine | Rilapinum | |
Rilapine is an atypical antipsychotic with high affinity for the 5-HT6 receptor. | |||
T31362 | Deferitazole | SPD602,FBS 0701,SPD-602,FBS0701,FBS-0701,SPD 602 | Others |
Deferitazole (FBS 0701) is a novel and orally active, selective and high affinity iron chelator. | |||
T20761 | RU 59063 | RU-59063,RU59063 | Androgen Receptor |
RU 59063 is a prototype of a new class of high-affinity nonsteroidal androgen receptor (AR) ligands. | |||
T34383 | Rofleponide | Glucocorticoid Receptor | |
Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor. | |||
T2229 | Tetraethylenepentamine Pentahydrochloride | Others | |
Tetraethylenepentamine Pentahydrochloride is a high affinity copper and zinc chelator. | |||
T15581 | Inolitazone | RS5444,Efatutazone,CS-7017 | PPAR |
Inolitazone (RS5444) a high-affinity PPARγ agonist. Inolitazone exhibits IC50 for growth inhibition is ~0.8 nM in vitro. | |||
T6333 | MM-102 | MM102,HMTase Inhibitor IX | Histone Methyltransferase |
MM-102 (HMTase Inhibitor IX) is a high-affinity peptidomimetic MLL1 inhibitor with IC50 of 0.4 μM. | |||
T11864 | Iptacopan | LNP023 | Others |
Iptacopan (LNP023) is an inhibitor with high affinity for factor B. | |||
T3497 | Ocaperidone | Ocaperidona,R79598 | Dopamine Receptor , 5-HT Receptor |
Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist. | |||
T2126 | MK-5046 | Bombesin Receptor | |
MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM). | |||
T9501 | Enterobactin | Enterochelin | Others |
Enterobactin (Enterochelin) is a high-affinity siderophore that acquires iron for microbial systems. | |||
TP1957L | PKI (5-24) Acetate(99534-03-9 free base) | PKA | |
PKI (5-24) Acetate is a high affinity PKA inhibitor (Ki = 2.3 nM). | |||
T7716 | TNCA | Lycoperodine-1 | Others |
TNCA (Lycoperodine-1) is a high-affinity CaSR ligand (CaSRL) with co-agonist activity. | |||
TP1044L | Pancreatic Polypeptide, rat acetate | Neuropeptide Y Receptor | |
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4. | |||
T15364 | G-1 | Estrogen Receptor/ERR , GPR | |
G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM). | |||
T11349 | GABAA receptor agent 1 | GABA Receptor | |
GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor. | |||
T3347 | PF3274167 | PF 3274167,Cligosiban,PF-3274167 | OX Receptor |
PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist. | |||
T11758L | KI696 | Nrf2 | |
KI696 is a high-affinity probe that potently inhibits the interaction of Keap1 and NRF2. |