Home Tools
Log in
Cart

Search Result

Search Results for " high-affinity "

20

Compounds

Cat No. Product Name Synonyms Targets
T13884 Shield-1 Others
Shield-1 is a specific, high-affinity and cell-permeant ligand of FK506-binding protein-12 (FKBP), and reverses the instability by binding to mutated FKBP (mtFKBP), allowing conditional expression of mtFKBP-fused protein...
T6054 GSK256066 PDE
GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380, 000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7.Phase 2.
T26085 Rilapine Rilapinum
Rilapine is an atypical antipsychotic with high affinity for the 5-HT6 receptor.
T31362 Deferitazole SPD602,FBS 0701,SPD-602,FBS0701,FBS-0701,SPD 602 Others
Deferitazole (FBS 0701) is a novel and orally active, selective and high affinity iron chelator.
T20761 RU 59063 RU-59063,RU59063 Androgen Receptor
RU 59063 is a prototype of a new class of high-affinity nonsteroidal androgen receptor (AR) ligands.
T34383 Rofleponide Glucocorticoid Receptor
Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.
T2229 Tetraethylenepentamine Pentahydrochloride Others
Tetraethylenepentamine Pentahydrochloride is a high affinity copper and zinc chelator.
T15581 Inolitazone RS5444,Efatutazone,CS-7017 PPAR
Inolitazone (RS5444) a high-affinity PPARγ agonist. Inolitazone exhibits IC50 for growth inhibition is ~0.8 nM in vitro.
T6333 MM-102 MM102,HMTase Inhibitor IX Histone Methyltransferase
MM-102 (HMTase Inhibitor IX) is a high-affinity peptidomimetic MLL1 inhibitor with IC50 of 0.4 μM.
T11864 Iptacopan LNP023 Others
Iptacopan (LNP023) is an inhibitor with high affinity for factor B.
T3497 Ocaperidone Ocaperidona,R79598 Dopamine Receptor , 5-HT Receptor
Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.
T2126 MK-5046 Bombesin Receptor
MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).
T9501 Enterobactin Enterochelin Others
Enterobactin (Enterochelin) is a high-affinity siderophore that acquires iron for microbial systems.
TP1957L PKI (5-24) Acetate(99534-03-9 free base) PKA
PKI (5-24) Acetate is a high affinity PKA inhibitor (Ki = 2.3 nM).
T7716 TNCA Lycoperodine-1 Others
TNCA (Lycoperodine-1) is a high-affinity CaSR ligand (CaSRL) with co-agonist activity.
TP1044L Pancreatic Polypeptide, rat acetate Neuropeptide Y Receptor
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.
T15364 G-1 Estrogen Receptor/ERR , GPR
G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
T11349 GABAA receptor agent 1 GABA Receptor
GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.
T3347 PF3274167 PF 3274167,Cligosiban,PF-3274167 OX Receptor
PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.
T11758L KI696 Nrf2
KI696 is a high-affinity probe that potently inhibits the interaction of Keap1 and NRF2.
1 2 3 4 5 ... 34
TargetMol