racemate — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T11178L	ELN318463 racemate	ELN318463 (racemate),ELN 318463 racemate	Gamma-secretase
	ELN318463 racemate (ELN 318463 racemate) is the racemate of ELN318463 which is an amyloid precursor protein (APP) selective γ-secretase inhibitor.		Gamma-secretase
T7359	CAY10471 Racemate	TM30089 Racemate	GPR , Prostaglandin Receptor
	CAY10471 Racemate (TM30089 Racemate) is a potent, highly selective CRTH2/DP 2 receptor antagonist. CAY10471 Racemate binds to the human CRTH2/DP2, DP1, and TP receptors( Ki values of 0.6, 1200, and >10,000 nM,respectivel...		GPR , Prostaglandin Receptor
T10591	BPO-27 racemate	BPO-27 (racemate)	CFTR , Autophagy
	BPO-27 racemate (BPO-27 (racemate)) is an effective CFTR inhibitor with IC50 of 8 nM.		CFTR , Autophagy
T10464L	Atuveciclib Racemate	BAY-1143572 Racemate	CDK
	Atuveciclib Racemate (BAY-1143572 Racemate) is the racemate mixture of Atuveciclib, which is a potent and highly selective, oral P-TEFb/CDK9 inhibitor which supresses CDK9/CycT1 with an IC50 of 13 nM.		CDK
T7504	Necrostatin 2 racemate	Necrostatin-2 racemate	RIP kinase
	Necrostatin 2 racemate (Necrostatin-2 racemate) is an potent and specific inhibitor of RIPK1.		RIP kinase
T12400	Peliglitazar racemate	(Rac)-Peliglitazar,(Rac)-BMS 426707-01,BMS 426707-01 racemate	PPAR
	Peliglitazar racemate(BMS 426707-01 racemate) is the racemate of Peliglitazar.Peliglitazar racemate may be used as a potential antidiabetic and anti-obesity agent.		PPAR
T16731	Rentiapril racemate	(Rac)-SA-446,SA-446 racemate,(Rac)-Rentiapril	Angiotensin-converting Enzyme (ACE)
	Rentiapril racemate (SA-446 racemate) is the racemate of Rentiapril.Rentiapril racemate has anti-inflammatory activity and may be used in glaucoma research.		Angiotensin-converting Enzyme (ACE)
T3534	Tetrabenazine Racemate	Nitoman,Ro 1-9569 Racemate,Rubigen,TETRABENAZINE	Monoamine Transporter
	Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2). Tetrabenazine Racemate blocks neurotransmitter uptake into adrenergic storage vesicles and has been ...		Monoamine Transporter
T22988	MK-4827 Racemate	Niraparib Racemate,2-(4-piperidin-3-ylphenyl)indazole-7-carboxamide	PARP
	MK-4827 Racemate (Niraparib Racemate) is a selective PARP1 and PARP2 inhibitor with IC50s of 3.8 nM and 2.1 nM, respectively, over 330-fold selectivity for PARP3, V-PARP and Tank1.		PARP
T2344L	LY 344864 racemate		5-HT Receptor
	LY 344864 racemate is a 5-HT1F receptor agonist.		5-HT Receptor
T12215	Nexopamil racemate	(Rac)-Nexopamil	Calcium Channel , 5-HT Receptor
	Nexopamil racemate（(Rac)-Nexopamil） is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.		Calcium Channel , 5-HT Receptor
T13331	WAY127093B racemate		PDE
	WAY127093B racemate is the racemate of WAY127093B. WAY127093B is a phosphodiesterase IV inhibitor with oral activity in rats and guinea pigs.		PDE
T6425	BTZ043 Racemate	BTZ044,BTZ10526038,Benzothiazinone 10526038	Antibacterial , DprE1
	BTZ043 Racemate (Benzothiazinone 10526038) is a decaprenylphosphoryl-β-D-ribose 2'-epimerase (DprE1) inhibitor, used as a new antimycobacterial agent.		Antibacterial , DprE1
T9005	VPC-80051 racemate		Others
	VPC-80051 is the first small molecule inhibitor of hnRNP A1 splicing activity by using a computer-aided drug discovery approach.		Others
T7220	Prohydrojasmon racemate	Propyl dihydrojasmonate,Prohydrojasmon	Others
	Prohydrojasmon racemate (Propyl dihydrojasmonate) is a synthesized plant gowth regulator, which has jasmonic acid activity.		Others
T6809	CPI-169 racemate	CPI 169,CPI-169,CPI169	Epigenetic Reader Domain , Histone Methyltransferase
	CPI-169 racemate (CPI 169) is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.		Epigenetic Reader Domain , Histone Methyltransferase
T5054	GSK963	GSK963 (Racemate)	RIP kinase
	GSK963 (Racemate), a structurally distinct, potent and selective inhibitor of RIP1 kinase(IC50=29 nM).		RIP kinase
T3449	Bay 41-4109 racemate		HBV
	BAY 41-4109 racemate is a potent inhibitor of human hepatitis B virus (HBV) with an IC50 of 53 nM.		HBV
T72753	RSV604 racemate	A-60444 racemate
	RSV604 (A-60444) racemate, a racemic mixture, exhibits lower potency against strains of respiratory syncytial virus (RSV) compared to its S-isomer.
T13293	Veledimex racemate	RG-115932 racemate,INXN-1001 racemate	Others
	Veledimex racemate, the racemic form of veledimex, is an orally available, small-molecule ligand that activates the RheoSwitch Therapeutic System.		Others