non-peptide — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T83671	CCP-biotin Peptide (non-cyclized)	Citrullinated Filaggrin (Q447H, S449C, G459R, E460G, S462C) (R455) (447-467)-biotin Peptide (non-cyclized),Cyclic Citrullinated Peptide-biotin Peptide (non-cyclized)
	CCP-biotin peptide (non-cyclized) is a linear, biotin-labeled derivative of the circular citrullinated peptide (CCP), mirroring the human filaggrin sequence from amino acids 447 to 467 with specific substitutions (Q447H,...
T3474	RO 46-8443		Endothelin Receptor
	RO 46-8443 is the first non-peptide endothelin ETB receptor selective antagonist. RO 46-8443 displays up to 2000-fold selectivity for ETB receptors both in terms of binding inhibitory potency and functional inhibition.		Endothelin Receptor
T2561	Macitentan	ACT-064992	Apoptosis , Endothelin Receptor
	Macitentan (ACT-064992) is an endothelin receptor antagonist that is used in the therapy of pulmonary arterial hypertension (PAH).		Apoptosis , Endothelin Receptor
TP1253	Argireline	Acetyl hexapeptide-3	Others
	Argireline (Acetyl hexapeptide-3) (Acetyl hexapeptide-3) is composed of chains of amino acids known as peptides. Argireline significantly inhibits Ca2+ dependent neurotransmitter release (acetylcholine) at the neuromuscu...		Others
T12895	SHA 68		Neuropeptide Y Receptor
	SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR)(NPSR Asn107 and NPSR Ile107 with IC50s of 22.0 and 23.8 nM, respectively).		Neuropeptide Y Receptor
TP2204L	CCK Octapeptide, non-sulfated acetate	CCK Octapeptide, non-sulfated acetate(25679-24-7 Free base)	cholecystokinin
	CCK Octapeptide, non-sulfated acetate is a synthetic desulfated peptide of cholecystokinin.		cholecystokinin
T26645	Aptiganel	CNS 1102,CNS-1102,CNS1102	NMDAR
	Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.		NMDAR
T4355	Fuscoside	OPC 21268	Vasopressin Receptor
	Fuscoside (OPC 21268) is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.		Vasopressin Receptor
T2537	Tirofiban hydrochloride monohydrate	Tirofiban Hydrochloride,MK-383 Hydrochloride	ATPase , Integrin
	Tirofiban hydrochloride monohydrate (MK-383 Hydrochloride) is a potent non-peptide, glycoprotein IIb/IIIa (integrins alphaIIbbetaIII) antagonist.		ATPase , Integrin
T12293L	Olcegepant	BIBN-4096,BIBN 4096BS	CGRP Receptor
	Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP).		CGRP Receptor
T2375	BX471	BX 471,BX-471,ZK-811752	CCR
	BX471 (BX 471) is a potent, selective non-peptide CCR1 antagonist.		CCR
TP1046	SLIGRL-NH2	Protease-Activated Receptor-2 Activating Peptide	Protease-activated Receptor
	SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a protease-activated receptor-2 (PAR-2) agonist that induces non-histaminergic pruritus.		Protease-activated Receptor
T68068L	(R)-CJ 11974		Neurokinin receptor
	(R)-CJ 11974 is a novel non-peptide neurokinin NK1 substance P receptor antagonist with potential analgesic activity that can be used to study chemotherapy-induced vomiting.		Neurokinin receptor
T35233	Y-29794 Tosylate	Y 29794,Y29794 tosylate,Y29794,Y-29794	Prolyl Endopeptidase (PREP)
	Y-29794 Tosylate (Y-29794) is an orally active, effective, and specific non-peptide-prolyl endopeptidase (PPCE) inhibitor.		Prolyl Endopeptidase (PREP)
T4540	ML-18		Bombesin Receptor
	ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.		Bombesin Receptor
T6658	SB-408124		OX Receptor
	SB408124 is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.		OX Receptor
T7112	Ibutamoren Mesylate	MK-0677,MK-677	GHSR
	Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.		GHSR
T8559	Galnon TFA(475115-35-6(free base))		Neuropeptide Y Receptor
	Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 and 34.1 μM respectively).		Neuropeptide Y Receptor
T69140	Burapitant	SSR 240600	Neurokinin receptor
	Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity.		Neurokinin receptor
T5048	SSR240612		Bradykinin Receptor
	SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors, respectively).		Bradykinin Receptor