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Aptiganel

Catalog No. T26645 CAS 137159-92-3

Synonyms: CNS 1102, CNS-1102, CNS1102

Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Aptiganel, CAS 137159-92-3

Pack Size	Availability	Price/USD
1 mg	In stock	$ 293.00
5 mg	In stock	$ 722.00
10 mg	In stock	$ 987.00
25 mg	In stock	$ 1,520.00
50 mg	6-8 weeks	$ 1,980.00
100 mg	6-8 weeks	$ 2,500.00

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Purity: 98.19%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.

Synonyms	CNS 1102, CNS-1102, CNS1102
Molecular Weight	303.4
Formula	C20H21N3
CAS No.	137159-92-3

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Kroppenstedt SN, et al. Neuroprotective properties of aptiganel HCL (Cerestat) following controlled cortical impact injury. Acta Neurochir Suppl. 1998;71:114-116. 2. McBurney RN. Development of the NMDA ion-channel blocker, aptiganel hydrochloride, as a neuroprotective agent for acute CNS injury. Int Rev Neurobiol. 1997;40:173-195. 3. Kroppenstedt SN,et al. Protective effects of aptiganel HCl (Cerestat) following controlled cortical impact injury in the rat. J Neurotrauma. 1998 Mar;15(3):191-7. 4. Bokesch PM, et al. Immediate-early gene expression in ovine brain after hypothermic circulatory arrest: effects of aptiganel. Ann Thorac Surg. 1997 Oct;64(4):1082-7; discussion 1088.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Aptiganel 137159-92-3 Neuroscience NMDAR CNS 1102 CNS-1102 CNS1102 Cerestat inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.