inhibition — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T5637	Triflumuron		Others
	Triflumuron is an insecticide belonging to the group of so-called insect growth regulators. It inhibits the synthesis of chitin by the insect larvae, causing the die.		Others
T5722	Nevadensin	Pedunculin	Anti-infection , Antibacterial
	Nevadensin is an important herb-based constituent inhibiting estragole bioactivation. Nevadensin protects against a methyleugenol-induced marker of hepatocarcinogenicity in male F344 rat. It also exhibits inhibition acti...		Anti-infection , Antibacterial
T8794	4-MMPB	15-Lipoxygenase Inhibitor 1	Apoptosis , Others , Lipoxygenase
	15-Lipoxygenase Inhibitor 1 is a selective inhibitor of 15-lipoxygenase, with an IC50 of 18 μM. 4-MMPB (15-Lipoxygenase Inhibitor 1) has IC50s of 19.5 μM and 19.1 μM for soybean 15-lipoxygenase (SLO) and human 15-lipoxyg...		Apoptosis , Others , Lipoxygenase
T5S0384	Rhapontin	Ponticin,Rhaponiticin,Rhaponticin,Rhapontigenin glucoside	Apoptosis , Others
	1. Rhapontin (Ponticin) can alleviate liver steatosis and improve blood glucose and lipid profiles in KK/Ay diabetic mice, indicates that rhaponticin has a noticeable antidiabetic effect and could be potentially used as ...		Apoptosis , Others
T14496	BAMB-4	ITPKA-IN-C14	Others
	BAMB-4 (ITPKA-IN-C14) is a highly membrane-permeable inhibitor of inositol-1,4,5-trisphosphate-3-kinase A (ITPKA). It acts by suppressing the metastasis-promoting effect of ITPKA in lung tumor cells(with IC50 of 37 μM in...		Others
T22733	DL-AP5		NMDAR
	DL-AP5 is a NMDA antagonist.		NMDAR
T60080	TMPH	2,2,6,6-Tetramethylpiperidin-4-yl heptanoate	AChR
	TMPH is an inhibitor of nAChR and inhibits nAChRs lacking α5, α6, or β3 subunits. TMPH can be used in studies about nAChR dysfunction or neurological disorders.		AChR
T1465	Mupirocin	Pseudomonic acid,BRL-4910A	DNA/RNA Synthesis , Antibacterial , Antibiotic
	Mupirocin (BRL-4910A) is a RNA synthetase inhibitor antibacterial. It has shown excellent activity against gram-positive staphylococci and streptococci.		DNA/RNA Synthesis , Antibacterial , Antibiotic
T2691	Oritavancin diphosphate	LY333328 diphosphate	Others , Antibacterial , Antibiotic
	Oritavancin diphosphate (LY333328 diphosphate) is a novel semisynthetic glycopeptide antibiotic which is being developed for the treatment of serious Gram-positive bacterial infections.		Others , Antibacterial , Antibiotic
T8148	Mupirocin calcium hydrate	Mupirocin calcium	Others , Antibacterial , Antibiotic
	Mupirocin calcium hydrate is an antibiotic produced by Pseudomonas fluorescens, showed a high level of activity against staphylococci and streptococci and against certain gram-negative bacteria		Others , Antibacterial , Antibiotic
T2051	SKLB4771	FLT3-IN-1,FLT3-IN-1	FLT
	SKLB4771 (FLT3-IN-1) is a novel potent and selective Flt3 inhibitor.		FLT
T7476	AS057278	3-Methylpyrazole-5-carboxylic acid	Others
	AS057278 (3-Methylpyrazole-5-carboxylic acid) is an D-amino acid oxidase (DAAO) inhibitor.		Others
T0171	Norethynodrel	Lynestrol	Estrogen/progestogen Receptor
	Norethynodrel (Lynestrol) is a synthetic progestational hormone with actions and uses similar to those of PROGESTERONE. It has been used in the treatment of functional uterine bleeding and endometriosis. As a contracepti...		Estrogen/progestogen Receptor
T10886	Crocetine dimethyl ester	Dimethylcrocetin	Antioxidant
	Crocetine dimethyl ester (Dimethylcrocetin) is a saffronin derivative with antioxidant activity, inhibition of AChE activity, and inhibition of cell growth and differentiation.		Antioxidant
T3880	Silydianin	Silidianin	Phosphatase
	Silydianin (Silidianin) exerts inhibition of UGT in human liver. Silydianin exerts inhibition of OATP1B1, OATP1B3 (unknown origin) expressed in HEK293 cells. Silydianin exerts inhibition of OATP2B1 (unknown origin) expre...		Phosphatase
T3899	Calceolarioside B	Desrhamnosyl isoacteoside,Nuomioside A	Aromatase
	Calceolarioside B (Desrhamnosyl isoacteoside) displays inhibition of aromatase. Calceolarioside B displays inhibition of human recombinant PKCalpha.		Aromatase
T3817	Darutigenol		Others
	Darutigenol has obvious antithrombotic effect, its mechanism may be related to inhibition of platelet aggregation and adhesion.		Others
T23284	Ryuvidine		Histone Demethylase , Histone Methyltransferase , CDK
	Ryuvidine is a dual inhibitor of KDM5A and SETD8, an inducer of the DNA damage response with potential anticancer activity, inhibition of H4K20 methylation, and inhibition of CDK4, and can be used to study breast cancer ...		Histone Demethylase , Histone Methyltransferase , CDK
T3401	Ginsenoside F1	20(S)-Ginsenoside F1	P450 , Endogenous Metabolite
	Ginsenoside F1 (20(S)-Ginsenoside F1) is an enzymatically modified derivative of ginsenoside Rg1, showing competitive inhibition of the activity of CYP3A4 and a weaker inhibition of the activity of CYP2D6.		P450 , Endogenous Metabolite
TN3460	Asebogenin		Antifungal
	Asebogenin is a compound fractionated from Salvia miltiorrhiza with antifungal activity, inhibition of GPVI-induced platelet reactions, and inhibition of NET formation induced by pro-inflammatory stimuli.		Antifungal