20
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T1009 | Estrone | Oestrone,Fluoroethyl,Aquacrine | Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite |
Estrone (Aquacrine) is an aromatized C18 steroid with a 3-hydroxyl group and a 17-ketone, a major mammalian estrogen. It is converted from ANDROSTENEDIONE directly, or from TESTOSTERONE via ESTRADIOL. In humans, it is pr... | |||
T12581 | Puerarin-4'-O-β-D-glucopyranoside | Puerarin4'-O-glucoside | Others |
Puerarin-4'-O-β-D-glucopyranoside (Puerarin4'-O-glucoside) is a natural product isolated from Pueraria lobata root having estrogenic activity and anti-proliferation in MCF-7 human breast carcinoma cells. | |||
T9454 | 4-Hydroxyestrone | Estrogen Receptor/ERR , Endogenous Metabolite | |
4-Hydroxyestrone, an endogenous estrogen metabolite, can strongly protect neuronal cells against oxidative damage. | |||
T1424 | Ethynyl estradiol | 17α-Ethynylestradiol,Ethinyl Estradiol | Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite |
Ethynyl estradiol is a semisynthetic alkylated ESTRADIOL with a 17-alpha-ethinyl substitution. It has high estrogenic potency when administered orally, and is often used as the estrogenic component in ORAL CONTRACEPTIVES... | |||
T12654 | (Rac)-Acolbifene | (Rac)-EM-652,EM-343 | Estrogen Receptor/ERR |
(Rac)-Acolbifene (EM-343) is the racemic form of Acolbifene. Acolbifene is a estrogen receptor antagonist. (Rac)-Acolbifene exhibits anti-estrogenic and estrogenic activities. (Rac)-Acolbifene contains a piperidine ring ... | |||
T33876L | Panomifene HCl | EGIS5650 HCl,GYKI 13504 HCl,Panomifene HCl(77599-17-8 Free base),EGIS 5650 HCl | HER |
Panomifene HCl is a selective anti-estrogenic compound with antitumor activity for the treatment of breast cancer. | |||
T0345 | Estropipate | Piperazine estrone sulfate,Pipestrone,Estrone sulfate piperazine salt | Estrogen Receptor/ERR , Estrogen/progestogen Receptor |
Estropipate (Piperazine estrone sulfate) is a natural estrogenic substance composed of estrone sulfate and piperazine. | |||
T13684 | Equilin | 7-Dehydroestrone | Calcium Channel |
Equilin (7-Dehydroestrone) is a neurotrophic estrogenic steroid with vasodilatory activity that increases monocyte-endothelial adhesion through NF-κB signalling.Equilin similarly relaxes mesenteric arterial resistance by... | |||
T7957 | 2-Isopropyl Thioxanthone | Others | |
2-Isopropyl Thioxanthone has potential anti-estrogenic and anti-androgenic properties. | |||
T23647 | Zindoxifene | D 16726 | Estrogen/progestogen Receptor |
Zindoxifene (D 16726) is an anti-estrogenic compound with antitumor activity that can be used in studies of breast and prostate cancer. | |||
T7465 | 4-Methylbenzylidene camphor | Enzacamene,4-MBC | AChE |
4-Methylbenzylidene camphor is an ultraviolet light blocker used in cosmetics and sunscreen preparations ,specifically UV B radiation, also has estrogenic activities. | |||
T6S0325 | Glycitein | Glycetein | Apoptosis , Others |
1. Gycitein has weak estrogenic activity. 2. Glycitein (Glycetein) inhibits glioma cell invasion through down-regulation of MMP-3 and MMP-9 gene expression. | |||
T8981 | WAY-169916 | WAY 169916,WAY169916 | NF-κB |
WAY-169916 is a pathway-selective inhibitor of estrogen receptor (ER). It acts by inhibiting NF-kB transcriptional activity but being devoid of conventional estrogenic activity. | |||
T3665 | Tectoridin | Shekanin | Estrogen Receptor/ERR , Reductase |
Tectoridin (Shekanin) possesses an estrogenic and thyroid hormone-like agent by activating estrogen and thyroid hormone receptors. Tectoridin has anti-oxidant, anti-inflammatory and hypoglycemic activities; Tectoridin an... | |||
T8984 | FLTX1 | Estrogen Receptor/ERR , Estrogen/progestogen Receptor | |
FLTX1 is a fluorescent derivative of Tamoxifen, designed to efficiently target and label intracellular Tamoxifen-binding sites (estrogen receptors) both under permeabilized and non-permeabilized conditions. Additionally,... | |||
TN1146 | 8-Prenylnaringenin | 8-Prenylnaringenin | Apoptosis , ROS |
8-Prenylnaringenin is a phytoestrogen with high estrogenic activity, | |||
T1514 | Norethindrone | Norethisterone | Estrogen/progestogen Receptor , Progesterone Receptor |
Norethindrone (Norethisterone) is a synthetic progestational hormone with actions similar to those of PROGESTERONE but functioning as a more potent inhibitor of ovulation. It has weak estrogenic and androgenic properties... | |||
T2569 | Chlorotrianisene | tris(p-methoxyphenyl)chloroethylene,CTA,tri-p-anisylchloroethylene,TACE | Estrogen Receptor/ERR , Estrogen/progestogen Receptor , COX |
Chlorotrianisene (tri-p-anisylchloroethylene) is an orally bioavailable, highly lipophilic, synthetic triphenylethylene (TPE) derivative and selective estrogen receptor modulator (SERM), with predominantly estrogenic but... | |||
T5S0993 | Kurarinone | BCL , Others , IκB/IKK , TNF , NF-κB , JAK , STAT | |
Kurarinone, a flavanoid derived from shrub Sophora flavescens,Kurarinone exhibits anti-tumor, estrogenic, and anti-inflammatory activities, it also shows strong inhibitory effect on immune responses. Kurarinone may ameli... | |||
T5625 | Zearalenone | Mycotoxin F2,RAL,F2 toxin,Toxin F2 | Others |
Zearalenone (F2 toxin) is a mycotoxin produced mainly by fungi belonging to the genus Fusarium in foods and feeds. Possess oestrogenic activity in cattle, pigs and sheep, with low acute toxicity. Causes precocious develo... |