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20

Compounds

Cat No. Product Name Synonyms Targets
T6406 Besifloxacin Hydrochloride BOL-303224-A,Besivance hydrochloride,Besifloxacin HCl Antibacterial , Antibiotic
Besifloxacin Hydrochloride (BOL-303224-A) is a fourth-generation fluoroquinolone antibiotic.
T68539 CEP-11981 BOL 303213X,ESK981 ; BOL 303213X,ESK981
CEP-11981 (ESK981; BOL 303213X) is an orally active tyrosine kinase inhibitor (TKI) that targets TIE2, VEGFR1-3, and FGFR1. It exhibits potential anti-tumor and anti-angiogenic effects.
T26910 Bromolysergide BOL
Bromolysergide is a serotonin antagonist.
T13451L Mapracorat BOL-303242X,ZK-245186 Others
Mapracorat is a novel non-steroidal selective agonist of glucocorticoid receptor.
T13451 (S)-Mapracorat (S)-ZK-245186,(S)-BOL-303242X Others
(S)-Mapracorat is a selective and less active agonist of glucocorticoid receptor.
T16338 Norgestimate metabolite Norelgestromin 17-Deacetyl norgestimate,17-Deacylnorgestimate Drug Metabolite
Norgestimate metabolite Norelgestromin (17-Deacylnorgestimate) is one of the active metabolites of norgestimate.It is a steroidal progestin used in contraceptive patches, where it is combined with the estrogen ethinyl es...
T16324 Nimbolide Apoptosis , NF-κB , CDK
Nimbolide suppresses CDK4/CDK6 kinase activity. Nimbolide inhibits the NF-κB, Wnt, PI3K-Akt, MAPK, and JAK-STAT signaling pathways. Nimbolide causes apoptosis through the inactivation of NF-κB. Nimbolide is a triterpene ...
T16045 Methotrexate metabolite DAMPA Antifolate , Drug Metabolite
Methotrexate metabolite (DAMPA) (DAMPA) is the active metabolite of Methotrexate. Methotrexate is a folic acid antagonist. Methotrexate is used as a chemotherapeutic agent and immunosuppressant.
T10814 Cinacalcet metabolite M4 Rarechem AL BW 1078 Calcium Channel
Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.
T12309 Omeprazole metabolite Omeprazole sulfone Omeprazole sulphone,Omeprazole sulfone Others
Omeprazole metabolite Omeprazole sulfone can inhibit proton pump.
T21059 Ticagrelor metabolite M5 Ticagrelor metabolite M5,,T437700,AR-C133913XX P2Y Receptor
Ticagrelor metabolite M5 (T437700) is a metabolite of Ticagrelor, the first reversible oral antagonist of P2Y12 receptor. Compared to Clopidogrel, Ticagrelor has faster and more consistent inhibition on ADP-receptors. Ti...
TN2549 1-Methoxycarbonyl-β-carboline 1-Methoxycarbonyl-beta-carboline Others
1-Methoxycarbonyl-β-carboline (1-Methoxycarbonyl-beta-carboline) is an alkaloid from Ailanthus altissima.
TN2019 Orobol 3'-Hydroxygenistein,3’,4’,5,7-tetrahydroxy-isoflavon BCL , Caspase , PI3K
Orobol (3’,4’,5,7-tetrahydroxy-isoflavon) is an inhibitor of tyrosine-specific protein kinase and phosphatidylinositol turnover. Orobol inhibits PI3K isoforms with IC50s of 3.46-5.27 μM for PI3K α/β/γ/K/δ. Orobol exhibit...
TN1445 Bisabolangelone p38 MAPK , MAPK
Bisabolangelone has anti-tumor, anti-inflammatory, anti-microbial, and antioxidant activities, it inhibits dendritic cell functions by blocking MAPK and NF-κB signaling.
T77149 Cobolimab TSR-022,GSK4069889 Others
Cobolimab (TSR-022) is a potent monoclonal antibody to TIM-3. Cobolimab induces internalization of TIM-3 with an IC50 value of 0.4464 nM. Cobolimab has antitumor activity and can be used to study advanced/metastatic mela...
T10738 Abemaciclib metabolite M20 CDK4/6-IN-4,LSN3106726 CDK
Abemaciclib metabolite M20 (CDK4/6-IN-4) is an active metabolite of Abemaciclib. Abemaciclib metabolite M20 is a selective CDK4/6 inhibitor and can be used for researches on the treatment of cancer.
T4037 Phorbol 4β-Phorbol,(+)-Phorbol PKC
Phorbol (4β-Phorbol), a plant-derived diterpene, is a tumor promoter through the activation of protein kinase C.
T5S1895 Norisoboldine Laurelliptine,(+)-Laurelliptine MAPK , Adenosine Receptor
1. Norisoboldine ((+)-Laurelliptine) might be a potential therapeutic agent for rheumatoid arthritis, and it functions through protecting joint destruction as well as regulating the abnormal immune responses. 2. Norisobo...
T21499 Dimebolin Latrepirdine,Dimebon,Dimebone 5-HT Receptor
Dimebolin (Latrepirdine) is a 5-HT6 antagonist.
TN7131 1-Formyl-β-carboline 9H-pyrido[3,4-b]indole-1-carbaldehyde Others
1-Formyl-β-carboline is an alkaloid derived from the leaves of Ailanthus altissima.

Compounds

Besifloxacin Hydrochloride
T6406
Synonym: BOL-303224-A,Besivance hydrochloride,Besifloxacin HCl
Target: Antibacterial, Antibiotic
CEP-11981
T68539
Synonym: BOL 303213X,ESK981 ; BOL 303213X,ESK981
Target:
Bromolysergide
T26910
Synonym: BOL
Target:
Mapracorat
T13451L
Synonym: BOL-303242X,ZK-245186
Target: Others
(S)-Mapracorat
T13451
Synonym: (S)-ZK-245186,(S)-BOL-303242X
Target: Others
Norgestimate metabolite Norelgestromin
T16338
Synonym: 17-Deacetyl norgestimate,17-Deacylnorgestimate
Target: Drug Metabolite
Nimbolide
T16324
Synonym:
Target: Apoptosis, NF-κB, CDK
Methotrexate metabolite
T16045
Synonym: DAMPA
Target: Antifolate, Drug Metabolite
Cinacalcet metabolite M4
T10814
Synonym: Rarechem AL BW 1078
Target: Calcium Channel
Omeprazole metabolite Omeprazole sulfone
T12309
Synonym: Omeprazole sulphone,Omeprazole sulfone
Target: Others
Ticagrelor metabolite M5
T21059
Synonym: Ticagrelor metabolite M5,,T437700,AR-C133913XX
Target: P2Y Receptor
1-Methoxycarbonyl-β-carboline
TN2549
Synonym: 1-Methoxycarbonyl-beta-carboline
Target: Others
Orobol
TN2019
Synonym: 3'-Hydroxygenistein,3’,4’,5,7-tetrahydroxy-isoflavon
Target: BCL, Caspase, PI3K
Bisabolangelone
TN1445
Synonym:
Target: p38 MAPK, MAPK
Cobolimab
T77149
Synonym: TSR-022,GSK4069889
Target: Others
Abemaciclib metabolite M20
T10738
Synonym: CDK4/6-IN-4,LSN3106726
Target: CDK
Phorbol
T4037
Synonym: 4β-Phorbol,(+)-Phorbol
Target: PKC
Norisoboldine
T5S1895
Synonym: Laurelliptine,(+)-Laurelliptine
Target: MAPK, Adenosine Receptor
Dimebolin
T21499
Synonym: Latrepirdine,Dimebon,Dimebone
Target: 5-HT Receptor
1-Formyl-β-carboline
TN7131
Synonym: 9H-pyrido[3,4-b]indole-1-carbaldehyde
Target: Others
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TargetMol