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20

Compounds

Cat No. Product Name Synonyms Targets
T3901 Solasonine Others
Solasonine exerts leishmanicidal activity against promastigote forms of L. amazonensis.
T4035 Khasianine Others
Khasianine has strong activity against liver damage induced by CCl4.
T3S1251 Neoruscogenin ROR
1. Neoruscogenin represents a universal pharmacological tool for RORα research due to its specific selectivity profile versus other nuclear receptors.
T3S0509 Gaultherin COX
Gaultherin has analgesic, and anti-inflammatory activities.Gaultherin lacks gastric ulcerogenic effect, because of it released salicylate in intestine slowly, not in stomach and it left the cyclooxygenase-1 unaffected, w...
T2550 Tolmetin Tolectin COX
Tolmetin (Tolectin) is a Nonsteroidal Anti-inflammatory Drug. The mechanism of action of tolmetin is as a Cyclooxygenase Inhibitor. The chemical classification of tolmetin is Nonsteroidal Anti-inflammatory Compounds.
T3S1265 Liriopesides B Nolinospiroside F Others
Liriopesides B (Nolinospiroside F) exhibited potential anticancer activity against human ovarian cancer A2780 cells.
T7024 Qingyangshengenin Qingyangshengenin A,Cynanchagenin Others
Qingyangshengenin (Cynanchagenin) is a steroid used in the preparation of antiepileptic agents.
T11399 Giredestrant GDC-9545 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Giredestrant (GDC-9545) potently competes with estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has anti-tumor activity. Giredestrant, a non-steroidal ER ligand,...
T0301 Ethisterone 17α-Ethynyltestosterone,Pregneninolone Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.
T0380 Bicalutamide ICI-176334 Androgen Receptor , Autophagy
Bicalutamide (ICI-176334), a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting the receptor binding of androgens.
T6737 Zaltoprofen CN100,Soleton COX
Zaltoprofen (Soleton) is a Cox-1 and Cox-2 inhibitor, which is used for the treatment of arthritis.
T1587 Exemestane EXE,FCE 24304,PNU155971 Aromatase
Exemestane (EXE) is an Aromatase Inhibitor. The mechanism of action of exemestane is as an Aromatase Inhibitor.
T26539 AC-262536 AC262536 Androgen Receptor
AC-262536 is a selective androgen receptor (SAR) modulator. It has partial agonist activity with respect to testosterone and suppresses luteinizing hormone.
T22371 Mivacurium dichloride Mivacurium chloride AChR
Mivacurium dichloride (Mivacurium chloride) is a non-depolarising, rapid neuromuscular blocker of short duration, used therefore as anesthetic, to provide skeletal muscle relaxation in minor surgical operations, in emerg...
T0383 Fenspiride hydrochloride Fenspiride HCl,Pneumorel,Fluiden,Decaspiride Adrenergic Receptor , PDE , Histamine Receptor
Fenspiride hydrochloride (Decaspiride) , an oxazolidinone spiro compound, is a drug used in the therapy of certain respiratory diseases. It is approved for use in Russia for the therapy of chronic and acute inflammatory ...
T4036 Solasodine Solancarpidine,Purapuridine,Solasodin Apoptosis , Others , E1/E2/E3 Enzyme , Antifungal
Solasodine (Purapuridine)(Purapuridine) is a poisonous alkaloid chemical compound that occurs in plants of the Solanaceae family. Solasodine showed selective cytotoxicity against cervical cancer cell line (HeLa) and huma...
T4602 Hydrocortisone hemisuccinate Hydrocortisone 21-he,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate Glucocorticoid Receptor , Others , Interleukin
Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.
T61444 Nonsteroidal aromatase inhibitor 1
Nonsteroidal aromatase inhibitor 1 (Compound 13h) effectively inhibits the enzyme CYP19A1 with an IC50 value of 0.09 nM. Due to its potent inhibitory activity, Nonsteroidal aromatase inhibitor 1 holds promise for researc...
T2S0250 Pseudoprotogracillin Others
Pseudoprotogracillin is a steroidal saponin extracted from Dioscoreae.
T8094 16-​Dehydroprogesterone 16-Dehydroprogesterone Endogenous Metabolite
16-Dehydroprogesterone is a endogenous Metabolite. 16-Dehydroprogesterone is a steroidal progestin.

Compounds

Solasonine
T3901
Synonym:
Target: Others
Khasianine
T4035
Synonym:
Target: Others
Neoruscogenin
T3S1251
Synonym:
Target: ROR
Gaultherin
T3S0509
Synonym:
Target: COX
Tolmetin
T2550
Synonym: Tolectin
Target: COX
Liriopesides B
T3S1265
Synonym: Nolinospiroside F
Target: Others
Qingyangshengenin
T7024
Synonym: Qingyangshengenin A,Cynanchagenin
Target: Others
Giredestrant
T11399
Synonym: GDC-9545
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Ethisterone
T0301
Synonym: 17α-Ethynyltestosterone,Pregneninolone
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Bicalutamide
T0380
Synonym: ICI-176334
Target: Androgen Receptor, Autophagy
Zaltoprofen
T6737
Synonym: CN100,Soleton
Target: COX
Exemestane
T1587
Synonym: EXE,FCE 24304,PNU155971
Target: Aromatase
AC-262536
T26539
Synonym: AC262536
Target: Androgen Receptor
Mivacurium dichloride
T22371
Synonym: Mivacurium chloride
Target: AChR
Fenspiride hydrochloride
T0383
Synonym: Fenspiride HCl,Pneumorel,Fluiden,Decaspiride
Target: Adrenergic Receptor, PDE, Histamine Receptor
Solasodine
T4036
Synonym: Solancarpidine,Purapuridine,Solasodin
Target: Apoptosis, Others, E1/E2/E3 Enzyme, Antifungal
Hydrocortisone hemisuccinate
T4602
Synonym: Hydrocortisone 21-he,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate
Target: Glucocorticoid Receptor, Others, Interleukin
Nonsteroidal aromatase inhibitor 1
T61444
Synonym:
Target:
Pseudoprotogracillin
T2S0250
Synonym:
Target: Others
16-​Dehydroprogesterone
T8094
Synonym: 16-Dehydroprogesterone
Target: Endogenous Metabolite
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TargetMol