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20

Compounds

Cat No. Product Name Synonyms Targets
T68260 Calmidazolium (cation)
Calmidazolium (cation) is a powerful inhibitor of or red blood cell Ca -ATPase & Ca transport into inside-out red blood cell vesicles; an antagonist of calmodulin.
T32984 LX-201 cation
LX-201 cation is a bioactive chemical.
T34817 Tetrabutylphosphonium cation Tetra-n-butylphosphonium,J279H,Tetrabutylphosphonium ion,Tetrabutylphosphonium,Phosphonium, tetrabutyl-
Tetrabutylphosphonium cation is a light orange solid and is the salt of the liphilic tetrabutylammonium cation and linear tribromide anion.
T25628 Lapyrium Lapyrium cation
Lapyrium is a cationic surfactant that is used in personal care products as a biocide and antistatic. It is also used by the chloride salt, lapyrium chloride, in waste-water treatment and corrosion inhibition formulation...
T32592 Lauralkonium Lauralkonium ion,Lauralkonium cation
Lauralkonium is a bioactive chemical.
T25636 Laudexium Laudexium ion,Laudexium cation
Laudexium is a neuromuscular blocking drug or skeletal muscle relaxant in the category of non-depolarizing neuromuscular-blocking drugs. It is used adjunctively in surgical anesthesia to facilitate endotracheal intubatio...
T25640 Laurolinium Laurolinium ion,Laurolinium cation
Laurolinium is an antimicrobial.
T26666 ASM-024 AChR
ASM-024, a potent nicotinic receptor agonist, is a small molecule synthetic piperazine compound that promotes different targets and signaling pathways of β2-adrenergic receptors mediating smooth muscle relaxation, and is...
T21623 AS1269574 AS 1269574 GPR , TRP/TRPV Channel
AS1269574 is a potent, orally available GPR119 agonist. AS1269574(AS 1269574) has the potential for the research of type 2 diabetes.
T68783 Stercuronium
Stercuronium is an aminosteroid neuromuscular blocking agent which was never marketed. It acts as a competitive antagonist of the nicotinic acetylcholine receptor, and is also reported to be an acetylcholinesterase inhib...
T70310 INCB-39110
INCB-39110 is a JAK1 inhibitor.
T68735 Ciclotropium (free base)
Ciclotropium (free base) is quaternary ammonium compound with anticholinergic and parasympatholytic activity. Oral Cyclotropium bromide inhibited fasting and meal-stimulated colonic motility significantly without causing...
T68502 Dibrospidium Free Base
Dibrospidium Free Base is a dispirotripiperazine derivative and alkylating agent with potential antineoplastic and anti-inflammatory activities. The duration of DNA synthesis inhibition in tumor cells was found to correl...
T9776 TRPM4 inhibitor 8 TRP/TRPV Channel
TRPM4 inhibitor 8 is an inhibitor of Transient receptor potential melastatin 4(TRPM4) which contributes to viability, migration, cell cycle shift, and adhesion.
T9245 TRPM4-IN-1 CBA,4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid TRP/TRPV Channel
TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
T10662L Calcimycin Antibiotic A-23187,A-23187 Apoptosis , Antibacterial , Antibiotic , Autophagy , Antifungal
Calcimycin (A-23187) is an ionophorous, polyether carboxylic antibiotic from Streptomyces chartreusensis. It binds and transports calcium and other divalent cations across membranes and uncouples oxidative phosphorylatio...
T1050 Prazosin hydrochloride Prazosin hydrochloride,Prazosin HCl,cp-12299-1,Peripress,Vasoflex,Minipress Potassium Channel , MRP , Adrenergic Receptor , ABC , Autophagy
Prazosin hydrochloride (Vasoflex) reduces peripheral resistance and relaxes vascular smooth muscles as a selective adrenergic alpha-1 antagonist by a mechanism not completely known. Prazosin hydrochloride is a synthetic ...
TQ0157 EIPA L593754,MH 12-43 Sodium Channel , TRP/TRPV Channel
EIPA (L593754) (L593754, MH 12-43) is a TRPP3 channel inhibitor (IC50: 10.5 μM). It also inhibits Na+/H+-exchanger (NHE) and macropinocytosis.
T1045 Trimipramine maleate Surmontil maleate Dopamine Receptor , 5-HT Receptor , Antibacterial , Adrenergic Receptor , Norepinephrine , Histamine Receptor
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Mal...
T81449 PKC-ε translocation inhibitor peptide PKC
PKC-ε Translocation Inhibitor Peptide is a selective modulator that controls the FcγR-mediated internalization rate of opsonized beads without affecting FcαR trafficking [1].

Compounds

Calmidazolium (cation)
T68260
Synonym:
Target:
LX-201 cation
T32984
Synonym:
Target:
Tetrabutylphosphonium cation
T34817
Synonym: Tetra-n-butylphosphonium,J279H,Tetrabutylphosphonium ion,Tetrabutylphosphonium,Phosphonium, tetrabutyl-
Target:
Lapyrium
T25628
Synonym: Lapyrium cation
Target:
Lauralkonium
T32592
Synonym: Lauralkonium ion,Lauralkonium cation
Target:
Laudexium
T25636
Synonym: Laudexium ion,Laudexium cation
Target:
Laurolinium
T25640
Synonym: Laurolinium ion,Laurolinium cation
Target:
ASM-024
T26666
Synonym:
Target: AChR
AS1269574
T21623
Synonym: AS 1269574
Target: GPR, TRP/TRPV Channel
Stercuronium
T68783
Synonym:
Target:
INCB-39110
T70310
Synonym:
Target:
Ciclotropium (free base)
T68735
Synonym:
Target:
Dibrospidium Free Base
T68502
Synonym:
Target:
TRPM4 inhibitor 8
T9776
Synonym:
Target: TRP/TRPV Channel
TRPM4-IN-1
T9245
Synonym: CBA,4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid
Target: TRP/TRPV Channel
Calcimycin
T10662L
Synonym: Antibiotic A-23187,A-23187
Target: Apoptosis, Antibacterial, Antibiotic, Autophagy, Antifungal
Prazosin hydrochloride
T1050
Synonym: Prazosin hydrochloride,Prazosin HCl,cp-12299-1,Peripress,Vasoflex,Minipress
Target: Potassium Channel, MRP, Adrenergic Receptor, ABC, Autophagy
EIPA
TQ0157
Synonym: L593754,MH 12-43
Target: Sodium Channel, TRP/TRPV Channel
Trimipramine maleate
T1045
Synonym: Surmontil maleate
Target: Dopamine Receptor, 5-HT Receptor, Antibacterial, Adrenergic Receptor, Norepinephrine, Histamine Receptor
PKC-ε translocation inhibitor peptide
T81449
Synonym:
Target: PKC
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TargetMol