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Trimipramine maleate

🥰Excellent
Catalog No. T1045Cas No. 521-78-8
Alias Surmontil maleate

Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Maleate is the maleate salt form of trimipramine, a tricyclic secondary amine of the dibenzazepine class, with an antidepressant property.

Trimipramine maleate
Other Forms of Trimipramine maleate:
TrimipramineT21364739-71-9
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Trimipramine maleate

🥰Excellent
Purity: 99.47%
Catalog No. T1045Alias Surmontil maleateCas No. 521-78-8
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Maleate is the maleate salt form of trimipramine, a tricyclic secondary amine of the dibenzazepine class, with an antidepressant property.
Pack SizePriceAvailabilityQuantity
50 mg$33In Stock
100 mg$47In Stock
200 mg$68In Stock
500 mg$112In Stock
1 mL x 10 mM (in DMSO)$50In Stock
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Purity:99.47%
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COA LCMS HNMR HPLC
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Product Introduction

Bioactivity
Description
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Maleate is the maleate salt form of trimipramine, a tricyclic secondary amine of the dibenzazepine class, with an antidepressant property.
Targets&IC50
5-HT 2 Receptor:8.10 (pKi), 5-HT 1C Receptor:6.39 (pKi), sPLA2:4.66 (pKi)
AliasSurmontil maleate
Chemical Properties
Molecular Weight410.51
FormulaC24H30N2O4
Cas No.521-78-8
SmilesOC(=O)\C=C/C(O)=O.CC(CN(C)C)CN1c2ccccc2CCc2ccccc12
Relative Density.1.029g/cm3
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 50 mg/mL (121.8 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.4360 mL12.1800 mL24.3599 mL121.7997 mL
5 mM0.4872 mL2.4360 mL4.8720 mL24.3599 mL
10 mM0.2436 mL1.2180 mL2.4360 mL12.1800 mL
20 mM0.1218 mL0.6090 mL1.2180 mL6.0900 mL
50 mM0.0487 mL0.2436 mL0.4872 mL2.4360 mL
100 mM0.0244 mL0.1218 mL0.2436 mL1.2180 mL

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Keywords

Trimipramine MaleateTrimipramine maleateTrimipramineSurmontil MaleateSert (Sodium-dependent)Serotonin ReceptorserotoninNoradrenaline transporter (Sodium-dependent)noradrenalineneurological diseaseInhibitorinhibithuman organic cation transportershSERThOCT3hOCT2hOCT1hNATHistamineReceptorHistamine ReceptorhDATH1 receptorDopamineReceptorDopamine ReceptordopamineDopamineDA transporterDA D2 receptorBacterialanxiolyticantidepressantsAdrenergicReceptorAdrenergic Receptor5-hydroxytryptamine Receptor5-hydroxytryptamine5HTReceptor5-HTlc receptors5-HTIA receptors5-HT25-HT1C5-HT1A5-HT Receptor5HT Receptor5-HT
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