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Trimipramine maleate

Catalog No. T1045 CAS 521-78-8

Synonyms: Surmontil maleate

Trimipramine maleate appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Maleate is the maleate salt form of trimipramine, a tricyclic secondary amine of the dibenzazepine class, with an antidepressant property.

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Trimipramine maleate, CAS 521-78-8

Pack Size	Availability	Price/USD
25 mg	In stock	31.00
50 mg	In stock	41.00
100 mg	In stock	50.00
200 mg	In stock	75.00
1 mL * 10 mM (in DMSO)	In stock	50.00

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Purity 98.02%

HNMR HPLC COA

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Storage & Solubility Information

Description	Trimipramine maleate appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Maleate is the maleate salt form of trimipramine, a tricyclic secondary amine of the dibenzazepine class, with an antidepressant property.
Targets&IC50	5-HT , Adrenergic Receptor , DA transporter , Dopamine , H1 receptor , Noradrenaline transporter (Sodium-dependent) , Sert (Sodium-dependent)

Synonyms	Surmontil maleate
Purity	98.02%
Molecular Weight	410.51
Formula	C24H30N2O4
CAS No.	521-78-8

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 6 months

Solubility Information

DMSO: 10 mM

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Diamond M, et al. Eur Neuropsychopharmacol. 2006 Oct;16(7):481-90.

Related compound libraries

This product is contained In the following compound libraries：

Approved Drug Library Bioactive Compound Library Inhibitor Library Anti-Cancer Compound Library Clinical Compound Library Adrenergic Receptor-Targeted Compound Library Anti-Infection Compound Library Neuronal Signaling Compound Library Histamine & Melatonin Receptor-Targeted Compound Library Serotonin Receptor-Targeted Compound Library FDA-Approved Drug Library Immunology/Inflammation Compound Library GPCR Compound Library Cardiotoxicity Compound Library Anti-Cardiovascular Disease Compound Library CNS-Penetrant Compound Library Drug Repurposing Compound Library Neurotransmitter Receptor Compound Library Anti-Neurodegenerative Disease Compound Library Drug-induced Liver Injury (DILI) Compound Library Nonsteroidal Anti-Inflammatory Compound Library FDA-Approved & Pharmacopeia Drug Library Anti-Parkinson's Disease Compound Library Anti-Alzheimer's Disease Compound Library

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Related compounds with same targets

Tandospirone GSK163090 Dexpramipexole Sumanirole maleate CP-809101 lumateperone Tosylate GSK189254A Bavisant

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