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20

Compounds

Cat No. Product Name Synonyms Targets
T11230 ERRα antagonist-1 ERR+/- antagonist-1,ERRa antagonist-1 Estrogen/progestogen Receptor
ERRα antagonist-1 (ERR+/- antagonist-1) is a high-affinity, selective antagonist of the estrogen-related receptor α (ERRα). It effectively prevents the interaction of ERRα with both Proliferator-activated Receptor γ Coac...
T39078 CXCR7 antagonist-1 CXCR7 antagonist-1 CXCR
CXCR7 antagonist-1 is a specific antagonist of the binding of the SDF-1 chemokine or I-TAC to the chemokine receptor CXCR7. CXCR7 antagonist-1 prevents tumor cell proliferation and tumor formation and can be used in stud...
T15785 LPA1 receptor antagonist 1 LPA1 R antagonist 1 LPA Receptor
LPA1 receptor antagonist 1(LPA1 R antagonist 1) is a selective and potent lysophosphatidic acid (LPA1) receptor antagonist (IC50 : 25 nM) for the study of idiopathic pulmonary fibrosis.
T10031 EP1-antagonist-1 EP1-antanoist-1,EP1 antagonist 1 Prostaglandin Receptor
EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).
T37792 A2A receptor antagonist 1 CPI-444 analog,A2A receptor antagonist 1 Adenosine Receptor
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
T13216 TSHR antagonist S37 TSH Receptor
TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).
T5698 TRPM8 antagonist 2 TRP/TRPV Channel
TRPM8 antagonist 2 is a potent and selective TRPM8 antagonist with an IC50 of 0.2 nM. TRPM8 antagonist 2 is used in the research of neuropathic pain syndromes.
T9709 TRPM8 antagonist 3 TRP/TRPV Channel
TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
T14881 CB1 antagonist 2 AM4113 Cannabinoid Receptor
CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with an IC50 of 25.5 nM.
T10058 A2B receptor antagonist 1 Adenosine Receptor
A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.
T10712 CCR2 antagonist 3 AZD-2927,AZD2927 CCR
CCR2 antagonist 3 (AZD-2927) is an antagonist of CCR2.
TP1935L1 RAGE antagonist peptide acetate Beta Amyloid
RAGE antagonist peptide acetate is an advanced antagonist of glycation end products (RAGE). RAGE antagonist peptide acetate possesses anti-tumor and anti-inflammatory activities. RAGE antagonist peptide acetate prevents ...
T12320 ORL1 antagonist 1 Opioid Receptor
ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).
T10156 CCR3 antagonist 1 CCR
CCR3 antagonist 1 is a potent CCR3 antagonist, used for the research of inflammatory and immunologic diseases.
T9983 CCR8 antagonist 1 LUN04765 CCR
CCR8 antagonist 1 is an antagonist of C-C Motif Chemokine Receptor 8 (CCR8) with a Ki value of 1.6 nM.
T5829 H4 Receptor antagonist 1 Histamine Receptor
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
T10056 Neurokinin antagonist 1 Neuropeptide Y Receptor
Neurokinin antagonist 1 is a potent is a neuropeptide antagonist that can be used to study neurological disorders.
T13453 CGRP antagonist 1 CGRP Receptor
CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the study of cardiovascular and neurovascular diseases.
T8848 GPR34 receptor antagonist 2 Tyrosine, N-[(2E)-3-(4'-chloro[1,1'-biphenyl]-4-yl)-1-oxo-2-propen-1-yl]-O-(phenylmethyl)-,gpr34-receptor-antagonist-2 Others
GPR34 receptor antagonist 2 (Tyrosine, N-[(2E)-3-(4'-chloro[1,1'-biphenyl]-4-yl)-1-oxo-2-propen-1-yl]-O-(phenylmethyl)-) is an anti-inflammatory agent.
T10169 5-HT4 antagonist 1 5-HT Receptor
5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).

Compounds

ERRα antagonist-1
T11230
Synonym: ERR+/- antagonist-1,ERRa antagonist-1
Target: Estrogen/progestogen Receptor
CXCR7 antagonist-1
T39078
Synonym: CXCR7 antagonist-1
Target: CXCR
LPA1 receptor antagonist 1
T15785
Synonym: LPA1 R antagonist 1
Target: LPA Receptor
EP1-antagonist-1
T10031
Synonym: EP1-antanoist-1,EP1 antagonist 1
Target: Prostaglandin Receptor
A2A receptor antagonist 1
T37792
Synonym: CPI-444 analog,A2A receptor antagonist 1
Target: Adenosine Receptor
TSHR antagonist S37
T13216
Synonym:
Target: TSH Receptor
TRPM8 antagonist 2
T5698
Synonym:
Target: TRP/TRPV Channel
TRPM8 antagonist 3
T9709
Synonym:
Target: TRP/TRPV Channel
CB1 antagonist 2
T14881
Synonym: AM4113
Target: Cannabinoid Receptor
A2B receptor antagonist 1
T10058
Synonym:
Target: Adenosine Receptor
CCR2 antagonist 3
T10712
Synonym: AZD-2927,AZD2927
Target: CCR
RAGE antagonist peptide acetate
TP1935L1
Synonym:
Target: Beta Amyloid
ORL1 antagonist 1
T12320
Synonym:
Target: Opioid Receptor
CCR3 antagonist 1
T10156
Synonym:
Target: CCR
CCR8 antagonist 1
T9983
Synonym: LUN04765
Target: CCR
H4 Receptor antagonist 1
T5829
Synonym:
Target: Histamine Receptor
Neurokinin antagonist 1
T10056
Synonym:
Target: Neuropeptide Y Receptor
CGRP antagonist 1
T13453
Synonym:
Target: CGRP Receptor
GPR34 receptor antagonist 2
T8848
Synonym: Tyrosine, N-[(2E)-3-(4'-chloro[1,1'-biphenyl]-4-yl)-1-oxo-2-propen-1-yl]-O-(phenylmethyl)-,gpr34-receptor-antagonist-2
Target: Others
5-HT4 antagonist 1
T10169
Synonym:
Target: 5-HT Receptor
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TargetMol