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EP1-antagonist-1

Name: EP1-antagonist-1
Brand: TargetMol
SKU: T10031
Price: 195 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T10031Cas No. 851204-35-8

Alias EP1-antanoist-1, EP1 antagonist 1

EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).

EP1-antagonist-1

🥰Excellent

Purity: 97.06%

Catalog No. T10031Alias EP1-antanoist-1, EP1 antagonist 1Cas No. 851204-35-8

EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).

Pack Size	Price	Availability
1 mg	$195	In Stock
5 mg	$396	In Stock
10 mg	$579	In Stock
25 mg	$912	In Stock
50 mg	$1,220	In Stock
100 mg	$1,650	In Stock
1 mL x 10 mM (in DMSO)	$449	In Stock

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Bulk & Custom

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:97.06%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).
Targets&IC50	EP1:8.5(pIC50), EP1:7.54(pKi)
Synonyms	EP1-antanoist-1, EP1 antagonist 1

Chemical Properties

Molecular Weight	470.14
Formula	C₁₉H₁₅BrCl₂N₂O₃
Cas No.	851204-35-8
Smiles	C(C1=C(OCC2=C(Cl)C=C(Cl)C=C2)C=CC(Br)=C1)N3N=C(C(O)=O)C=C3C
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 55 mg/mL (116.99 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.1270 mL	10.6351 mL	21.2703 mL	106.3513 mL
5 mM	0.4254 mL	2.1270 mL	4.2541 mL	21.2703 mL
10 mM	0.2127 mL	1.0635 mL	2.1270 mL	10.6351 mL
20 mM	0.1064 mL	0.5318 mL	1.0635 mL	5.3176 mL
50 mM	0.0425 mL	0.2127 mL	0.4254 mL	2.1270 mL
100 mM	0.0213 mL	0.1064 mL	0.2127 mL	1.0635 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc