acting — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T0202	Sulbentine	Dibenzthione	Antifungal
	Sulbentine (Dibenzthione) is an antifungal agent.		Antifungal
T5051	Isopropamide Iodide		AChR
	Isopropamide iodide is a long-acting anticholinergic drug. It is used in the treatment of peptic ulcers and other gastrointestinal disorders. It also acts as a muscarinic receptor antagonist which can be applied to the t...		AChR
T4985	Neticonazole Hydrochloride		Antifungal
	Neticonazole Hydrochloride is an imidazole antifungal for the treatment of fungal skin infections. Neticonazole is reported as a potent exosome inhibitor which can block the activity of exosomes.		Antifungal
T1674	Nateglinide	A4166,Senaglinide	Potassium Channel , Proteasome , PPAR
	Nateglinide (Senaglinide) is an oral hypoglycemic agent and amino acid derivative that stimulates insulin secretion from the pancreas and is used in the therapy of type 2 diabetes. Nateglinide has been linked to rare ins...		Potassium Channel , Proteasome , PPAR
T19862	Voxilaprevir		HCV Protease
	Voxilaprevir is an inhibitor of hepatitis C virus (HCV) nonstructural (NS) protein 3/4A protease.		HCV Protease
T0388	Cilnidipine	FRC-8653	Calcium Channel
	Cilnidipine (FRC-8653)(FRC8653) is a dual L- and N-type calcium channel blocker and displays antihypertensive, sympatholytic and neuroprotective activity.		Calcium Channel
T2390	Cevimeline hydrochloride hemihydrate		AChR
	Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug for xerostomia in Sjogren's syndrome.		AChR
T7943	Fluphenazine decanoate		Dopamine Receptor
	Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.		Dopamine Receptor
T3716	Rolapitant	SCH619734	Neurokinin receptor
	Rolapitant (SCH619734) Hydrochloride is the hydrochloride salt form of rolapitant, an orally bioavailable, centrally-acting, selective, neurokinin 1 receptor (NK1-receptor) antagonist with potential antiemetic activity. ...		Neurokinin receptor
T6504	Flupirtine maleate	Katadolon maleate	Potassium Channel , NMDAR , iGluR
	Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. It is an NMDA receptor antagonist , and also a specific neuronal potassium channel opener.		Potassium Channel , NMDAR , iGluR
T5159	Olodaterol hydrochloride	BI-1744 HCl,BI 1744 hydrochloride	Adrenergic Receptor
	Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and activating β2-adrenergic receptors...		Adrenergic Receptor
T20720	Norethisterone enanthate	NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,NSC-9564	Estrogen/progestogen Receptor
	Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects.		Estrogen/progestogen Receptor
T0373	Erlotinib	OSI-744,NSC 718781,CP358774,R1415	EGFR , Autophagy
	Erlotinib (NSC-718781) is an EGFR inhibitor (IC50: 2 nM). It is used for the treatment of non-small cell lung cancer.		EGFR , Autophagy
T0364L	Dibucaine hydrochloride	Cinchocaine HCl,Dibucaine HCl,Cinchocaine hydrochloride	Sodium Channel , AChR
	Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.		Sodium Channel , AChR
T31716	Etidocaine Hydrochloride	W-19053,Duranest,W19053,W 19053	Sodium Channel
	Etidocaine Hydrochloride (W19053) is a long-acting anesthetic and a blocker of the voltage-gated sodium channel.		Sodium Channel
T0749	Succinylsulfathiazole	Succinylsulphathiazole	Antibacterial , Antibiotic , Autophagy
	Succinylsulfathiazole (Succinylsulphathiazole) is a sulfonamide. An ultra long-acting drug.		Antibacterial , Antibiotic , Autophagy
T68087	Inaperisone		Others
	Inaperisone is a novel centrally acting muscle relaxant that inhibits the voiding reflex. Inaperisone may inhibit the voiding reflex by acting indirectly on GABAB receptors in the brainstem.		Others
T33386	Milveterol HCl	Milveterol,GSK-159797,GSK 159797,GSK159797	Adrenergic Receptor
	Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).		Adrenergic Receptor
T28360	PF-00489791	PF-4634817,PF 4634817,PF00489791,PF 00489791,PF4634817	PDE
	PF-00489791 (PF4634817) is a long-acting PDE5 inhibitor with hypotensive activity for the study of diabetic nephropathy.		PDE
T4548	Procaterol hydrochloride		Adrenergic Receptor
	Short-acting β2-adrenergic receptor agonist used to treat asthma.		Adrenergic Receptor