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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7107 | δ-Sleep Inducing Peptide | DSIP,Delta-Sleep Inducing Peptide | Antioxidant |
δ-Sleep Inducing Peptide (DSIP) is a neuropeptide, with antioxidant and anxiolytic properties. | |||
T78005 | δ-Sleep Inducing Peptide acetate | Delta-Sleep Inducing Peptide acetate | |
δ-Sleep Inducing Peptide acetate, a neuropeptide, exhibits antioxidant and anxiolytic properties [1] [2]. | |||
T82587 | Delta (Phospho) Sleep Inducing Peptide | DSIP-P | |
Delta (Phospho) Sleep Inducing Peptide (DSIP-P), a peptide that promotes sustained sleep, elicits alterations in circadian locomotor activity in rats [1] [2] [3]. | |||
T36949 | Niaprazine | 5-HT Receptor , Adrenergic Receptor , Histamine Receptor | |
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for sleep disorder research[1][2]. Niaprazine exhibits a low aff... | |||
T7694 | 6-fluoro-DL-Tryptophan | 5-HT Receptor | |
6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis. | |||
T7413 | JNJ-5207852 | Histamine Receptor | |
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor. | |||
T4S1999 | Valepotriate | Valtrate | Apoptosis , HIV Protease |
Valepotriate (Valtrate) fraction can have sedative effects and affect behavioral parameters related to recognition memory. Valepotriates, a new class of cytotoxic and antitumor agents, they are very potent cytotoxic agen... | |||
T16421 | P-MPPI hydrochloride | 5-HT Receptor | |
p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects. | |||
T8944 | TTA-A2 | Calcium Channel | |
TTA-A2 is a selective T-type calcium channel antagonist as a potent anticonvulsant that the Cav3.1 isoform plays a prominent role in mediating. TTA-A2 is equally potent against the Cav3.1 (a1G) and Cav3.2 (a1H) channels ... | |||
T8822 | JNJ-5207852 dihydrochloride | Histamine Receptor | |
JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor. | |||
T12877L | Seltorexant | JNJ-42847922 | OX Receptor |
Seltorexant (JNJ-42847922) crosses the blood-brain barrier and quickly occupies OX2R binding sites in the rat brain. Seltorexant is a high-affinity and selective orexin-2 receptor antagonist (pKi: 8.0 and 8.1 for human a... | |||
T3722 | MK-1064 | Urokinase inhibitor 1,MK 1064 | OX Receptor |
MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA). | |||
TN3910 | Ecdysone | Apoptosis , ATPase , Glucocorticoid Receptor , Potassium Channel , Sodium Channel , Endogenous Metabolite , Autophagy | |
Ecdysone is a major steroid hormone in insects and herbs. Ecdysone triggers mineralocorticoid receptor activation and induces cellular apoptosis. Ecdysone signaling through Ecdysone receptor isoform B1 is required cell a... | |||
T2S0842 | Scutellarin methyl ester | Scutellarin methylester | Others |
Scutellarin methyl ester has the effect of improving sleep, such as prolonging sleep time, increasing the incidence of sleep, shortening sleep latency, which also helps to delay aging process. | |||
T63736 | Bafrekalant | Others | |
Bafrekalant is a diazabicyclo-substituted imidazo[1,2-a]pyrimidine derivative that can be used to study sleep-related breathing disorders such as obstructive and central sleep apnoea and snoring. | |||
T14974 | Citenamide | Cytenamide,AY-15613 | Others |
Citenamide (AY-15613) has anticancer and anticonvulsant activity and is used in the study of neurological disorders because of its sleep-promoting properties. | |||
T24421 | LY-2624803 | DB-7,LY2624803,HY-10275,LY 2624803 | 5-HT Receptor , Histamine Receptor |
LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep. | |||
T33824 | Orotirelin | CG 3509,Orotireline | Others |
Orotirelin(CG 3509), a thyrotropin-releasing hormone analog, reversed pentobarbital-induced sleep time.Orotirelin may be beneficial in animals with focal cerebral ischemia. | |||
T5756 | Hastatoside | Others | |
Hastatoside and verbenalin are major sleep-promoting components of V. officinalis. Hastatoside has anti-inflammatory activity. | |||
T26559 | ACT-462206 | OX Receptor | |
ACT-462206 is an orally available Orexin 1/Orexin 2 receptor antagonist that crosses the blood-brain barrier.ACT-462206 is highly potent and can be used in studies of sleep and anxiety. |