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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12910 | Sigma-1 receptor antagonist 1 | Sigma receptor | |
Sigma-1 receptor antagonist 1 is an effective and selective antagonist of sigma-1 receptor. Sigma-1 receptor antagonist 1 exhibits antineuropathic pain activity and can be used in the treatment of neuropathic pain studie... | |||
T4031 | S1p receptor agonist 1 | S1p-receptor-agonist-1 | S1P Receptor , LPL Receptor |
S1p receptor agonist 1 (S1p-receptor-agonist-1) is an S1P receptor agonist. | |||
T10058 | A2B receptor antagonist 1 | Adenosine Receptor | |
A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist. | |||
T5829 | H4 Receptor antagonist 1 | Histamine Receptor | |
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. | |||
T13736 | Interferon receptor inducer-1 | IFNAR | |
Interferon receptor inducer-1 Used in the treatment of a disorder in which the induction of interferon is involved. is an interferon (IFN) receptor inducer. | |||
T11211 | EP4 receptor antagonist 1 | Prostaglandin Receptor | |
EP4 Receptor Antagonist 1 is a highly potent and selective competitive prostanoid EP4 receptor antagonist, effective for cancer immunotherapy. It inhibits both human and mouse EP4 receptors with IC50 values of 6.1 nM and... | |||
T9244 | σ1 Receptor antagonist-1 | Sigma receptor | |
σ1 Receptor antagonist-1 is a selective sigma 1 receptor antagonist. | |||
T11349 | GABAA receptor agent 1 | GABA Receptor | |
GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor. | |||
T12911 | Sigma-1 receptor antagonist 2 | Sigma receptor | |
Sigma-1 receptor antagonist 2 is a potent and selective antagonist of sigma 1 receptor (σ1 R) (σ1 and σ2 receptor with Kis of 3.88 and 1288 nM , respectively). | |||
T12912 | Sigma-1 receptor antagonist 3 | Sigma receptor , HER | |
Sigma-1 receptor antagonist 3 is a potent and selective antagonist of Sigma-1 (σ1) receptor(Ki : 1.14 nM), has the potential for the neuropathic pain. | |||
T37792 | A2A receptor antagonist 1 | CPI-444 analog,A2A receptor antagonist 1 | Adenosine Receptor |
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. | |||
T4521 | Edg-2 receptor inhibitor 1 | SAR-100842 | LPA Receptor |
Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM). | |||
T9247 | Vanilloid receptor antagonist 1 | 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile | TRP/TRPV Channel |
Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist. | |||
T15785 | LPA1 receptor antagonist 1 | LPA1 R antagonist 1 | LPA Receptor |
LPA1 receptor antagonist 1(LPA1 R antagonist 1) is a selective and potent lysophosphatidic acid (LPA1) receptor antagonist (IC50 : 25 nM) for the study of idiopathic pulmonary fibrosis. | |||
T37908 | Glucocorticoid receptor agonist-1 | Glucocorticoid Receptor | |
Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1]. | |||
T10307 | AMPA receptor modulator-1 | iGluR | |
AMPA receptor modulator-1 can be activated by glutamate, thereby modulating ion channels. | |||
T10499 | H3 receptor-MO-1 | Histamine Receptor | |
H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders. | |||
T9579L | GLP-1 receptor agonist 9 citrate | GLP-1 receptor agonist 9 citrate (2401892-71-3 Free base) | Glucagon Receptor |
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1. | |||
T11137 | (E)-GABAB receptor antagonist 1 | GABA Receptor | |
(E)-GABAB receptor antagonist 1 is a trans-GABAB receptor antagonist 1. (E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM. GABAB receptor antagonist 1 is ... | |||
T12404 | CCK-A receptor inhibitor 1 | cholecystokinin | |
CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: 340 nM).CCK-A receptor inhibitor 1 can be used for the study of diseases related to the digestive system. |