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Search Results for " anti-histamine "

20

Compounds

Cat No. Product Name Synonyms Targets
T11723L JNJ-39758979 Histamine Receptor
JNJ-39758979 is a selective and high-affinity histamine H4 receptor antagonist (Kis: 12.5, 5.3, and 25 nM for human, mouse, and monkey histamine H4 receptor, respectively). JNJ-39758979 functionally antagonizes histamine...
T22746 Tesmilifene fumarate DPPE fumarate Histamine Receptor
Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。
T0797 Cimetidine SKF-92334 Histamine Receptor
Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological actions. It inhibits GASTRIC ACID secretion, as well as PEP...
T1336 Benztropine mesylate Benzotropine mesylate,Benzatropine mesylate,Benztropine methanesulfonate Dopamine Receptor , AChR , Histamine Receptor
Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON DISEASE. Benztropine also inhibits the uptake of dopamine.
T26253 Tecastemizole Norastemizole,R-43512,R43512,R 43512,T 1348 Histamine Receptor
Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.
T6426 Buclizine dihydrochloride Longifene,Buclina,Buclizine HCl,UCB-4445 5-HT Receptor , AChR , Histamine Receptor
Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and antivertigo activities. Buclizine dihydrochloride binds to and ...
T1110 Meclizine dihydrochloride Meclozine dihydrochloride,NSC28728,Meclizine 2HCl Apoptosis , Histamine Receptor
Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation sickness.
T1090 Perphenazine Perphenazin,Etaperazine,Trilafon CaMK , Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
T0147 Clemastine fumarate HS-592 (fumarate),Meclastine fumarate,Meclastine (fumarate) Autophagy , Histamine Receptor
Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
T27159 DF-1111301 DF1111301,DF 1111301 Platelet aggregation , Histamine Receptor
DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.
T10945 D18024 Others
D18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.
T0298 Dimenhydrinate Dramamine,Chloranautine,Vomex A Histamine Receptor
Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.
T3979 Emedastine LY188695,Emadine Histamine Receptor
Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. Emedastine reversibly and competitively blocks histamine by binding to H1 receptors, thus blocking its...
T20712 Conessine Conessinum,Wrightine,Roquessine,Neriine,Konessin Histamine Receptor
Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.
TN1661 Ganoderic acid C2 Reductase , Histamine Receptor , Immunology/Inflammation related
Ganoderic acid C2 has anti-inflammatory,and anti-tumor-promoting activities. Ganoderic acid C2 can inhibit histamine release, it also has inhibitory effects on the induction of Epstein-Barr Virus early antigen.
T5S1286 (+)-Columbianetin (S)-Columbianetin,Columbianetin Antifungal
(+)-Columbianetin ((S)-Columbianetin) is a new phytoalexin associated with celery (Apium graveolens) resistance to pathogens during storage, it also has antifungal activity. (+)-Columbianetin has anti-inflammatory effect...
T34709 ST-1006 ST 1006 Histamine Receptor
ST-1006 is a potent histamine H4 receptor agonist (pKi: 7.94).ST-1006 has anti-inflammatory effects.ST-1006 is a potent inducer of basophil migration and induces basophil migration.ST-1006 is a potent inducer of basophil...
T0217L (+)-Dropropizine (+)-Dropropizine Histamine Receptor
(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex and by interfering with stimulus activation of peripheral endings of sensory ...
T1639 Amlexanox CHX3673,Amoxanox,AA673 IL Receptor , FGFR , Others , IκB/IKK
Amlexanox (AA673) is an anti-aphthous ulcer drug. Amlexanox inhibits the synthesis and release of inflammatory mediators, including leukotrienes and histamine, from mast cells, neutrophils, and mononuclear cells. Amlexan...
T4195 Betahistine PT 9 base,Vasomotal,Serc base Histamine Receptor
Betahistine (Vasomotal) is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but may exacerbate bronchial asthma and peptic ulcers. Betahisti...

Compounds

JNJ-39758979
T11723L
Synonym:
Target: Histamine Receptor
Tesmilifene fumarate
T22746
Synonym: DPPE fumarate
Target: Histamine Receptor
Cimetidine
T0797
Synonym: SKF-92334
Target: Histamine Receptor
Benztropine mesylate
T1336
Synonym: Benzotropine mesylate,Benzatropine mesylate,Benztropine methanesulfonate
Target: Dopamine Receptor, AChR, Histamine Receptor
Tecastemizole
T26253
Synonym: Norastemizole,R-43512,R43512,R 43512,T 1348
Target: Histamine Receptor
Buclizine dihydrochloride
T6426
Synonym: Longifene,Buclina,Buclizine HCl,UCB-4445
Target: 5-HT Receptor, AChR, Histamine Receptor
Meclizine dihydrochloride
T1110
Synonym: Meclozine dihydrochloride,NSC28728,Meclizine 2HCl
Target: Apoptosis, Histamine Receptor
Perphenazine
T1090
Synonym: Perphenazin,Etaperazine,Trilafon
Target: CaMK, Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Clemastine fumarate
T0147
Synonym: HS-592 (fumarate),Meclastine fumarate,Meclastine (fumarate)
Target: Autophagy, Histamine Receptor
DF-1111301
T27159
Synonym: DF1111301,DF 1111301
Target: Platelet aggregation, Histamine Receptor
D18024
T10945
Synonym:
Target: Others
Dimenhydrinate
T0298
Synonym: Dramamine,Chloranautine,Vomex A
Target: Histamine Receptor
Emedastine
T3979
Synonym: LY188695,Emadine
Target: Histamine Receptor
Conessine
T20712
Synonym: Conessinum,Wrightine,Roquessine,Neriine,Konessin
Target: Histamine Receptor
Ganoderic acid C2
TN1661
Synonym:
Target: Reductase, Histamine Receptor, Immunology/Inflammation related
(+)-Columbianetin
T5S1286
Synonym: (S)-Columbianetin,Columbianetin
Target: Antifungal
ST-1006
T34709
Synonym: ST 1006
Target: Histamine Receptor
(+)-Dropropizine
T0217L
Synonym: (+)-Dropropizine
Target: Histamine Receptor
Amlexanox
T1639
Synonym: CHX3673,Amoxanox,AA673
Target: IL Receptor, FGFR, Others, IκB/IKK
Betahistine
T4195
Synonym: PT 9 base,Vasomotal,Serc base
Target: Histamine Receptor
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TargetMol