Powder: -20°C for 3 years | In solvent: -80°C for 1 year
ST-1006 is a potent histamine H4 receptor agonist (pKi: 7.94).ST-1006 has anti-inflammatory effects.ST-1006 is a potent inducer of basophil migration and induces basophil migration.ST-1006 is a potent inducer of basophil migration. ST-1006 has anti-inflammatory and anti-pruritic effects.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 197.00 | |
2 mg | In stock | $ 293.00 | |
5 mg | In stock | $ 496.00 | |
10 mg | In stock | $ 795.00 | |
25 mg | In stock | $ 1,290.00 | |
50 mg | In stock | $ 1,590.00 | |
100 mg | In stock | $ 1,980.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 562.00 |
Description | ST-1006 is a potent histamine H4 receptor agonist (pKi: 7.94).ST-1006 has anti-inflammatory effects.ST-1006 is a potent inducer of basophil migration and induces basophil migration.ST-1006 is a potent inducer of basophil migration. ST-1006 has anti-inflammatory and anti-pruritic effects. |
Targets&IC50 | H4 receptor:7.94(pKi ) |
In vitro |
ST-1006 (10 μM) is an effective inducer of eosinophil migration, promoting eosinophil migration [3]. ST-1006 (0-100 μM) inhibits FceRI-mediated eosinophil activation and reduces the expression levels of CD63 and CD203c in activated eosinophils through FceRI activation [3]. |
In vivo | ST-1006 (1-100 mg/kg; s.c.; male CD-1 mice) exhibits anti-inflammatory and anti-itch properties [5]. |
Synonyms | ST 1006 |
Molecular Weight | 367.28 |
Formula | C16H20Cl2N6 |
CAS No. | 1196994-11-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 3.67 mg/mL (10 mM)
You can also refer to dose conversion for different animals. More
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ST-1006 1196994-11-2 GPCR/G Protein Immunology/Inflammation Neuroscience Histamine Receptor ST1006 ST 1006 inhibitor inhibit