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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T28357 | PET-16 | PET16,PET 16 | |
PET-16 is a HSP70 inhibitor. | |||
T23252 | Rp-8-Br-PET-cGMPS | Others | |
cGMP-dependent protein kinase (PKG) inhibitor | |||
T79577 | CB2 PET Radioligand 1 | Cannabinoid Receptor | |
CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.7 nM). It is synthesized via Cu-mediated 18F-fluorination an... | |||
T8637 | DMNB | 6-Nitroveratraldehyde | DNA-PK |
DMNB (6-Nitroveratraldehyde) is DNA-dependent protein kinase (DNA-PK) inhibitor with IC50 of 15 μM, an enzyme involved in the non-homologous end-joining (NHEJ) pathway of double-stranded DNA break (DSB) repair in human c... | |||
T17842 | DOTA-NHS-ester | Others | |
DOTA-NHS-ester is a linker of affibody molecules for small animal PET, SPECT and CT. DOTA-NHS-ester can be used to label radiotherapeutic agents or imaging probes for tumor detection. | |||
T7196 | HG-10-102-01 | LRRK2 | |
HG-10-102-01 is an inhibitor of leucine-rich repeat kinase 2 (LRRK2, IC50 of 20.3 nM). | |||
TN1711 | Gossypetin | Antioxidant , p38 MAPK , MAPK , Antibacterial | |
Gossypetin, a hexahydroxylated flavonoid extractable from Rhodiola rosea Linn. is a potent MKK3 and MKK6 inhibitor that strongly attenuates the MKK3/6-p38 signaling pathway.Gossypetin exhibits antimutagenic, antiatherosc... | |||
T31614 | Elpetrigine | GW-273293,JZP 4,JZP4,GW273293,JZP-4,GW 273293 | |
Elpetrigine( GW 273293, JZP-4) is effective calcium and sodium channel blocker and is currently being evaluated in patients as an anticonvulsant and mood stabilizer. | |||
T8287 | Edpetiline | Sipeimine-3β-D-glucoside | Others |
Edpetiline(Sipeimine-3β-D-glucoside), a principal alkaloid from P. eduardi., has significant anti-inflammatory effects. | |||
T76890 | Petosemtamab | MCLA 158 | EGFR |
Petosemtamab (MCLA 158) is a highly potent monoclonal antibody against EGFR (Kd: 0.22 nM) and LGR5 (Kd: 0.86 nM). Petosemtamab promotes EGFR signaling disruption and receptor breakdown in LGR5+ cancer cells. Petosemtamab... | |||
T4870 | Petroselinic acid | 5-Heptadecylene-1-carboxylic acid | Endogenous Metabolite |
Petroselinic acid (5-Heptadecylene-1-carboxylic acid) is a monounsaturated omega-12 fatty acid found naturally in plant and animal oils and fats. | |||
T9409 | Mesdopetam hemitartrate | IRL790 hemitartrate,1-Propanamine, N-[2-[3-fluoro-5-(methylsulfonyl)phenoxy]ethyl]-, (2R,3R)-2,3-dihydroxybutanedioate (2:1) | Dopamine Receptor |
Mesdopetam hemitartrate (IRL790 hemitartrate) is an antagonist of dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM for human recombinant D3 receptor). It has psychomotor stabilizing properties. | |||
T31648 | Epetirimod | S 30563,S-30563,S30563 | Antiviral |
Epetirimod (S-30563) is a small molecule immunomodulator with antitumor and anti-infective activity for the study of papillomavirus infections. | |||
TN1154 | Nepetin | 6-Methoxyluteolin | Calcium Channel , Histamine Receptor |
Nepetin (6-Methoxyluteolin) has antioxidant activity, it is a potent inhibitor of histamine release and calcium influx via down-regulation of the FcεRI α chain. | |||
T4045 | Epetraborole hydrochloride | GSK2251052 hydrochloride | Antibacterial |
Epetraborole hydrochloride (GSK2251052 hydrochloride) is a potent and selective leucyl-tRNA synthetase inhibitor. | |||
T38828 | Mesdopetam | IRL790 | |
Mesdopetam (IRL790) is a dopamine D3 receptor antagonist with a Ki of 90 nM and an IC50 of 9.8 μM for the human recombinant D3 receptor. It exhibits psychomotor stabilizing properties and is utilized in the study of moto... | |||
T126078 | 6-Dehydropetasol | ||
6-Dehydropetasol is a useful organic compound for research related to life sciences. The catalog number is T126078 and the CAS number is 129704-82-1. | |||
TN3530 | Borapetoside B | Others | |
Borapetoside B is a natural product of Tinospora, Menispermaceae. The catalog number is TN3530 and the CAS number is 104901-05-5. Borapetoside B can be used as a reference standard. | |||
TN1732 | Herpetone | HBV | |
Herpetone exhibits protective effects on CCl(4)-induced hepatocyte injury, it shows anti-hepatitis B virus (HBV) activity. | |||
TN4264 | Isoapetalic acid | HIV Protease , Antifection | |
Isoapetalic acid and apetalic acid exhibit cytotoxic activities towards both cancer cell lines(human breast cancer (MCF-7) and human lung carcinoma (A-549) cell lines) and both Gram-positive bacteria(two Gram-positive ba... |