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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T22223 | 3PO | Glucokinase , Autophagy | |
3PO is a small-molecule inhibitor of PFKFB3 (IC50: 22.9 μM), inhibiting the proliferation of several human malignant hematopoietic and adenocarcinoma cell lines (IC50: 1.4-24 μM). It suppresses glucose uptake, and decrea... | |||
T8574 | SPHINX | Others | |
SPHINX is a new generation inhibitor of SPRK1 | |||
T14557 | BI-1935 | Epoxide Hydrolase | |
BI-1935 is an inhibitor of soluble epoxide hydrolase (sEH). For diseases related to cardiovascular disease. | |||
T7156 | NIBR189 | EBI2/GPR183 | |
NIBR189 is a potent and selective antagonist of EBI2 (GPR183) receptor (IC50 of 11 and 15 nM for human and mouse EBI2 receptors, respectively) | |||
T6031 | GNE0877 | GNE 0877,GNE-0877 | LRRK2 |
GNE0877 (GNE 0877) is a highly effective and specific leucine-rich repeat kinase 2 (LRRK2) inhibitor (Ki: 0.7 nM). | |||
T14074 | A-770041 | Src | |
A-770041 is a selective and orally active inhibitor targeting the Src-family kinase, Lck, which plays a crucial role in T-cell signaling. With an IC50 value of 147 nM at 1 mM ATP, A-770041 demonstrates high specificity b... | |||
T28881 | Sulmazole | Vardax,AR-L 115BS,AR-L 115-BS | PDE , Parasite , Adenosine Receptor |
Sulmazole (AR-L 115-BS) is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.Sulmazole has been shown to improve cardiac index, low pulmonary... | |||
T15471 | Hepronicate | Megrin | Others |
Hepronicate(Megrin) is a small molecule compound with hypolipidemic and vasodilatory activity. | |||
T29041 | UCCF-853 | UCCF853,UCCF 853 | CFTR |
UCCF-853 is a small-molecule CFTR modulator that can be used to study cystic fibrosis. | |||
T68018 | Tuvatexib | VDAC | |
Tuvatexib is a small molecule VDAC/HK2 dual modulator. | |||
T28817 | SM4 | SM-4,SM 4 | Others |
SM4 is a SOX18 small molecule inhibitor of HemSC vessel formation in vivo. | |||
T27838 | Lirequinil | RO413696,RO-413696,RO41-3696,RO 413696,Ro 41-3696,Ro-41-3696 | GABA Receptor |
Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders. | |||
T33940 | PF-03382792 | PF 03382792,PF03382792 | 5-HT Receptor |
PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease. | |||
TNU0685 | Dipropofol | 4,4-Bis(2,6-di-isopropylphenol) | GABA Receptor |
Dipropofol (4,4-Bis(2,6-di-isopropylphenol)) is a small molecule GABAA receptor agonist that can be used to study epilepsy. | |||
T9995 | Antituberculosis agent-5 | Others | |
Antituberculosis agent-5 is a small molecule used for high-throughput assays. | |||
T2545 | Lomitapide Mesylate | BMS-201038 mesylate,AEGR-733 mesylate | CETP |
Lomitapide Mesylate (BMS-201038 mesylate) is a methanesulfonic acid form of lomitapide, a small molecule inhibitor of microsomal triglyceride transfer protein. | |||
T2281 | GSK2256098 | GSK 2256098,GSK-2256098,GTPL7939 | Apoptosis , FAK |
GSK2256098 (GTPL7939) is a small molecule FAK kinase inhibitor. | |||
T9359 | PDL-1 cpd 10 | PD-1/PD-L1 | |
PDL-1 cpd 10 is a novel small molecule PD-L1 inhititor. | |||
T61172 | NRX-1532 | NRX1532,NRX 1532 | Others |
NRX-1532 is a small molecule β-catenin:β-TrCP interaction enhancer. | |||
T27122 | Dasantafil | SCH446132,SCH-446132,SCH 446132 | PDE |
Dasantafil (SCH446132) is a small molecule phosphodiesterase-5A (PDE5A) inhibitor used to treat genitourinary disorders and study erectile dysfunction. |