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20

Compounds

Cat No. Product Name Synonyms Targets
T37101 1-Hydroxyanthraquinone DNA/RNA Synthesis
1-Hydroxyanthraquinone is an anthraquinone that has been found in Morinda officinalis and has genotoxic and carcinogenic activities. 1-Hydroxyanthraquinone generates strong DNA repair response.
T3381 Lysionotin Others
Lysionotin (Nevadensin) has expectorant, eliminating phlegm, softening effects.
T0793 Kanamycin sulfate Kanamycin monosulfate,Kanamycin A monosulfate,Ophtalmokalixan ribosome , Antibacterial , Antibiotic
Kanamycin sulfate (Kanamycin monosulfate) is an aminoglycoside bacteriocidal antibiotic.
T8065 Tiamulin Thiamutilin Others , Antibacterial , Antibiotic
Tiamulin (Thiamutilin) is a semisynthetic pleuromutilin antibiotic
T6231 Tebipenem Pivoxil ME1211,Orapenem Antibacterial , Antibiotic
Tebipenem Pivoxil (Orapenem) , an orally activity carbapenem antibiotic, is utilized in treating otolaryngologic and respiratory infections.
T1491 Atovaquone Atavaquone Others , P450 , Dehydrogenase , Antibiotic , Parasite
Atovaquone (Atavaquone) is a hydroxynaphthoquinone that has antimicrobial activity and is being used in antimalarial protocols.
T23133 Pentamidine Phosphatase , Antibacterial , Antibiotic , Parasite , Antifungal
Pentamidine is an antifungal and antiprotozoal agent, interacting directly with the pathogen genome by binding to AT-rich regions of duplex DNA and the minor groove of DNA, thereby interfering with DNA replication.
T3907 Tenuigenin Senegenin,Senegin NF-κB , Caspase , Antibacterial
Tenuigenin (Senegenin) is a natural product from Polygala tenuifolia used in Chinese medicine with antioxidative and anti-inflammatory activity.
T4267 Tulathromycin A CP 472295,Draxxin,Tulathromycin Antibacterial , Antibiotic
Tulathromycin A (CP 472295) is a macrolide antibiotic.
T5189 Omadacycline PTK 0796,Amadacycline ribosome , Antibacterial , Antibiotic
Omadacycline (Amadacycline), a new tetracycline antibiotic, can inhibit the 30s subunit of bacterial ribosome.
T2691 Oritavancin diphosphate LY333328 diphosphate Others , Antibacterial , Antibiotic
Oritavancin diphosphate (LY333328 diphosphate) is a novel semisynthetic glycopeptide antibiotic which is being developed for the treatment of serious Gram-positive bacterial infections.
T1262 Tazobactam Tazobactamum,Tazobactam acid,YTR-830H,CL-298741 Antibacterial , Antibiotic
Tazobactam (YTR-830H) is an antibacterial penicillin derivative which inhibits the action of bacterial beta-lactamases.
T1654 Pentamidine isethionate Pentamidine isethionate salt,Pentamidine diisethionate Phosphatase , Antibacterial , Antibiotic , Parasite , Antifungal
Pentamidine isethionate (Pentamidine diisethionate) is a synthetic amidine derivative, Pentamidine Isethionate is an antiprotozoal and antifungal agent.
T4201 Avibactam sodium AVE-1330A,NXL-104 Antibacterial , Antibiotic
Avibactam sodium (NXL-104) is a reversible β-lactamase inhibitor (IC50: 8/80/38 nM, for TEM-1/P99/KPC-2 β-lactamases).
T0331 Moxifloxacin hydrochloride BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl Topoisomerase , Antibacterial , Antibiotic
Moxifloxacin hydrochloride (BAY12-8039 HCl) is a fourth generation fluoroquinolone with expanded activity against gram-positive bacteria as well as atypical pathogens. Moxifloxacin has been linked to mild ALT elevations ...
T1153 Trimethoprim NIH 204,BW 56-72,NSC-106568 DHFR , DNA/RNA Synthesis , Antifolate , Antibacterial , Antibiotic
Trimethoprim (NSC-106568) is a Dihydrofolate Reductase Inhibitor Antibacterial. The mechanism of action of trimethoprim is as a Dihydrofolate Reductase Inhibitor, and Cytochrome P450 2C8 Inhibitor, and Organic Cation Tra...
T23132 Pentamidine dihydrochloride MP-601205 dihydrochloride Phosphatase , Antibacterial , Antibiotic , Parasite , Antifungal
Pentamidine dihydrochloride (MP-601205 dihydrochloride) is an aromatic diamidine agent with activity against a number of microorganisms including protozoa (Trypanosoma brucei, Leishmania spp., and Babesia spp.) and fungi...
T7804 Garenoxacin mesylate hydrate Garenoxacin mesylate [USAN],BMS284756 (Mesylate hydrate) Antibacterial
Garenoxacin mesylate hydrate (Garenoxacin mesylate [USAN]) with potent antimicrobial activity, against common respiratory pathogens, including resistant strains.
T7179 Garenoxacin BMS284756 Antibacterial
Garenoxacin (BMS284756) is a novel oral des-fluoro(6) quinolone for the treatment of Gram-positive and Gram-negative bacterial infections.
T79088 Chlamydia pneumoniae-IN-1
Chlamydia pneumoniae-IN-1 (compound 55), a benzimidazole derivative, exhibits potent antibacterial activity, inhibiting 99% of C. pneumoniae growth at a concentration of 10 μM and maintaining 95% viability of the host ce...

Compounds

1-Hydroxyanthraquinone
T37101
Synonym:
Target: DNA/RNA Synthesis
Lysionotin
T3381
Synonym:
Target: Others
Kanamycin sulfate
T0793
Synonym: Kanamycin monosulfate,Kanamycin A monosulfate,Ophtalmokalixan
Target: ribosome, Antibacterial, Antibiotic
Tiamulin
T8065
Synonym: Thiamutilin
Target: Others, Antibacterial, Antibiotic
Tebipenem Pivoxil
T6231
Synonym: ME1211,Orapenem
Target: Antibacterial, Antibiotic
Atovaquone
T1491
Synonym: Atavaquone
Target: Others, P450, Dehydrogenase, Antibiotic, Parasite
Pentamidine
T23133
Synonym:
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Tenuigenin
T3907
Synonym: Senegenin,Senegin
Target: NF-κB, Caspase, Antibacterial
Tulathromycin A
T4267
Synonym: CP 472295,Draxxin,Tulathromycin
Target: Antibacterial, Antibiotic
Omadacycline
T5189
Synonym: PTK 0796,Amadacycline
Target: ribosome, Antibacterial, Antibiotic
Oritavancin diphosphate
T2691
Synonym: LY333328 diphosphate
Target: Others, Antibacterial, Antibiotic
Tazobactam
T1262
Synonym: Tazobactamum,Tazobactam acid,YTR-830H,CL-298741
Target: Antibacterial, Antibiotic
Pentamidine isethionate
T1654
Synonym: Pentamidine isethionate salt,Pentamidine diisethionate
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Avibactam sodium
T4201
Synonym: AVE-1330A,NXL-104
Target: Antibacterial, Antibiotic
Moxifloxacin hydrochloride
T0331
Synonym: BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl
Target: Topoisomerase, Antibacterial, Antibiotic
Trimethoprim
T1153
Synonym: NIH 204,BW 56-72,NSC-106568
Target: DHFR, DNA/RNA Synthesis, Antifolate, Antibacterial, Antibiotic
Pentamidine dihydrochloride
T23132
Synonym: MP-601205 dihydrochloride
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Garenoxacin mesylate hydrate
T7804
Synonym: Garenoxacin mesylate [USAN],BMS284756 (Mesylate hydrate)
Target: Antibacterial
Garenoxacin
T7179
Synonym: BMS284756
Target: Antibacterial
Chlamydia pneumoniae-IN-1
T79088
Synonym:
Target:
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TargetMol