partial — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T4246	Varenicline dihydrochloride		AChR
	Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.		AChR
T12855	SB 258719		5-HT Receptor
	SB 258719 is a selective antagonist of 5-HT7 receptor(pKi of 7.5).		5-HT Receptor
T3565	VU0155041	UV0155041,VU-0155041	GluR
	VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).		GluR
T22016	A-582941 dihydrochloride	A 582941	5-HT Receptor , AChR
	A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial		5-HT Receptor , AChR
T7806	Licarbazepine	10,11-hydroxy-10,11 Dihydrocarbamezer	Others
	Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial seizures and bipolar disorders.		Others
T26890	BP14979	BP 14979,BP1,4979,BP-14979,BP 1,4979,BP-1,4979
	BP14979 is D3R-selective partial agonist.
TP2048L	α-helical CRF 9-41 acetate	α-helical CRF 9-41 acetate(90880-23-2 Free base)	CRFR
	α-helical CRF 9-41 acetate is a competitive antagonist of CRF2 (KB = 100 nM) and a partial agonist of CRF1 (EC50 = 140 nM).		CRFR
T22817	GSK 789472 hydrochloride	GSK-789472 HCl,1-phenyl-3-(piperidin-2-ylmethyl)imidazolidin-2-one hydrochloride,4,5-Dihydro-1-phenyl-3-(2-piperidinyl)methylimidazol-2(1H)-one	Dopamine Receptor
	GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.		Dopamine Receptor
T28303	Pazinaclone	A-77000,DN-2327,DN2327,DN 2327,A 77000,A77000	GABA Receptor
	Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.		GABA Receptor
T22671	CJ 033466		5-HT Receptor
	CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.		5-HT Receptor
T3285L	Eslicarbazepine	Pazzul,EC 810-248-9,BIA 2-194,Stedesa,Erelib	Beta-Secretase , Sodium Channel
	Eslicarbazepine (Stedesa) can be used for adjunctive therapy for adults with partial-onset seizures.		Beta-Secretase , Sodium Channel
T72027	6-Methyl-3-pyridinecarboxaldehyde	6-Methoxynicotinaldehyde
	6-Methyl-3-pyridinecarboxaldehyde (6-Methoxynicotinaldehyde) has partial antitumor activity.
T27845	Losigamone	ADD-137022,AO33,AO 33,ADD 137022,AO-33,ADD137022;Losigamone	GABA Receptor
	Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures.		GABA Receptor
T22348	Isonipecotic acid	4-Piperidinecarboxylic acid,Hexahydroisonicotinic acid,4-Carboxypiperidine	GABA Receptor
	Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.		GABA Receptor
T3431	Pardoprunox hydrochloride	SLV-308 hydrochloride,DU-126891 hydrochloride	Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
	Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist and 5-HT1A recept...		Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
T0818	Decamethonium bromide	Decacuran,Syncurine	AChR , AChE
	Decamethonium bromide (Syncurine) is a neuromuscular blocker and nicotinic AChR partial agonist.		AChR , AChE
T68154	TC-2216		AChR
	TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to treat anxiety and depression.		AChR
T23168	PNU 22394 hydrochloride		5-HT Receptor
	PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist		5-HT Receptor
T13424	(1R,2S)-VU0155041		GluR
	(1R,2S)-VU0155041 is the cis regioisomer of VU0155041 and a partial agonist of mGluR4.		GluR
T68065	Enloplatin
	Enloplatin is a carboplatin analog that has a partial role in advanced ovarian cancer.