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Varenicline dihydrochloride

Name: Varenicline dihydrochloride
Brand: TargetMol
SKU: T4246
Price: 67 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T4246Cas No. 866823-63-4

Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.

Varenicline dihydrochloride

🥰Excellent

Purity: 99.97%

Catalog No. T4246Cas No. 866823-63-4

Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.

Pack Size	Price	Availability
5 mg	$67	In Stock
10 mg	$97	In Stock
25 mg	$187	In Stock
50 mg	$281	In Stock
100 mg	$421	In Stock
1 mL x 10 mM (in DMSO)	$74	In Stock

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Batch Information

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Purity:99.97%

Resource Download

COA HNMR

Product Introduction

Bioactivity

Description

Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.

Chemical Properties

Molecular Weight	284.18
Formula	C₁₃H₁₅Cl₂N₃
Cas No.	866823-63-4
Smiles	Cl.Cl.c1c4c(cc2nccnc12)C3CC4CNC3
Relative Density.	no data available
Color	Yellow
Appearance	Solid

Storage & Solubility Information

Storage

store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (175.94 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.5189 mL	17.5945 mL	35.1890 mL	175.9448 mL
5 mM	0.7038 mL	3.5189 mL	7.0378 mL	35.1890 mL
10 mM	0.3519 mL	1.7594 mL	3.5189 mL	17.5945 mL
20 mM	0.1759 mL	0.8797 mL	1.7594 mL	8.7972 mL
50 mM	0.0704 mL	0.3519 mL	0.7038 mL	3.5189 mL
100 mM	0.0352 mL	0.1759 mL	0.3519 mL	1.7594 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc