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20

Compounds

Cat No. Product Name Synonyms Targets
T8134 Cefathiamidine Antibacterial , Antibiotic
Cefathiamidine exhibits a wide spectrum of antimicrobial activity against bacteria. Cefathiamidine is used for the treatment of respiratory, liver, five senses, urinary tract infections, endocarditis and sepsis
T8345 Carbutamide Others
Carbutamide is a sulfonylurea antidiabetic agent with hypoglycemic activity.
T15656 KGA-2727 SGLT
KGA-2727 is a potent and selective SGLT1 inhibitor, with Kis of 97.4 nM and 43.5 nM for human and rat SGLT1, respectively. The selectivity ratios (Ki for SGLT2/Ki for SGLT1) of KGA-2727 are 140 (human) and 390 (rat). KGA...
T6451 Clodronic acid disodium salt Loron,Clodronate Disodium,Lodronate Others
Clodronic acid disodium salt (Lodronate), a bisphosphonate, is a potent antiosteolytic agent which inhibits bone resorption.
T0370 Pheniramine maleate Daneral,Inhiston,Trimetose 5-HT Receptor , Histamine Receptor
Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors, thereby inhibiting phospholipase A2 and production of the endothelium-derived re...
T0141 Cephalonium Cefalonium Others
Cephalonium (Cefalonium) is a first-generation cephalosporin antibiotic.
TP1419L HAEGTFT acetate(926018-95-3 free base) Glucagon Receptor
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
TP1381L HAEGT TFA(852155-81-8 free base) Others
HAEGT TFA is the first N-terminal 1-5 residues of GLP-1 peptide.
T8063 Cephapirin Benzathine Others , Antibacterial , Antibiotic
Cephapirin Benzathine is a semisynthetic, broad-spectrum, first-generation cephalosporin with antibacterial activity.
T0803 Acetrizoic acid Urokon,Opacaron,Acetrizoesaeure Others
Acetrizoic acid (Urokon) is the first monomeric ionic compound used as an X-ray contrast agent.
T4584 BMS-813160 BMS 813160 CCR
BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.
T2733 Sarsasapogenin Parigenin,Sarsagenin Apoptosis , NF-κB , Endogenous Metabolite
Sarsasapogenin (Parigenin) is a steroidal sapogenin, that is the aglycosidic portion of a plant saponin. It is named after sarsaparilla (Smilax sp.), a family of climbing plants found in subtropical regions. It was one o...
T26195 SMI481 NPPM-6748-481,NPPM 6748-481,NPPM6748481,SMI-481 SMI 481,NPPM 6748481 Others
SMI481 (NPPM6748481) is the first small-molecule Sec14-like phosphatidylinositol transfer proteins (PITPs) inhibitor.
T9901 Adalimumab TNF
Adalimumab (anti-TNF-alpha) is the first fully human recombinant IgG1 monoclonal antibody that specifically targets human TNF-alpha.
T5763 Sedanolide Others , Autophagy
Sedanolide is a natural phthalide first isolated from seed oil of the Umbelliferae family, including celery.
T6859 I-BRD9 GSK602 Epigenetic Reader Domain
I-BRD9 (GSK602) is the first selective cellular inhibitor for BRD9 with pIC50 of 7.3.
T4S0647 Butylphthalide 3-Butylphthalide,3-n-Butylphathlide,3-n-Butylphthalide Others
Butylphthalide (3-Butylphthalide) is an anti-cerebral-ischemia drug; first isolated from the seeds of Apium graveolens Linn.
T14547 JWG-071 JWG071,JWG 071 ERK , Epigenetic Reader Domain
JWG-071, the first reported chemical probe for ERK5 kinase selectivity, is a BET-selective inhibitor with a 1 μM BRD4 IC that enhances both ERK5 activity and BRD4 selectivity.
T8374 LJ570 PPAR
LJ570 is the first PPARα/γ dual agonist (PPARα,PPARγ with EC50s of 1.05 and 0.12 μM, respectively[)
TP1382L HAEGTFTSDVS acetate HAEGTFTSDVS acetate(864915-61-7 free base) Glucagon Receptor
HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells.
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TargetMol