besylate — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T6177	PF-562271 besylate	PF-00562271 Besylate	FAK , PYK2 , CDK
	PF-562271 besylate (PF-00562271 Besylate) is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of 1.5 nM, ~10-fold less potent for Pyk2 than FAK and >100-fold selectivity against other protein kinases, exc...		FAK , PYK2 , CDK
T4284	Levamlodipine besylate	(S)-Amlodipine Besylate (103129-82-4(free base))	Calcium Channel
	Levamlodipine besylate ((S)-Amlodipine Besylate (103129-82-4(free base))) , also known as S-amlodipine, is a pharmacologically active enantiomer of amlodipine, an antihypertensive and anti-anginal medication. Levamlodipi...		Calcium Channel
T0231	Amlodipine Besylate	Amlodipine benzenesulfonate	Calcium Channel
	Amlodipine Besylate(Amlodipine benzenesulfonate) is a long-lasting calcium channel blocker.		Calcium Channel
T1459	Cisatracurium besylate	51W89	Adrenergic Receptor , AChR , Autophagy
	Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant for intravenous administration.		Adrenergic Receptor , AChR , Autophagy
T6397	Atracurium besylate	Tracrium,51W89,BW-33A	AChR
	Atracurium besylate (51W89) is a non-depolarizing neuromuscular blocking agent with short duration of action. Its lack of significant cardiovascular effects and its lack of dependence on good kidney function for eliminat...		AChR
T3086	Mesoridazine Besylate	Mesoridazine benzenesulfonate,Serentil	Dopamine Receptor , 5-HT Receptor
	Mesoridazine Besylate (Serentil) is a piperidine neuroleptic drug belonging to the class of drugs called phenothiazines, used in the treatment of schizophrenia. It is a metabolite of thioridazine.		Dopamine Receptor , 5-HT Receptor
T11472L	Molibresib besylate	I-BET 762 besylate,GSK 525762C	CCR
	Molibresib besylate is an inhibitor of BET bromodomain (IC50: 32.5-42.5 nM).		CCR
T14357	Spebrutinib besylate	CC-292 (besylate),AVL-292 (benzenesulfonate)	BTK
	Spebrutinib besylate (AVL-292 benzenesulfonate; CC-292 besylate) is a Btk kinase activity inhibitor (IC50<0.5 nM, Kinact/Ki=7.69×104 M-1s-1s).		BTK
T6174	R406	R-406 besylate	Apoptosis , FLT , Syk
	R406 (R-406 besylate) is an effective Syk inhibitor (IC50: 41 nM) and shows no effects on Lyn.		Apoptosis , FLT , Syk
T0231L3	Amlodipine besylate monohydrate
	Amlodipine besylate monohydrate is a medication used to lower blood pressure and prevent chest pain.
T69399	MK-0359 besylate
	MK-0359 besylate is a Phosphodiesterase-4 (PDE4) inhibitor.
T68567	AMG-131 besylate
	AMG-131 besylate is a hypoglycemic agent. It is a potent PPARγ partial agonist that displays robust glucose-lowering activity in rodent models of diabetes while exhibiting a reduced side-effects profile compared to marke...
T70158	Quilseconazole besylate
	Quilseconazole besylate, also known as VT-1129 besylate, is a potent, orally active fungal Cyp51 (lanosterol 14-α-demethylase) inhibitor.
T10589	BPN-15606 besylate (1914989-49-3 free base)	BPN-15606 besylate	Others
	BPN-15606 besylate is a highly potent, orally active γ-secretase modulator, attenuates the production of Aβ40 and Aβ42 by SHSY5Y neuroblastoma cells (IC50s: 7 nM and 17nM).		Others
T11400	Gisadenafil besylate	UK 369003-26	Others
	Gisadenafil besylate (UK 369003-26) is a specific, orally active phosphodiesterase 5 (PDE5) inhibitor ,prevents degradation of cyclic guanosine monophosphate (cGMP), with an IC50 of 3.6 nM .		Others
T30001	Amlodipine besylate, (R)-
	Amlodipine besylate, (R)- is a medication used to lower blood pressure and prevent chest pain.
T31647	Epelsiban besylate	GSK-557296B,GSK557296B
	Epelsiban Besylate is an oral drug that is a highly selective anamol oxytocin receptor antagonist.
T78217	(R)-Azasetron besylate	SENS-401	Phosphatase
	(R)-Azasetron besylate (SENS-401), an orally active calcineurin inhibitor, has been shown to mitigate cisplatin-induced hearing loss and cochlear damage [1][2].		Phosphatase
T64425	Crenolanib besylate
	Crenolanib besylate is a useful organic compound for research related to life sciences and the catalog number is T64425.
T61434	Mirogabalin besylate
	Mirogabalin besylate is a potent and orally active ligand that selectively targets the α2δ subunit of voltage-gated calcium channels. It displays high affinity (K d ) values, namely 13.5 nM, 22.7 nM, 27 nM, and 47.6 nM, ...