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Cat No. | Product Name | Synonyms | Targets |
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TNU0541 | 8-Azaguanosine | Nucleoside Antimetabolite/Analog | |
8-Azaguanosine is a purine nucleoside analog with a broad spectrum of antitumor activity and is used in the study of a variety of tumor diseases. | |||
T25742 | Linzagolix choline | GNRH Receptor | |
Linzagolix choline is an orally available non-peptide gonadotropin-releasing hormone (GnRH) antagonist. It can be used to study pain associated with uterine fibroids and endometriosis. | |||
T6236 | Ozagrel | OKY-046,Domenan | Thrombin , Prostaglandin Receptor |
Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of postoperative cerebrovascular contraction and accompanying cerebral isch... | |||
T16083 | Mizagliflozin | GSK-1614235 free base,KGA-3235 free base,DSP-3235 free base | SGLT |
Mizagliflozin (GSK-1614235 free base) is a sodium-glucose transporter inhibitor( Ki of 27 nM for human SGLT1). Mizagliflozin displays 303-fold selectivity over SGLT2. Mizagliflozin is used as an antidiabetic drug that ca... | |||
T12883 | Fezagepras | PBI-4050,Setogepram | GPR |
Fezagepras (Setogepram) is an orally active GPR40 agonist and is an antagonist or inverse agonist of GPR84 with anti-inflammatory, anti-fibrotic, and anti-proliferative actions. | |||
T27837 | Linzagolix | GNRH Receptor | |
Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei Pharmaceutical and ObsEva for the treatment of uterine fibroids,... | |||
T76726 | Zagotenemab | LY33003560 | Microtubule Associated |
Zagotenemab is a humanized antibody against the microtubule-associated protein tau that selectively regulates tau deposits in the brain. Zagotenemab can be used to study neurological disorders such as Alzheimer's disease... | |||
T15159 | Dorzagliatin | HMS5552 | Glucokinase |
Dorzagliatin (HMS5552) is a dual-acting glucokinase (GK) activator. It also improves glycaemic control and pancreatic β-cell function in type 2 diabetes. | |||
T6625 | Ozagrel hydrochloride | Ozagrel HCl,OKY-046 HCl | Thrombin , Prostaglandin Receptor |
Ozagrel hydrochloride (OKY-046 HCl) is a selective thromboxane A(2) synthetase inhibitor used for the improvement of postoperative cerebrovascular contraction and accompanying cerebral ischaemia. | |||
T12375 | Fezagepras sodium | Setogepram sodium salt,PBI-4050 sodium salt | GPR |
Fezagepras sodium (Setogepram sodium salt) is an orally active GPR40 agonist and is an antagonist or inverse agonist for GPR84, with anti-fibrotic, anti-inflammatory and anti-proliferative actions. | |||
T76620 | (D-Tyr5,D-Ser(tBu)6,Azagly10)-LHRH | ||
(D-Tyr5,D-Ser(tBu)6,Azagly10)-LHRH, an analogue of luteinizing hormone-releasing hormone (LHRH), plays a pivotal role in reproductive control by promoting the pituitary release of luteinizing hormone (LH) and follicle-st... | |||
T76615 | (D-Ser(tBu)6,D-Leu7,Azagly10)-LHRH | ||
(D-Ser(tBu)6,D-Leu7,Azagly10)-LHRH, an analogue of the luteinizing hormone-releasing hormone (LHRH), fundamentally mediates reproductive processes by promoting the secretion of pituitary luteinizing hormone (LH) and foll... | |||
TNU0180 | 7-Deazaguanosine | ||
Nucleoside Derivatives - 7-Deaza-purine nucleosides; Drugs and Inhibitors; Antiviral agent, anti-HCV | |||
T69792 | Atuzaginstat | ||
Atuzaginstat is a bacterial protease lysine gingipain inhibitor. | |||
TNU0275 | 8-Aza-7-bromo-7-deazaguanosine | ||
8-Aza-7-bromo-7-deazaguanosine is a Nucleoside Derivative - 7-Deaza-8-aza-purine nucleoside; Halo-nucleoside; Scaffold and Template. | |||
T71340 | Mizagliflozin sebacate | ||
Mizagliflozin sebacate is a sodium-glucose transporter inhibitor. It is expected to improve postprandial hyperglycemia by suppressing glucose absorption from the intestine with a novel mechanism of action different from... | |||
TNU0174 | 7-Cyano-7-deazaguanosine | ||
Nucleoside Derivatives - 7-Deaza-purine nucleosides;Naturally modified ribo-nucleosides | |||
TNU0173 | 7-(N-Acetylaminomethyl)-7-deazaguanosine | ||
Nucleoside Derivatives –7-Deaza-purine nucleosides; Amino nucleosides | |||
T76616 | (D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH | ||
(D-Ser4, D-Ser(tBu)6, Azagly10)-LHRH, an analogue of luteinizing hormone-releasing hormone (LHRH), plays a pivotal role in reproductive regulation by promoting the secretion of pituitary luteinizing hormone (LH) and foll... | |||
T37388 | Afizagabar | ||
Afizagabar (S44819) is a first-in-class, competitive, and selective antagonist at the GABA-binding site of the α5-GABAAR, with an IC50 of 585 nM for α5β2γ2 and a Ki of 66 nM for α5β3γ2. Afizagabar enhances hippocampal sy... | |||
T78379 | 9-Deazaguanine | Others | |
9-Deazaguanine is a nucleoside analog that exhibits potent inhibitory activity against purine nucleoside phosphorylase (PNP) [1]. | |||
T19148 | 5-Aza-7-deazaguanine | Others | |
5-Aza-7-deazaguanine is a substrate for E. coli purine nucleoside phosphorylase (wild-type/Ser90Ala mutant) in the synthesis of base-modified nucleosides. | |||
T6236L | Ozagrel Sodium | KCT 0809,KCT-0809,Xanbo,KCT0809,Cataclot | |
Ozagrel Sodium is a thromboxane A2 synthase inhibitor. It is used to treat cerebrovascular diseases. | |||
TNU1526 | N2-iso-Butyryl-8-azaguanosine | ||
N2-iso-Butyryl-8-azaguanosine is a Nucleoside Derivative - 8-Modified purine nucleoside. | |||
T77084 | Mezagitamab | ||
Mezagitamab (TAK-079), an IgG1λ anti-CD38 monoclonal antibody, functions by depleting tumor cells that express CD38 through both antibody and complement-dependent cytotoxicity. It shows potential for use in the treatment... | |||
T31406 | Dezaguanine | Dezaguanina,NSC 261726,CI-908,CI 908 | |
Dezaguanine is a novel antipurine antimetabolite with significant activity against transplantable rodent solid tumors, particularly breast adenocarcinoma. | |||
T39673 | Zagociguat | ||
Zagociguat is a soluble guanylate cyclase stimulator that enhances nitric oxide (NO) signaling, resulting in increased production of cyclic guanosine monophosphate. This compound shows promise for investigating non-centr... |
Cat No. | Product Name | Synonyms | Targets |
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TN7185 | 7-Cyano-7-deazaguanine | 7-CN-7-deazaG | Others |
7-Cyano-7-deazaguanine (7-CN-7-deazaG) is a marine derived natural products found in Streptomyces qinglanensis. | |||
T2218 | 8-Azaguanine | Azaguanine-8,SK 1150,NSC-749,SF-337 | Nucleoside Antimetabolite/Analog , Others , Endogenous Metabolite |
8-Azaguanine (SK 1150) is a purine analogue with potential antineoplastic activity. |
Cat No. | Product Name | Species | Expression System |
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TMPY-03117 | Zinc Alpha 2 Glycoprotein/AZGP1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Alpha-2-glycoprotein, also known as AZGP1, belongs to the MHC class I family. It can be detected in body fluids such as serum, sweat, and seminal and breast cyst fluids. It has been shown that alpha-2-glycoprotein can st... |