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Linzagolix

Linzagolix
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Purity:99.68%
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Linzagolix

Catalog No. T27837Cas No. 935283-04-8
Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei Pharmaceutical and ObsEva for the treatment of uterine fibroids, endometriosis, and adenomyosis. As of December 2020, it is under review for approval for uterine fibroids, is in phase III clinical trials for endometriosis, and is in phase II clinical studies for adenomyosis.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
Pack SizePriceAvailabilityQuantity
1 mg$48In Stock
5 mg$97In Stock
10 mg$163In Stock
25 mg$319In Stock
50 mg$578In Stock
1 mL x 10 mM (in DMSO)$117In Stock
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Product Introduction

Bioactivity
Description
Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei Pharmaceutical and ObsEva for the treatment of uterine fibroids, endometriosis, and adenomyosis. As of December 2020, it is under review for approval for uterine fibroids, is in phase III clinical trials for endometriosis, and is in phase II clinical studies for adenomyosis.
Chemical Properties
Molecular Weight508.42
FormulaC22H15F3N2O7S
Cas No.935283-04-8
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year
Solubility Information
DMSO: 55 mg/ml (108.18 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM1.9669 mL9.8344 mL19.6688 mL98.3439 mL
5 mM0.3934 mL1.9669 mL3.9338 mL19.6688 mL
10 mM0.1967 mL0.9834 mL1.9669 mL9.8344 mL
20 mM0.0983 mL0.4917 mL0.9834 mL4.9172 mL
50 mM0.0393 mL0.1967 mL0.3934 mL1.9669 mL
100 mM0.0197 mL0.0983 mL0.1967 mL0.9834 mL

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