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Linzagolix choline

Catalog No. T25742 CAS 1321816-57-2

Linzagolix choline is an orally available non-peptide gonadotropin-releasing hormone (GnRH) antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.

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Linzagolix choline, CAS 1321816-57-2

Pack Size	Availability	Price/USD
1 mg	In stock	$ 195.00
5 mg	In stock	$ 483.00
10 mg	In stock	$ 692.00
25 mg	In stock	$ 1,080.00
50 mg	In stock	$ 1,490.00
100 mg	In stock	$ 1,970.00

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Biological Description

Chemical Properties

Storage & Solubility Information

Description

Linzagolix choline is an orally available non-peptide gonadotropin-releasing hormone (GnRH) antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.

Molecular Weight	611.59
Formula	C27H28F3N3O8S
CAS No.	1321816-57-2

Storage

keep away from direct sunlight

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Kobayashi K, et al. Non-clinical studies indicating lack of interactions between iron/calcium ions and linzagolix, an orally available GnRH antagonist. Xenobiotica. 2022 May;52(5):488-497. 2. de Lange ME, et al. Considerations on implementation of the newest treatment for symptomatic uterine fibroids: Oral GnRH antagonists. Br J Clin Pharmacol. 2024 Feb;90(2):392-405. 3. Donnez J,et al. Evolution of uterine adenomyosis volume during and after GnRH antagonist (linzagolix) treatment: lessons for further clinical trials. Fertil Steril. 2023 Nov;120(5):1071-1073. 4. Tezuka M, et al. Suppression of hypothalamic-pituitary-gonadal function by linzagolix in benign prostatic hyperplasia and polycystic ovary syndrome animal models. Clin Exp Pharmacol Physiol. 2023 Nov;50(11):914-923.

Related Products

Related compounds with same targets

AG 045572 (R)-Elagolix Deslorelin acetate(57773-65-6 free base) Linzagolix Ganirelix Acetate LGnRH-III, lamprey acetate(147859-97-0 free base) GnRH-R antagonist 1 Nafarelin acetate(76932-56-4 free base)

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Linzagolix choline 1321816-57-2 GPCR/G Protein GNRH Receptor inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.