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Search Result

Search Results for " melk "

Targets

MELK MELK

16

Compounds

1

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T11997 MELK-IN-1 Nintedanib Impurity L,MELK inhibitor 17 MELK
MELK-IN-1 (MELK inhibitor 17) is a potent inhibitor of maternal embryonic leucine zipper kinase (MELK),(IC50:3nm;Ki:0.39 nM).
T11996 MELK-8a hydrochloride MELK
MELK-8a hydrochloride is a potent inhibitor of maternal embryonic leucine zipper kinase (MELK, IC50 = 2 nM). 
T1759 OTSSP167 MELK inhibitor,OTS167 MELK
OTSSP167 (OTS167) is an orally available inhibitor of maternal embryonic leucine zipper kinase (MELK) with potential antineoplastic activity.
T35342 MELK-8a Dihydrochloride MELK
MELK-8a Dihydrochloride is a useful organic compound for research related to life sciences and the catalog number is T35342.
T62417 MELK-8a
MELK-8a (NVS-MELK8a) is a potent and selective inhibitor of maternal embryonic leucine elongation kinase (MELK) (IC50: 2 nM). 0.42 μM). Among them, MELK plays an important role in regulating mitosis in cancer cells.
T11725 JNJ-47117096 hydrochloride MELK-T1 hydrochloride Others
JNJ-47117096 hydrochloride is potent and selective MELK inhibitor, with an IC50 of 23 nM, also effectively inhibits Flt3, with an IC50 of 18 nM.
T21559 OTSSP167 hydrochloride MELK
OTSSP167 hydrochloride is a highly potent inhibitor of MELK(IC50 : 0.41 nM).
T4327 Prexasertib dihydrochloride LY2606368 (dihydrochloride),Prexasertib HCl,LY2606368 Apoptosis , Chk , S6 Kinase
Prexasertib dihydrochloride (LY2606368) is an ATP-competitive CHK1 inhibitor (Ki: 0.9 nmol/L). in the cell-free assay, its IC50 values are 8 nM and 9 nM for CHK2 and RSK, respectively.
T4310 Prexasertib LY2606368 Apoptosis , Chk
Prexasertib (LY2606368) is an inhibitor of checkpoint kinase 1 (chk1) with potential antineoplastic activity.
T24152 HTH-01-091 HTH-01091,HTH01-091,HTH 01-091,HTH 01091 Serine/threonin kinase , Pim , MELK , DYRK , CDK , RIP kinase
HTH-01-091 is a potent and selective maternal embryonic leucine zipper kinase (MELK) inhibitor (IC50: 10.5 nM).HTH-01-091 inhibits PIM1/2/3, RIPK2, DYRK3, smMLCK and CLK2. HTH-01-091 can be used to study breast cancer.
T71197 JW-7-25-1
JW-7-25-1 is a potent multi-target inhibitor, acting on MELK, PIK3CA, mTOR, GSK3A and CDK7.
T79582 Antitumor agent-116 MELK
Antitumor Agent-116 (Compound 6C) is an anti-tumor agent that exhibits anti-proliferative properties and induces apoptosis. It demonstrates binding affinity for the MELK receptor [1].
T73867 HTH-01-091 TFA
HTH-01-091 TFA, a potent and selective inhibitor of maternal embryonic leucine zipper kinase (MELK), exhibits an IC50 of 10.5 nM. Besides its primary target, it also inhibits PIM1/2/3, RIPK2, DYRK3, smMLCK, and CLK2, pos...
T82385 FMF-06-098-1 PROTACs
FMF-06-098-1 is a multitargeted depressant capable of promoting the degradation of a wide array of kinases, including AAK1, ABL2, AURKA, AURKB, BUB1B, CDC7, CDK1, CDK12, CDK13, CDK2, CDK4, CDK6, CDK7, CDK9, CHEK1, CSNK1D...
T12237 NMS-P715 Casein Kinase , Kinesin , MELK , MAPK
NMS-P715 is a selective and ATP-competitive MPS1 inhibitor(IC50 of 182 nM).
T16142 MRT199665 Others
MRT199665 is an effective and ATP-competitive, selective MARK/SIK/AMPK inhibitor (IC50s of 2/2/3/2 nM, 10/10 nM, and 110/12/43 nM for MARK1/MARK2/MARK3/MARK14, AMPKα1/AMPKα2, and SIK1/SIK2/SIK3, respectively). MRT199665 ...

Recombinant Proteins

Species：
Human (1)
Expression System：
E. coli (1)
Tag：
N-terminal 10xHis-tagged and C-terminal Myc-tagged (1)
Cat No. Product Name Species Expression System
TMPH-01642 MELK Protein, Human, Recombinant (His & Myc) Human E. coli
Serine/threonine-protein kinase involved in various processes such as cell cycle regulation, self-renewal of stem cells, apoptosis and splicing regulation. Has a broad substrate specificity; phosphorylates BCL2L14, CDC25...
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