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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T21724L | Fas C-Terminal Tripeptide Acetate | Fas C-Terminal Tripeptide Acetate (189109-90-8 free base) | Others , Fatty Acid Synthase |
Fas C-Terminal Tripeptide Acetate shows inhibitory activity of Fas/FAP-1 binding. | |||
T11266L | FAS-IN-1 Tosylate | Fatty Acid Synthase | |
FAS-IN-1 Tosylate is an effective fatty acid synthase inhibitor;Has an IC50 of 10 nM. | |||
T80442 | Fasciculin-II | Fas-2 | |
Fasciculin-II (Fas-2) acts as a potential inhibitor of acetylcholinesterase (AChE) [1]. | |||
T82415 | Fasciculin-I | FAS-I | |
Fasciculin-I, a toxin isolated from mamba venom, exerts its toxicity primarily by inhibiting acetylcholinesterase (AChE). Additionally, it impedes the action of α-neurotoxins on nicotinic acetylcholine receptors and neut... | |||
T11266 | FASN-IN-4 | FAS-IN-1 | Others |
FAS-IN-1 is a potent inhibitor of Fatty acid synthase (FAS) wtih IC50 of 10 nM. | |||
T80584 | Anti-Mouse Fas Ligand Antibody (MFL3) | ||
Anti-Mouse Fas Ligand Antibody is an Armenian hamster-derived IgG inhibitor that targets the mouse Fas Ligand. | |||
T21936 | M50054 | Caspase | |
Apoptosis Inhibitor was a novel inhibitor of programmed cell death associate with caspase-3 inhibition. | |||
T5S0246 | Pseudoprotodioscin | Others , Fatty Acid Synthase | |
1. Pseudoprotodioscin has moderate cytotoxicity. | |||
T8616 | Fasentin | N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide | transporter |
Fasentin (N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide) is an inhibitor of GluT1. | |||
T10549 | Bisindolylmaleimide VIII acetate | Ro 31-7549 acetate,Bis VIII acetate | Apoptosis , PKC |
Bisindolylmaleimide VIII acetate (Ro 31-7549 acetate) is a potent and selective PKC inhibitor (IC50: 158 nM for rat brain PKC). It has IC50s of 53, 195, 163, 213, and 175 nM for PKC-α, PKC-βI, PKC-βII, PKC-γ, PKC-ε, resp... | |||
T39308 | Boc-Asp(OMe)-fluoromethyl ketone | Boc-Asp(OMe)-fluoromethyl ketone,Boc-Asp(OMe)-FMK | Caspase |
Boc-Asp(OMe)-fluoromethyl ketone (Boc-Asp(OMe)-FMK) is a broad range caspase inhibitor. Boc-Asp(OME)-Fluoromethyl Ketone inhibits Fas-mediated phagocytosis and oxidative rupture inhibition, but does not affect the chemot... | |||
T5045 | GSK4112 | 1,1-Dimethylethyl-N-[(4-chlorophenyl)methyl]-N-[(5-nitro-2-thienyl)methyl])glycinate,SR6452 | Autophagy |
GSK4112 (SR6452) is a Rev-erbα agonist with EC50 of 0.4 μM, also is a small molecule chemical probe for the cell biology of the nuclear heme receptor Rev-erbα. | |||
T4276L | Hydroxyfasudil | Hydroxy-Fasudil,HA-1100 | ROCK , PKA |
Hydroxyfasudil (Hydroxy-Fasudil) is a ROCK inhibitor(IC50s of 0.73 and 0.72 μM for ROCK1 and ROCK2, respectively). | |||
TP1029 | Thymalfasin | Thymosin α1 | Others |
Thymalfasin (Thymosin α1) (thymosin-alpha 1) is an immunomodulating agent able to enhance the Thl immune response. | |||
T11267 | FASN-IN-1 | TVB-2460 | Fatty Acid Synthase |
FASN-in-1 is an effective, specific inhibitor of fatty acid synthase (FASN), a compound specifically designed to target and inhibit the activity of the enzyme involved in fatty acid synthesis, potentially disrupting fatt... | |||
T27307 | Fasnall | Fatty Acid Synthase | |
Fasnall is a selective FASN inhibitor that acts through its co-factor binding sites. Fasnall shows potent anti-tumor activity in the MMTV-Neu model of HER2(+) breast cancer, particularly when combined with carboplatin. | |||
T77135 | Tafasitamab | MOR00208,XmAb5574,Tafasitamab-cxix | Apoptosis , Immunology/Inflammation related |
Tafasitamab (XmAb5574) is an FC-modified humanized monoclonal antibody targeting the human B-cell surface antigen CD19 for the study of diffuse large B-cell lymphoma. | |||
T3060 | Fasudil hydrochloride | Fasudil (HA-1077) HCl,HA-1077,Fasudil HCl,HA-1077 hydrochloride,AT-877 | ROCK , Serine/threonin kinase , Calcium Channel , HIV Protease , PKA , PKC , Autophagy |
Fasudil hydrochloride (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Ki of 0.33 μM, 1.0 μM, 9.3 μM and 55 μM, respectively. | |||
T4276 | Hydroxyfasudil Hydrochloride | Hydroxyfasudil (HA-1100) HCl,HA 1100 hydrochloride | ROCK |
Hydroxyfasudil Hydrochloride (HA 1100 hydrochloride) is a ROCK1/2 inhibitor (IC50s: 0.73/0.72 μM). | |||
T2351 | Fasiglifam | TAK875 | GPR |
Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist. |