Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
50 mg | In stock | $ 33.00 | |
100 mg | In stock | $ 47.00 | |
200 mg | In stock | $ 60.00 | |
500 mg | In stock | $ 95.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 47.00 |
Description | Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM. |
Targets&IC50 | CYP2C9:19.3 nM(Ki) |
In vivo | In oocytes expressing URAT1 (IC50 <0.1 μM), Benzbromarone (50 μM) completely inhibited the uptake of uric acid. In rat hepatocytes, Benzbromarone (100 μM) increased mitochondrial size and induced apoptosis in 11% of cells. |
Synonyms | Desuric, Normurat, Urinorm |
Molecular Weight | 424.08 |
Formula | C17H12Br2O3 |
CAS No. | 3562-84-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: 9 mg/mL (21.22 mM)
DMSO: 79 mg/mL (186.3 mM)
H2O: < 1 mg/mL (insoluble or slightly soluble)
You can also refer to dose conversion for different animals. More
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Benzbromarone 3562-84-3 Apoptosis Metabolism Xanthine Oxidase P450 inhibit Desuric Normurat Inhibitor Urinorm inhibitor