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Search Results for " dihydrochloride "

20

Compounds

Cat No. Product Name Synonyms Targets
T11727 JPH203 dihydrochloride KYT-0353 dihydrochloride Others
JPH203 dihydrochloride (KYT-0353 dihydrochloride) is a tyrosine analog, acts as a selective inhibitor of L-type amino acid transporter 1 (LAT1), and is used in cancer research.
T12241 Norbinaltorphimine dihydrochloride nor-BNI dihydrochloride,Nor-BNI dihydrochloride,nor-Binaltorphimine dihydrochloride,Nor-Binaltorphimine dihydrochloride Opioid Receptor
Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.
T7821 DG172 dihydrochloride DG172 (dihydrochloride),DG-172 dihydrochloride PPAR
DG172 dihydrochloride (DG-172 dihydrochloride) is an antagonist of PPARβ/δ(IC50 : 27 nM).
T11345L Lerociclib dihydrochloride G1T38 dihydrochloride CDK
Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 2 nM and 1 nM for CDK6/CyclinD3 and CDK4/CyclinD1, respectively.
T22354 Levocetirizine Dihydrochloride Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride Histamine Receptor
Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydro...
T15374 Ipatasertib dihydrochloride GDC-0068 dihydrochloride,RG-7440 dihydrochloride Akt , PKA
Ipatasertib dihydrochloride (GDC-0068 dihydrochloride) is a highly selective and ATP-competitive inhibitor of pan-Akt (IC50s: 5, 18 and 8 nM for Akt1, Akt2 and Akt3, respectively).
T13675 Elacestrant dihydrochloride RAD1901 dihydrochloride Estrogen/progestogen Receptor
Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM for ERβ, respectively.
T9012 Preq1-Dihydrochloride pre-queuosine1 Dihydrochloride Others
Preq1-Dihydrochloride (pre-queuosine1 Dihydrochloride) is an intermediate of the queuosine pathway, it binds with high affinity to the aptamer of PreQ1 riboswitch, which attenuates protein expression.
T3597 Cutamesine dihydrochloride AGY94806 dihydrochloride,SA4503 (dihydrochloride),SA4503 dihydrochloride Sigma receptor
Cutamesine dihydrochloride (SA4503 dihydrochloride) is a selective σ1 receptor agonist (IC50: 17.4 nM). It shows selectivity for σ1 over σ2 receptors, and inhibits angiotensin II-induced cardiomyocyte hypertrophy in vitr...
T10358 Netarsudil Dihydrochloride AR-13324 Dihydrochloride ROCK
Netarsudil Dihydrochloride (AR-13324 Dihydrochloride) is an inhibitor of Rho-associated protein kinase (ROCK) and norepinephrine transporter (NET) with effective in intraocular pressure (IOP) reduction.
T4676 Sardomozide dihydrochloride CGP 48664 dihydrochloride,Sardomozide dihydrochloride Others
Sardomozide dihydrochloride (CGP 48664 dihydrochloride) is an inhibitor of S-adenosylmethionine decarboxylase (SAMDC, IC50 = 5 nM).
T9172 Simufilam dihydrochloride PTI-125 dihydrochloride Others
Simufilam dihydrochloride (PTI-125 dihydrochloride) is a low toxicity, orally active filamin A (FLNA) activator, which can be used for the research of Alzheimer's disease. Simufilam dihydrochloride preferentially binds a...
T12374 PAβN dihydrochloride MC-207,110 dihydrochloride,Phe-Arg-β-naphthylamide dihydrochloride Others , Antibacterial
PAβN dihydrochloride (MC-207,110 dihydrochloride) is an inhibitor of efflux pump.
T4467 UAMC00039 dihydrochloride UAMC 00039 dihydrochloride Proteasome
UAMC00039 dihydrochloride is a potent, reversible and competitive dipeptidyl peptidase II inhibitor with an IC50 of 0.48 nM.
T5135 Flupentixol dihydrochloride Fupentixol Dihydrochloride,Flupenthixol dihydrochloride,(E/Z)-Flupentixol Dihydrochloride Dopamine Receptor
Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.
T7153 Vanoxerine dihydrochloride GBR-12909 dihydrochloride,I893 dihydrochloride Dopamine Receptor
Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)
T19069 TMB dihydrochloride BM blue dihydrochloride,Sure Blue TMB dihydrochloride,3,3',5,5'-Tetramethylbenzidine dihydrochloride Others
TMB dihydrochloride (Sure Blue TMB dihydrochloride) is an enzyme-linked immunosorbent assays (ELISA) and an excellent colorimetric substrate for the detection of horseradish peroxidase (HRP)-labeled probes used in staini...
T11011 Dexpramipexole dihydrochloride KNS-760704 dihydrochloride,R-(+)-Pramipexole dihydrochloride,(R)-Pramipexole dihydrochloride Dopamine Receptor
Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine agonist.
T4754 Pyridoxylamine dihydrochloride Pyridorin,Pyridoxamine dihydrochloride Others , Endogenous Metabolite
Pyridoxylamine dihydrochloride (Pyridorin) is a hydrochloride salt of one form of vitamin B6.
T5495 Decloxizine dihydrochloride UCB 1402 dihydrochloride Histamine Receptor
Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.

Compounds

JPH203 dihydrochloride
T11727
Synonym: KYT-0353 dihydrochloride
Target: Others
Norbinaltorphimine dihydrochloride
T12241
Synonym: nor-BNI dihydrochloride,Nor-BNI dihydrochloride,nor-Binaltorphimine dihydrochloride,Nor-Binaltorphimine dihydrochloride
Target: Opioid Receptor
DG172 dihydrochloride
T7821
Synonym: DG172 (dihydrochloride),DG-172 dihydrochloride
Target: PPAR
Lerociclib dihydrochloride
T11345L
Synonym: G1T38 dihydrochloride
Target: CDK
Levocetirizine Dihydrochloride
T22354
Synonym: Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride
Target: Histamine Receptor
Ipatasertib dihydrochloride
T15374
Synonym: GDC-0068 dihydrochloride,RG-7440 dihydrochloride
Target: Akt, PKA
Elacestrant dihydrochloride
T13675
Synonym: RAD1901 dihydrochloride
Target: Estrogen/progestogen Receptor
Preq1-Dihydrochloride
T9012
Synonym: pre-queuosine1 Dihydrochloride
Target: Others
Cutamesine dihydrochloride
T3597
Synonym: AGY94806 dihydrochloride,SA4503 (dihydrochloride),SA4503 dihydrochloride
Target: Sigma receptor
Netarsudil Dihydrochloride
T10358
Synonym: AR-13324 Dihydrochloride
Target: ROCK
Sardomozide dihydrochloride
T4676
Synonym: CGP 48664 dihydrochloride,Sardomozide dihydrochloride
Target: Others
Simufilam dihydrochloride
T9172
Synonym: PTI-125 dihydrochloride
Target: Others
PAβN dihydrochloride
T12374
Synonym: MC-207,110 dihydrochloride,Phe-Arg-β-naphthylamide dihydrochloride
Target: Others, Antibacterial
UAMC00039 dihydrochloride
T4467
Synonym: UAMC 00039 dihydrochloride
Target: Proteasome
Flupentixol dihydrochloride
T5135
Synonym: Fupentixol Dihydrochloride,Flupenthixol dihydrochloride,(E/Z)-Flupentixol Dihydrochloride
Target: Dopamine Receptor
Vanoxerine dihydrochloride
T7153
Synonym: GBR-12909 dihydrochloride,I893 dihydrochloride
Target: Dopamine Receptor
TMB dihydrochloride
T19069
Synonym: BM blue dihydrochloride,Sure Blue TMB dihydrochloride,3,3',5,5'-Tetramethylbenzidine dihydrochloride
Target: Others
Dexpramipexole dihydrochloride
T11011
Synonym: KNS-760704 dihydrochloride,R-(+)-Pramipexole dihydrochloride,(R)-Pramipexole dihydrochloride
Target: Dopamine Receptor
Pyridoxylamine dihydrochloride
T4754
Synonym: Pyridorin,Pyridoxamine dihydrochloride
Target: Others, Endogenous Metabolite
Decloxizine dihydrochloride
T5495
Synonym: UCB 1402 dihydrochloride
Target: Histamine Receptor
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TargetMol