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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T11727 | JPH203 dihydrochloride | KYT-0353 dihydrochloride | Others |
JPH203 dihydrochloride (KYT-0353 dihydrochloride) is a tyrosine analog, acts as a selective inhibitor of L-type amino acid transporter 1 (LAT1), and is used in cancer research. | |||
T12241 | Norbinaltorphimine dihydrochloride | nor-BNI dihydrochloride,Nor-BNI dihydrochloride,nor-Binaltorphimine dihydrochloride,Nor-Binaltorphimine dihydrochloride | Opioid Receptor |
Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice. | |||
T7821 | DG172 dihydrochloride | DG172 (dihydrochloride),DG-172 dihydrochloride | PPAR |
DG172 dihydrochloride (DG-172 dihydrochloride) is an antagonist of PPARβ/δ(IC50 : 27 nM). | |||
T11345L | Lerociclib dihydrochloride | G1T38 dihydrochloride | CDK |
Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 2 nM and 1 nM for CDK6/CyclinD3 and CDK4/CyclinD1, respectively. | |||
T22354 | Levocetirizine Dihydrochloride | Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride | Histamine Receptor |
Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydro... | |||
T15374 | Ipatasertib dihydrochloride | GDC-0068 dihydrochloride,RG-7440 dihydrochloride | Akt , PKA |
Ipatasertib dihydrochloride (GDC-0068 dihydrochloride) is a highly selective and ATP-competitive inhibitor of pan-Akt (IC50s: 5, 18 and 8 nM for Akt1, Akt2 and Akt3, respectively). | |||
T13675 | Elacestrant dihydrochloride | RAD1901 dihydrochloride | Estrogen/progestogen Receptor |
Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM for ERβ, respectively. | |||
T9012 | Preq1-Dihydrochloride | pre-queuosine1 Dihydrochloride | Others |
Preq1-Dihydrochloride (pre-queuosine1 Dihydrochloride) is an intermediate of the queuosine pathway, it binds with high affinity to the aptamer of PreQ1 riboswitch, which attenuates protein expression. | |||
T3597 | Cutamesine dihydrochloride | AGY94806 dihydrochloride,SA4503 (dihydrochloride),SA4503 dihydrochloride | Sigma receptor |
Cutamesine dihydrochloride (SA4503 dihydrochloride) is a selective σ1 receptor agonist (IC50: 17.4 nM). It shows selectivity for σ1 over σ2 receptors, and inhibits angiotensin II-induced cardiomyocyte hypertrophy in vitr... | |||
T10358 | Netarsudil Dihydrochloride | AR-13324 Dihydrochloride | ROCK |
Netarsudil Dihydrochloride (AR-13324 Dihydrochloride) is an inhibitor of Rho-associated protein kinase (ROCK) and norepinephrine transporter (NET) with effective in intraocular pressure (IOP) reduction. | |||
T4676 | Sardomozide dihydrochloride | CGP 48664 dihydrochloride,Sardomozide dihydrochloride | Others |
Sardomozide dihydrochloride (CGP 48664 dihydrochloride) is an inhibitor of S-adenosylmethionine decarboxylase (SAMDC, IC50 = 5 nM). | |||
T9172 | Simufilam dihydrochloride | PTI-125 dihydrochloride | Others |
Simufilam dihydrochloride (PTI-125 dihydrochloride) is a low toxicity, orally active filamin A (FLNA) activator, which can be used for the research of Alzheimer's disease. Simufilam dihydrochloride preferentially binds a... | |||
T12374 | PAβN dihydrochloride | MC-207,110 dihydrochloride,Phe-Arg-β-naphthylamide dihydrochloride | Others , Antibacterial |
PAβN dihydrochloride (MC-207,110 dihydrochloride) is an inhibitor of efflux pump. | |||
T4467 | UAMC00039 dihydrochloride | UAMC 00039 dihydrochloride | Proteasome |
UAMC00039 dihydrochloride is a potent, reversible and competitive dipeptidyl peptidase II inhibitor with an IC50 of 0.48 nM. | |||
T5135 | Flupentixol dihydrochloride | Fupentixol Dihydrochloride,Flupenthixol dihydrochloride,(E/Z)-Flupentixol Dihydrochloride | Dopamine Receptor |
Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders. | |||
T7153 | Vanoxerine dihydrochloride | GBR-12909 dihydrochloride,I893 dihydrochloride | Dopamine Receptor |
Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM) | |||
T19069 | TMB dihydrochloride | BM blue dihydrochloride,Sure Blue TMB dihydrochloride,3,3',5,5'-Tetramethylbenzidine dihydrochloride | Others |
TMB dihydrochloride (Sure Blue TMB dihydrochloride) is an enzyme-linked immunosorbent assays (ELISA) and an excellent colorimetric substrate for the detection of horseradish peroxidase (HRP)-labeled probes used in staini... | |||
T11011 | Dexpramipexole dihydrochloride | KNS-760704 dihydrochloride,R-(+)-Pramipexole dihydrochloride,(R)-Pramipexole dihydrochloride | Dopamine Receptor |
Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine agonist. | |||
T4754 | Pyridoxylamine dihydrochloride | Pyridorin,Pyridoxamine dihydrochloride | Others , Endogenous Metabolite |
Pyridoxylamine dihydrochloride (Pyridorin) is a hydrochloride salt of one form of vitamin B6. | |||
T5495 | Decloxizine dihydrochloride | UCB 1402 dihydrochloride | Histamine Receptor |
Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist. |