containing — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
TP1491	Kv3, Channel Containing Protein 567-585
	Kv3 channel protein is expressed by parvalbumin (PV)-containing pallidal neurons.Kv3, Channel Containing Protein (567-585) corresponds to amino acids 567 to 585 fragment of the Kv3.1b channel containing protein.
TP2292	Survivin (baculoviral IAP repeat-containing protein 5) (21-28)		Others
	Survivin (baculoviral inhibitor of apoptosis IAP repeat-containing protein-5) is a member of the IAP gene family, which has been implicated in both inhibitions of apoptosis and mitosis regulation1. Survivin is one of the...		Others
T39668	Methyl propyl disulfide		Others
	Methyl propyl disulfide is a natural compound containing volatile sulfur produced in garlic and onions. Methyl propyl disulfide displays an anticaner effect.		Others
T7877	Thiacetazone	Diazam,Thioacetazone,Neustab,Neotibil	Others , Antibacterial , Antibiotic
	Thiacetazone (Diazam) is a thiosemicarbazone that thioacetazone treatment of pulmonary tuberculosis		Others , Antibacterial , Antibiotic
T9552	BAZ1A-IN-1		Epigenetic Reader Domain
	BAZ1A-IN-1 is a potent BAZ1A inhibitor with the KD value of 0.52 μM for the BAZ1A bromodomain. BAZ1A-IN-1 shows good anti-survival activity against cancer cell lines with high BAZ1A expression, but weak or no activity ag...		Epigenetic Reader Domain
T6593	ML324		Histone Demethylase , Others , HSV
	ML324(IC50=920 nM) is a specific inhibitor of jumonji histone demethylase (JMJD2).		Histone Demethylase , Others , HSV
TP1088	N-Acetylcarnosine	N-Acetyl-L-carnosine	Others
	N-Acetylcarnosine (N-Acetyl-L-carnosine) is thought to be able to combat some of the effects of oxidative stress as it has anti-oxidant properties.		Others
T6830	Epoxomicin	BU-4061T,BU-4061T,Aids010837	Apoptosis , Proteasome
	Epoxomicin (BU-4061T,Aids010837) is a selective proteasome inhibitor with anti-inflammatory activity, inhibits primarily the CH-L activity of the 20S proteasome, while T-L and PGPH catalytic activities are also inhibited...		Apoptosis , Proteasome
T19081	1,3-Dithiane	1,3-Dithian,M-DITHIANE,1,3-Dithiacyclohexane	Anti-infection , Endogenous Metabolite , Antibacterial
	1,3-Dithiane (1,3-Dithian) is a protected formaldehyde anion equivalent that could serve as a useful labeled synthon. 1,3-Dithiane is also a sulfur-containing Maillard reaction products found in boiled beef extracts.		Anti-infection , Endogenous Metabolite , Antibacterial
T6859	I-BRD9	GSK602	Epigenetic Reader Domain
	I-BRD9 (GSK602) is the first selective cellular inhibitor for BRD9 with pIC50 of 7.3.		Epigenetic Reader Domain
T7165	Basmisanil	RG1662,RO5186582	GABA Receptor
	Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the treatment of cognitive impairments associated with Down syndro...		GABA Receptor
T2167	Lutidinic acid	2,4-Pyridinedicarboxylic acid,2,4-Dicarboxypyridine,2, 4-PDCA,2,4-PDCA	Histone Methyltransferase
	lutidinic acid (2,4-Dicarboxypyridine) is an in vitro and in cell inhibitor, as well as a known inhibitor of the histone lysine demethylases.		Histone Methyltransferase
T4583	PFI-2 hydrochloride	(R)-PFI-2 hydrochloride,PFI-2 HCl	Histone Methyltransferase
	PFI-2 hydrochloride ((R)-PFI-2 hydrochloride) is a potent, highly selective, and cell-active inhibitor of the methyltransferase activity of SETD7 (IC50: 2 nM), 500 fold active than (S)-PFI-2.		Histone Methyltransferase
T1987	PFI-2	PFI2,PFI 2,(R)-PFI-2	Histone Methyltransferase
	PFI-2 is an effective, specific and cell-active lysine methyltransferase SETD7 inhibitor (Ki/IC50: 0.33/2 nM), 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.		Histone Methyltransferase
T24807	S-Methylglutathione	S-Methyl glutathione,Glutathione S-methyl ester,Glutathione ester
	S-methyl glutathione is an inhibitor of methionine-containing peptide and glyoxylate.
T8994	ML-226	ML226,ML-226	MAGL
	ML226 is a α/β hydrolase domain-containing protein 11 (ABHD11) inhibitor that inhibits ABHD11 in vitro and in situ.		MAGL
T5S2205	Sibiricaxanthone B		Others
	Sibiricaxanthone B is an oxygen-containing xanthone isolated from Polygala tenuifolia.		Others
T29022	TU-2100	Azeloyl diethyl salicylate,Azasal-2100,TU 2100,TU2100	Others
	TU-2100 is an ethyl salicylate-containing compound with potential anti-acne effects for the study of acne.		Others
T10877	CPDA		Phosphatase
	CPDA is a new potent inhibitor of SH2 domain-containing inositol phosphatase 2 (SHIP2).		Phosphatase
T2187	Orthanilamide	O-Aminobenzenesulfonamide,Benzenesulfonamide,O-Sulfanilamide	Carbonic Anhydrase , Autophagy
	Orthanilamide (Orthanilamide) is a molecule containing the sulfonamide functional group attached to an aniline.		Carbonic Anhydrase , Autophagy