20
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T15090 | Decoglurant | RO4995819 | GluR |
Decoglurant (RO4995819) is a negative allosteric modulator of mGluR2 and mGluR3 and it also is developed as an antidepressant. | |||
T13318 | VU0650786 | GluR | |
VU0650786 is a selective and potent CNS penetrant negative allosteric modulator of metabotropic glutamate receptor subtype 3 (mGlu3 NAM) (IC50: 392 nM), with antidepressant and anxiolytic activity in rodents. | |||
T22027 | AH-7614 | AH 7614 | GPR |
AH-7614 (AH 7614) is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist. | |||
T9699 | TAK-615 | LPA Receptor | |
TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of LPA1 receptors. | |||
TN6660 | 2-Ethylhexyl trans-4-methoxycinnamate | Others | |
2-Ethylhexyl trans-4-methoxycinnamate is a sunscreen agent. | |||
T66390 | 4-(4-Amino-3-fluorophenoxy)-N-methylpicolinamide | ||
4-(4-Amino-3-fluorophenoxy)-N-methylpicolinamide is an aromatic enigma that is is a metabolite of the antitumor drug rafenil. | |||
T9124 | Laninamivir octanoate | CS-8958 | Influenza Virus |
Laninamivir octanoate (CS-8958) is a long acting influenza neuraminidase (NA) inhibitor which shows superior anti-influenza virus activity. | |||
TN5922 | 3,4-Dimethoxycinnamyl alcohol | (E)-3-(3,4-dimethoxyphenyl)prop-2-en-1-ol | Others |
3,4-Dimethoxycinnamyl alcohol ((E)-3-(3,4-dimethoxyphenyl)prop-2-en-1-ol) shows significant antimicrobial and cytotoxic activities. | |||
TN1352 | N-(3-Methoxybenzyl-(9z,12z)-octadecadienamide | (9Z,12Z)-N-(3-Methoxybenzyl)octadeca-9,12-dienamide,n-3-methoxybenzyl-9z-12z-octadecadienamide | Drug Metabolite |
N-(3-Methoxybenzyl-(9z,12z)-octadecadienamide ((9Z,12Z)-N-(3-Methoxybenzyl)octadeca-9,12-dienamide) is a Macamide impurity that may be used in the study of metabolic diseases. | |||
T9323 | 4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide | 4-Amino-6-(trifluoromethyl)benzene-1,3-d,2,4-Disulfamyl-5-trifluoromethylaniline,2-amino-4-trifluoromethyl-1,5-benzendisulfonamide | Carbonic Anhydrase |
4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) is a carbonic anhydrase inhibitor, used as a potential anti-tumor and antiglaucoma drug. | |||
T39043 | Tenofovir amibufenamide | HS-10234 | HBV |
Tenofovir amibufenamide (HS-10234) (HS-10234) is a Tenofovir prodrug, an antiviral compound with oral activity. Tenofovir amibufenamide inhibits hepatitis B virus (HBV) and can be used in chronic hepatitis B (CHB) studie... | |||
TP1907L1 | Dynamin inhibitory peptide, myristoylated acetate | Dynamin inhibitory peptide, myristoylated acetate(251634-22-7 free base) | Dynamin |
Dynamin inhibitory peptide, myristoylated acetate is a DynaMin inhibitor to interfere with the binding of amphiphysin with dynamin. DynaMin inhibitory peptide, myristoylated TFA is a membrane-permeant form of the peptide... | |||
T12343 | Benzquinamide | BZQ,P2647,Benzoquinamide | Adrenergic Receptor |
Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer drugs in multidrug-resistant cells.The Ki values of Benzqui... | |||
T21798L | Dynamin inhibitory peptide Acetate | Dynamin inhibitory peptide Acetate(251634-21-6 Free base) | GTPase |
Dynamin inhibitory peptide Acetate is a peptide with the sequence Gln-Val-Pro-Ser-Arg-Pro-Asn-Arg-Ala-Pro that inhibit the GTPase dynamin. | |||
T83632 | Usenamine A | ||
Usenamine A is a small molecule compound derived from lichen Usnea longissima that has antitumor activity and can be used in the study of tumors. | |||
T50062 | 2,5-dichloro-4-(difluoromethoxy)-N,N-dimethylbenzene-1-sulfonamide | PDE | |
2,5-dichloro-4-(difluoromethoxy)-N,N-dimethylbenzene-1-sulfonamide is a PDE inhibitor. | |||
T50061 | [4-(4-phenylpiperazin-1-yl)oxan-4-yl]methanamine | Others | |
[4-(4-phenylpiperazin-1-yl)oxan-4-yl]methanamine is a piperazine derivative that is a partial agonist at serotonin and dopamine receptors, making it a candidate for the treatment of psychiatric disorders such as depressi... | |||
T9256 | N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine | Serine/threonin kinase , PKC | |
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine is a novel 2,6-naphthyridine identified by high throughput screen (HTS) as a dual protein kinase C/D (PKC/PKD) inhibitor[1]. | |||
T5881 | Fluazinam | Antifungal | |
Fluazinam is a pyridinamine fungicide with a broad spectrum of antifungal activity and had a strong inhibition effect on mycelial growth of S. sclerotiorum populations. | |||
T63290 | (R,1R)-Tenofovir amibufenamide | (R,1R)-HS-10234 | Antiviral |
(R,1R)-Tenofovir amibufenamide ((R,1R)-HS-10234) can be used as a Tenofovir prodrug, which can be taken orally and has antiviral activity. Tynofovir is a nucleotide reverse transcriptase inhibitor. |